Development of a reliable, sensitive, and convenient assay for the discovery of new eIF5A hypusination inhibitors.

eIF5A is a translation factor dysregulated in several pathologies such as cancer and diabetes. eIF5A activity depends upon its hypusination, a unique post-translational modification catalyzed by two enzymes: DHPS and DOHH. Only a few molecules able to inhibit hypusination have been described, and no...

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Bibliographic Details
Main Authors: Oumayma Benaceur, Paula Ferreira Montenegro, Michel Kahi, Fabien Fontaine-Vive, Nathalie M Mazure, Mohamed Mehiri, Frederic Bost, Pascal Peraldi
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2025-01-01
Series:PLoS ONE
Online Access:https://doi.org/10.1371/journal.pone.0308049
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