Nucleophilic aromatic substitutions enable diversity-oriented synthesis of heterocyclic atropisomers via non-atropisomeric intermediates

Abstract Atropisomers are sterically hindered molecules whose formation typically proceeds via atropisomeric intermediates and encumbered transition states. It is therefore largely accepted that the activation energy is higher for synthesis of atropisomers than for synthesis of similar, less sterica...

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Bibliographic Details
Main Authors: Michal Šimek, Paritosh Dey, Vilém Blahout, Krishanu Mondal, Jeanne Ernenwein, Martin Dračínský, Daniel Bím, Paulo H. S. Paioti
Format: Article
Language:English
Published: Nature Portfolio 2025-05-01
Series:Nature Communications
Online Access:https://doi.org/10.1038/s41467-025-60101-z
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