Discovery of compound 1105486 as a selective inhibitor of B4GALT1: potential for pancreatic cancer therapy

Targeting aberrant β-1,4-galactosyltransferase 1 (B4GALT1) activity represents an unexplored therapeutic avenue for pancreatic ductal adenocarcinoma (PDAC). Guided by a concise active-learning structure-based workflow, we rapidly triaged 22.6 million compounds and singled out 1105486 for experimenta...

Full description

Saved in:
Bibliographic Details
Main Authors: Xu Yunyun, Mou Yiping
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-08-01
Series:Frontiers in Chemistry
Subjects:
Online Access:https://www.frontiersin.org/articles/10.3389/fchem.2025.1651402/full
Tags: Add Tag
No Tags, Be the first to tag this record!