α-Heteroarylthiomethyl ketones: Small molecule inhibitors of 3CLpro

The main protease 3CLpro of the SARS-CoV-2 virus is a well--established therapeutic target for the treatment of COVID-19. In this study, we screened an in-house compound library and identified a series of α-heteroarylthiomethyl ketones as inhibitors of 3CLpro. Among these, analogues 31 and 33 emerge...

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Bibliographic Details
Main Authors: Knez Damijan, Proj Matic, Bozovičar Krištof, Gobec Stanislav
Format: Article
Language:English
Published: Sciendo 2025-06-01
Series:Acta Pharmaceutica
Subjects:
Online Access:https://doi.org/10.2478/acph-2025-0023
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