Synthesis, molecular docking, and anti-inflammatory evaluation of novel 4-(benzo[d][1,3]dioxol-5-yloxy)-N,N-2-yn-1-amine derivatives as potent cysteinyl leukotriene receptor (CysLT2) antagonists

Cysteinyl leukotrienes (CysLTs), derived from arachidonic acid, play a crucial role in regulating inflammation. We synthesized a novel series of CysLT2 antagonists containing the benzo[d][1,3]dioxole moiety using a synthetic strategy based on the Mannich reaction, resulting in the formation of 4-(be...

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Bibliographic Details
Main Authors: Areej M. Jaber, Mohammed M. Al-Mahadeen, Belal O. Al-Najjar, Raed A. Al-Qawasmeh
Format: Article
Language:English
Published: Pensoft Publishers 2025-02-01
Series:Pharmacia
Online Access:https://pharmacia.pensoft.net/article/143171/download/pdf/
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