Arylsulfonamido-alkyl-sulfamates act as inhibitors of bovine carbonic anhydrase II
A small library of arylsulfonamido-alkyl sulfamates was prepared by a two-step synthesis from readily available starting materials. The compounds were tested for their ability to inhibit bovine carbonic anhydrase II. Several of them were found as good competitive inhibitors holding Ki values as low...
Saved in:
| Main Authors: | Toni C. Denner, Niels V. Heise, René Csuk |
|---|---|
| Format: | Article |
| Language: | English |
| Published: |
Elsevier
2024-12-01
|
| Series: | European Journal of Medicinal Chemistry Reports |
| Subjects: | |
| Online Access: | http://www.sciencedirect.com/science/article/pii/S2772417424000499 |
| Tags: |
Add Tag
No Tags, Be the first to tag this record!
|
Similar Items
-
Determination of trace sodium cyclohexyl sulfamate in Baijiu by HPLC
by: WEI Gong, WANG Le, LI Chunfang, ZHANG Zhiyang, REN Guojun, YAN Wei, WANG Hui
Published: (2024-04-01) -
A case-control study on the role of carbonic anhydrase autoantibodies in the pathogenesis and diagnosis of fibromyalgia
by: Hülya Kılıç, et al.
Published: (2025-04-01) -
Study of biotransformation of new selective carbonic anhydrase II inhibitor 4-(2-methyl-1,3-oxazole-5-yl)-benzenesulfonamide
by: A. L. Khokhlov, et al.
Published: (2023-11-01) -
<i>In Silico</i> Assessment of Enaminone–Sulfanilamides as Potential Carbonic Anhydrase II Inhibitors: Molecular Docking and ADMET Prediction
by: Yousra Ouafa Bouone, et al.
Published: (2024-11-01) -
Prospects for the application of inhibitors of carbonic anhydrase isoforms IX and XII in oncology
by: S. А. Kalinin, et al.
Published: (2024-04-01)