Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis

Colorectal cancer (CRC) is a major global health issue due to its aggressiveness and high mortality rates. While curcumin, the bioactive compound from turmeric (Curcuma longa L.), exhibits anticancer properties, its low water solubility limits therapeutic potential. The present study developed a nov...

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Main Authors: Atthapan Morchang, Keerakarn Somsuan, Artitaya Rongjumnong, Churat Weeraphan, Sasivimon Pramual, Theetat Ruangjaroon, Daranee Chokchaichamnankit, Wuttichai Jaidee, Phateep Hankittichai, Chanatip Pramvichai, Rawiwan Charoensup, Arunothai Wanta, Chantragan Srisomsap, Jisnuson Svasti, Siripat Aluksanasuwan
Format: Article
Language:English
Published: Elsevier 2025-06-01
Series:Carbohydrate Polymer Technologies and Applications
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Online Access:http://www.sciencedirect.com/science/article/pii/S2666893925001148
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author Atthapan Morchang
Keerakarn Somsuan
Artitaya Rongjumnong
Churat Weeraphan
Sasivimon Pramual
Theetat Ruangjaroon
Daranee Chokchaichamnankit
Wuttichai Jaidee
Phateep Hankittichai
Chanatip Pramvichai
Rawiwan Charoensup
Arunothai Wanta
Chantragan Srisomsap
Jisnuson Svasti
Siripat Aluksanasuwan
author_facet Atthapan Morchang
Keerakarn Somsuan
Artitaya Rongjumnong
Churat Weeraphan
Sasivimon Pramual
Theetat Ruangjaroon
Daranee Chokchaichamnankit
Wuttichai Jaidee
Phateep Hankittichai
Chanatip Pramvichai
Rawiwan Charoensup
Arunothai Wanta
Chantragan Srisomsap
Jisnuson Svasti
Siripat Aluksanasuwan
author_sort Atthapan Morchang
collection DOAJ
description Colorectal cancer (CRC) is a major global health issue due to its aggressiveness and high mortality rates. While curcumin, the bioactive compound from turmeric (Curcuma longa L.), exhibits anticancer properties, its low water solubility limits therapeutic potential. The present study developed a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin (CUR-A-Poly-β-CD) inclusion complex to enhance solubility and evaluated its anticancer potential in CRC cell lines. The complex exhibited a zeta potential of -22.9 ± 1.1 mV, a particle size of 496.8 ± 1.9 nm, a solubility of 13.6 mg/L, and a pH of 4.5. CUR-A-Poly-β-CD was non-toxic to normal colon cells (CCD-841 CoN) but significantly reduced the viability of CRC cell lines HT-29, SW-48, and SW-480, with SW-480 cells being the most responsive. CUR-A-Poly-β-CD induced apoptosis and inhibited proliferation, clonogenicity, and migration of SW-480 cells. Proteomic analysis identified 105 altered proteins in SW-480 cells treated with CUR-A-Poly-β-CD, primarily involved in cell growth and ribosome biogenesis pathways. Western blot analysis confirmed increased levels of ribosomal proteins RPL13a and RPS3. In conclusion, the CUR-A-Poly-β-CD inclusion complex demonstrates anticancer effects against CRC by modulating ribosome biogenesis. These findings suggest its potential as a therapeutic approach to improve the effectiveness of CRC treatments.
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spelling doaj-art-e76c28402271471884574554604fee5d2025-08-20T03:20:58ZengElsevierCarbohydrate Polymer Technologies and Applications2666-89392025-06-011010077510.1016/j.carpta.2025.100775Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesisAtthapan Morchang0Keerakarn Somsuan1Artitaya Rongjumnong2Churat Weeraphan3Sasivimon Pramual4Theetat Ruangjaroon5Daranee Chokchaichamnankit6Wuttichai Jaidee7Phateep Hankittichai8Chanatip Pramvichai9Rawiwan Charoensup10Arunothai Wanta11Chantragan Srisomsap12Jisnuson Svasti13Siripat Aluksanasuwan14School of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandSchool of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandCancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandMedicinal Plants Innovation Center of Mae Fah Luang University, Chiang Rai 57100, ThailandSchool of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandSchool of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandMedicinal Plants Innovation Center of Mae Fah Luang University, Chiang Rai 57100, Thailand; School of Integrative Medicine, Mae Fah Luang University, Chiang Rai 57100, ThailandSchool of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandLaboratory of Biochemistry, Chulabhorn Research Institute, Bangkok 10210, ThailandSchool of Medicine, Mae Fah Luang University, Chiang Rai 57100, Thailand; Cancer and Immunology Research Unit (CIRU), Mae Fah Luang University, Chiang Rai 57100, Thailand; Corresponding author: School of Medicine, Mae Fah Luang University, 333 Moo 1, Thasud, Muang, Chiang Rai 57100, Thailand.Colorectal cancer (CRC) is a major global health issue due to its aggressiveness and high mortality rates. While curcumin, the bioactive compound from turmeric (Curcuma longa L.), exhibits anticancer properties, its low water solubility limits therapeutic potential. The present study developed a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin (CUR-A-Poly-β-CD) inclusion complex to enhance solubility and evaluated its anticancer potential in CRC cell lines. The complex exhibited a zeta potential of -22.9 ± 1.1 mV, a particle size of 496.8 ± 1.9 nm, a solubility of 13.6 mg/L, and a pH of 4.5. CUR-A-Poly-β-CD was non-toxic to normal colon cells (CCD-841 CoN) but significantly reduced the viability of CRC cell lines HT-29, SW-48, and SW-480, with SW-480 cells being the most responsive. CUR-A-Poly-β-CD induced apoptosis and inhibited proliferation, clonogenicity, and migration of SW-480 cells. Proteomic analysis identified 105 altered proteins in SW-480 cells treated with CUR-A-Poly-β-CD, primarily involved in cell growth and ribosome biogenesis pathways. Western blot analysis confirmed increased levels of ribosomal proteins RPL13a and RPS3. In conclusion, the CUR-A-Poly-β-CD inclusion complex demonstrates anticancer effects against CRC by modulating ribosome biogenesis. These findings suggest its potential as a therapeutic approach to improve the effectiveness of CRC treatments.http://www.sciencedirect.com/science/article/pii/S2666893925001148CurcuminCyclodextrinsColorectal cancerProteomicsRibosome biogenesis
spellingShingle Atthapan Morchang
Keerakarn Somsuan
Artitaya Rongjumnong
Churat Weeraphan
Sasivimon Pramual
Theetat Ruangjaroon
Daranee Chokchaichamnankit
Wuttichai Jaidee
Phateep Hankittichai
Chanatip Pramvichai
Rawiwan Charoensup
Arunothai Wanta
Chantragan Srisomsap
Jisnuson Svasti
Siripat Aluksanasuwan
Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
Carbohydrate Polymer Technologies and Applications
Curcumin
Cyclodextrins
Colorectal cancer
Proteomics
Ribosome biogenesis
title Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
title_full Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
title_fullStr Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
title_full_unstemmed Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
title_short Proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin-ascorbic acid-polysaccharide-β-cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
title_sort proteomic analysis reveals a potential anticancer mechanism for a novel effervescent curcumin ascorbic acid polysaccharide β cyclodextrin inclusion complex towards colorectal cancer cells through modulation of ribosome biogenesis
topic Curcumin
Cyclodextrins
Colorectal cancer
Proteomics
Ribosome biogenesis
url http://www.sciencedirect.com/science/article/pii/S2666893925001148
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