Single-plate kinome screening in live-cells to enable highly cost-efficient kinase inhibitor profiling

Cancer research, cancer treatment, and the field of chemical biology are examples which heavily rely on the discovery of selective kinase inhibitors. While determining on-target potency is often feasible for most laboratories, the equally critical but frequently neglected selectivity screening remai...

Full description

Saved in:
Bibliographic Details
Main Authors: Martin P. Schwalm, Stefan Knapp
Format: Article
Language:English
Published: Elsevier 2025-03-01
Series:SLAS Discovery
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2472555225000073
Tags: Add Tag
No Tags, Be the first to tag this record!