Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury

Abstract Background Bone marrow mesenchymal stem cells (BMSCs) and their secreted exosomes have been shown to possess therapeutic potential in various diseases, including diabetic retinopathy (DR). Retinal microvascular endothelial cell (RMEC) injury is a key factor in DR, and understanding the unde...

Full description

Saved in:
Bibliographic Details
Main Authors: Chao Niu, Daoquan Dong, Longjiang Cui, Yingli Dong, Wei Wang
Format: Article
Language:English
Published: BMC 2025-06-01
Series:Diabetology & Metabolic Syndrome
Subjects:
Online Access:https://doi.org/10.1186/s13098-025-01804-7
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849685901741916160
author Chao Niu
Daoquan Dong
Longjiang Cui
Yingli Dong
Wei Wang
author_facet Chao Niu
Daoquan Dong
Longjiang Cui
Yingli Dong
Wei Wang
author_sort Chao Niu
collection DOAJ
description Abstract Background Bone marrow mesenchymal stem cells (BMSCs) and their secreted exosomes have been shown to possess therapeutic potential in various diseases, including diabetic retinopathy (DR). Retinal microvascular endothelial cell (RMEC) injury is a key factor in DR, and understanding the underlying molecular mechanisms is crucial for the treatment of DR. The study investigated the role of MSC-derived exosomes in RMEC injury and the underlying mechanism. Methods Human retinal microvascular endothelial cells (HRMECs) were exposed to high glucose (HG) to establish an in vitro DR model. Exosomes were isolated from BMSCs using differential centrifugation and co-incubated with HRMECs for functional studies. mRNA expression of ataxin 2 like (ATXN2L), methyltransferase-like 3 (METTL3), and forkhead box L1 (FOXL1) was assessed by quantitative real-time polymerase chain reaction. Protein expression was evaluated by western blotting. Cell viability was measured with a cell counting kit-8 assay, and pro-inflammatory cytokines (TNF-α, IL-1β, and IL-6) were analyzed by enzyme-linked immunosorbent assays. Apoptosis was analyzed through flow cytometry. MDA levels, GSH-Px activity, and ROS levels were determined by colorimetric methods and fluorescence microscopy, respectively. The association of METTL3 with ATXN2L and FOXL1 was investigated using a dual-luciferase reporter assay and RNA immunoprecipitation assay. Results HG treatment increased the secretion of pro-inflammatory factors, apoptosis rate, and oxidative stress in HRMECs. BMSC-derived exosomes inhibited inflammation, apoptosis and oxidative stress in HRMECs by transferring FOXL1 into HRMECs. FOXL1 functioned as an RNA-binding protein of METTL3, which stabilized ATXN2L mRNA expression through m6A methylation in HRMECs. ATXN2L expression was reduced in DR patients’ serum and HG-treated HRMECs. Overexpression of ATXN2L mitigated the high glucose-induced inflammation, apoptosis, and oxidative stress in HRMECs. Conclusion Exosomal FOXL1 from BMSCs stabilized METTL3 to increase ATXN2L expression, thus offering a protective effect against high glucose-induced injury in HRMECs. This finding holds clinical significance for the development of targeted therapies for DR.
format Article
id doaj-art-d2d221322bdb45d7be8133d033f6d872
institution DOAJ
issn 1758-5996
language English
publishDate 2025-06-01
publisher BMC
record_format Article
series Diabetology & Metabolic Syndrome
spelling doaj-art-d2d221322bdb45d7be8133d033f6d8722025-08-20T03:22:54ZengBMCDiabetology & Metabolic Syndrome1758-59962025-06-0117111310.1186/s13098-025-01804-7Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injuryChao Niu0Daoquan Dong1Longjiang Cui2Yingli Dong3Wei Wang4Department of Ophthalmology, Henan Provincial People’s HospitalDepartment of Ophthalmology, Henan Provincial People’s HospitalDepartment of Ophthalmology, Henan Provincial People’s HospitalDepartment of Ophthalmology, Henan Provincial People’s HospitalDepartment of Oncology, Henan Provincial People’s HospitalAbstract Background Bone marrow mesenchymal stem cells (BMSCs) and their secreted exosomes have been shown to possess therapeutic potential in various diseases, including diabetic retinopathy (DR). Retinal microvascular endothelial cell (RMEC) injury is a key factor in DR, and understanding the underlying molecular mechanisms is crucial for the treatment of DR. The study investigated the role of MSC-derived exosomes in RMEC injury and the underlying mechanism. Methods Human retinal microvascular endothelial cells (HRMECs) were exposed to high glucose (HG) to establish an in vitro DR model. Exosomes were isolated from BMSCs using differential centrifugation and co-incubated with HRMECs for functional studies. mRNA expression of ataxin 2 like (ATXN2L), methyltransferase-like 3 (METTL3), and forkhead box L1 (FOXL1) was assessed by quantitative real-time polymerase chain reaction. Protein expression was evaluated by western blotting. Cell viability was measured with a cell counting kit-8 assay, and pro-inflammatory cytokines (TNF-α, IL-1β, and IL-6) were analyzed by enzyme-linked immunosorbent assays. Apoptosis was analyzed through flow cytometry. MDA levels, GSH-Px activity, and ROS levels were determined by colorimetric methods and fluorescence microscopy, respectively. The association of METTL3 with ATXN2L and FOXL1 was investigated using a dual-luciferase reporter assay and RNA immunoprecipitation assay. Results HG treatment increased the secretion of pro-inflammatory factors, apoptosis rate, and oxidative stress in HRMECs. BMSC-derived exosomes inhibited inflammation, apoptosis and oxidative stress in HRMECs by transferring FOXL1 into HRMECs. FOXL1 functioned as an RNA-binding protein of METTL3, which stabilized ATXN2L mRNA expression through m6A methylation in HRMECs. ATXN2L expression was reduced in DR patients’ serum and HG-treated HRMECs. Overexpression of ATXN2L mitigated the high glucose-induced inflammation, apoptosis, and oxidative stress in HRMECs. Conclusion Exosomal FOXL1 from BMSCs stabilized METTL3 to increase ATXN2L expression, thus offering a protective effect against high glucose-induced injury in HRMECs. This finding holds clinical significance for the development of targeted therapies for DR.https://doi.org/10.1186/s13098-025-01804-7Diabetic retinopathyMesenchymal stem cellsExosomesFOXL1METTL3ATXN2L
spellingShingle Chao Niu
Daoquan Dong
Longjiang Cui
Yingli Dong
Wei Wang
Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
Diabetology & Metabolic Syndrome
Diabetic retinopathy
Mesenchymal stem cells
Exosomes
FOXL1
METTL3
ATXN2L
title Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
title_full Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
title_fullStr Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
title_full_unstemmed Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
title_short Exosomal FOXL1 from bone marrow mesenchymal stem cells activates the METTL3/ATXN2L pathway to ameliorate high glucose-induced human retinal microvascular endothelial cell injury
title_sort exosomal foxl1 from bone marrow mesenchymal stem cells activates the mettl3 atxn2l pathway to ameliorate high glucose induced human retinal microvascular endothelial cell injury
topic Diabetic retinopathy
Mesenchymal stem cells
Exosomes
FOXL1
METTL3
ATXN2L
url https://doi.org/10.1186/s13098-025-01804-7
work_keys_str_mv AT chaoniu exosomalfoxl1frombonemarrowmesenchymalstemcellsactivatesthemettl3atxn2lpathwaytoamelioratehighglucoseinducedhumanretinalmicrovascularendothelialcellinjury
AT daoquandong exosomalfoxl1frombonemarrowmesenchymalstemcellsactivatesthemettl3atxn2lpathwaytoamelioratehighglucoseinducedhumanretinalmicrovascularendothelialcellinjury
AT longjiangcui exosomalfoxl1frombonemarrowmesenchymalstemcellsactivatesthemettl3atxn2lpathwaytoamelioratehighglucoseinducedhumanretinalmicrovascularendothelialcellinjury
AT yinglidong exosomalfoxl1frombonemarrowmesenchymalstemcellsactivatesthemettl3atxn2lpathwaytoamelioratehighglucoseinducedhumanretinalmicrovascularendothelialcellinjury
AT weiwang exosomalfoxl1frombonemarrowmesenchymalstemcellsactivatesthemettl3atxn2lpathwaytoamelioratehighglucoseinducedhumanretinalmicrovascularendothelialcellinjury