The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis

Abstract Approximately 50% of the patients with ulcerative colitis (UC) are primarily nonresponsive to anti‐tumor necrosis factor (TNF) therapy or lose their responsiveness over time. The gut microbiota plays an important role in the resistance of UC to anti‐TNF therapy; however, the underlying mech...

Full description

Saved in:
Bibliographic Details
Main Authors: Jing Lei, Lin Lv, Li Zhong, Feng Xu, Wenhao Su, Yan Chen, Zhixuan Wu, Song He, Yongyu Chen
Format: Article
Language:English
Published: Wiley 2025-02-01
Series:Advanced Science
Subjects:
Online Access:https://doi.org/10.1002/advs.202413128
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850138327050616832
author Jing Lei
Lin Lv
Li Zhong
Feng Xu
Wenhao Su
Yan Chen
Zhixuan Wu
Song He
Yongyu Chen
author_facet Jing Lei
Lin Lv
Li Zhong
Feng Xu
Wenhao Su
Yan Chen
Zhixuan Wu
Song He
Yongyu Chen
author_sort Jing Lei
collection DOAJ
description Abstract Approximately 50% of the patients with ulcerative colitis (UC) are primarily nonresponsive to anti‐tumor necrosis factor (TNF) therapy or lose their responsiveness over time. The gut microbiota plays an important role in the resistance of UC to anti‐TNF therapy; however, the underlying mechanism remains unknown. Here, it is found that the transplantation of gut fecal microbiota from patients with UC alters the diversity of the gut microbiota in dextran sulfate sodium‐induced colitis mice and may affect the therapeutic responsiveness of mice to infliximab. Furthermore, the abundances of Romboutsia and Fusobacterium increase in the tissues of patients with UC who do not respond to anti‐TNF therapy. Differentially abundant metabolites are mainly enriched in nicotinate and nicotinamide metabolism in NCM460 cells after Fusobacterium nucleatum infection. Mechanistically, F. nucleatum promotes the nicotinamide adenine dinucleotide (NAD+) salvage pathway by upregulating NAMPT expression, which subsequently leads to the activation of the p38 mitogen‐activated protein kinase (MAPK) signaling pathway and promotes the secretion of inflammatory factors, ultimately inhibiting the therapeutic response to anti‐TNF drugs. These findings demonstrate that the gut microbiota can influence the response to anti‐TNF therapy in patients with UC and highlight the therapeutic potential of targeting F. nucleatum and its associated pathways for preventing and treating drug resistance in UC.
format Article
id doaj-art-b2c2014aca184901ae9bdeea364a7652
institution OA Journals
issn 2198-3844
language English
publishDate 2025-02-01
publisher Wiley
record_format Article
series Advanced Science
spelling doaj-art-b2c2014aca184901ae9bdeea364a76522025-08-20T02:30:35ZengWileyAdvanced Science2198-38442025-02-01128n/an/a10.1002/advs.202413128The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative ColitisJing Lei0Lin Lv1Li Zhong2Feng Xu3Wenhao Su4Yan Chen5Zhixuan Wu6Song He7Yongyu Chen8Department of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology Renmin Hospital of Wuhan University Hubei 430060 ChinaDepartment of Dermatovenereology Chengdu Second People's Hospital Sichuan 610011 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaDepartment of Gastroenterology The Second Affiliated Hospital of Chongqing Medical University Chongqing 400010 ChinaAbstract Approximately 50% of the patients with ulcerative colitis (UC) are primarily nonresponsive to anti‐tumor necrosis factor (TNF) therapy or lose their responsiveness over time. The gut microbiota plays an important role in the resistance of UC to anti‐TNF therapy; however, the underlying mechanism remains unknown. Here, it is found that the transplantation of gut fecal microbiota from patients with UC alters the diversity of the gut microbiota in dextran sulfate sodium‐induced colitis mice and may affect the therapeutic responsiveness of mice to infliximab. Furthermore, the abundances of Romboutsia and Fusobacterium increase in the tissues of patients with UC who do not respond to anti‐TNF therapy. Differentially abundant metabolites are mainly enriched in nicotinate and nicotinamide metabolism in NCM460 cells after Fusobacterium nucleatum infection. Mechanistically, F. nucleatum promotes the nicotinamide adenine dinucleotide (NAD+) salvage pathway by upregulating NAMPT expression, which subsequently leads to the activation of the p38 mitogen‐activated protein kinase (MAPK) signaling pathway and promotes the secretion of inflammatory factors, ultimately inhibiting the therapeutic response to anti‐TNF drugs. These findings demonstrate that the gut microbiota can influence the response to anti‐TNF therapy in patients with UC and highlight the therapeutic potential of targeting F. nucleatum and its associated pathways for preventing and treating drug resistance in UC.https://doi.org/10.1002/advs.202413128anti‐tumor necrosis factor therapyfusobacterium nucleatummicrobiotaNAD+ salvage pathwayulcerative colitis
spellingShingle Jing Lei
Lin Lv
Li Zhong
Feng Xu
Wenhao Su
Yan Chen
Zhixuan Wu
Song He
Yongyu Chen
The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
Advanced Science
anti‐tumor necrosis factor therapy
fusobacterium nucleatum
microbiota
NAD+ salvage pathway
ulcerative colitis
title The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
title_full The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
title_fullStr The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
title_full_unstemmed The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
title_short The Gut Microbiota Affects Anti‐TNF Responsiveness by Activating the NAD+ Salvage Pathway in Ulcerative Colitis
title_sort gut microbiota affects anti tnf responsiveness by activating the nad salvage pathway in ulcerative colitis
topic anti‐tumor necrosis factor therapy
fusobacterium nucleatum
microbiota
NAD+ salvage pathway
ulcerative colitis
url https://doi.org/10.1002/advs.202413128
work_keys_str_mv AT jinglei thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT linlv thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT lizhong thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT fengxu thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT wenhaosu thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT yanchen thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT zhixuanwu thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT songhe thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT yongyuchen thegutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT jinglei gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT linlv gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT lizhong gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT fengxu gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT wenhaosu gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT yanchen gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT zhixuanwu gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT songhe gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis
AT yongyuchen gutmicrobiotaaffectsantitnfresponsivenessbyactivatingthenadsalvagepathwayinulcerativecolitis