Organocatalyzed asymmetric [2+2] cycloaddition of saccharin-derived endocyclic ketimines and allenoates for the synthesis of fused azetidines

We report a novel enantioselective [2 + 2] cycloaddition of allenoate and endocyclic ketimine derived from saccharin, catalyzed by a chiral tertiary amine. The methodology enables the synthesis of fused tricyclic azetidines with a quaternary stereogenic center, exhibiting high enantioselectivity and...

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Bibliographic Details
Main Authors: Xinyu Liu, Yunfeng Zhang, Luning Zhou, Dehai Li, De Wang
Format: Article
Language:English
Published: Elsevier 2025-06-01
Series:Tetrahedron Chem
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Online Access:http://www.sciencedirect.com/science/article/pii/S2666951X25000154
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