Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides

Herein, we report an intramolecular 6-endo-dig cyclization of N-ferrocenyl propiolamides for the synthesis of planar chiral ferrocenes enabled by gold(I)-catalyzed hydroarylation. By using this protocol, a variety of planar chiral ferrocenopyridin-2(1H)-ones were obtained in good yields and excellen...

Full description

Saved in:
Bibliographic Details
Main Authors: Qian Zhou, Lulin Qiao, An-An Zhang, Lu Li, Tuan-Jie Meng, Baomin Fan, Yuan-Yuan Gao, Lantao Liu
Format: Article
Language:English
Published: KeAi Communications Co. Ltd. 2025-05-01
Series:Green Synthesis and Catalysis
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2666554924000279
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849427008734363648
author Qian Zhou
Lulin Qiao
An-An Zhang
Lu Li
Tuan-Jie Meng
Baomin Fan
Yuan-Yuan Gao
Lantao Liu
author_facet Qian Zhou
Lulin Qiao
An-An Zhang
Lu Li
Tuan-Jie Meng
Baomin Fan
Yuan-Yuan Gao
Lantao Liu
author_sort Qian Zhou
collection DOAJ
description Herein, we report an intramolecular 6-endo-dig cyclization of N-ferrocenyl propiolamides for the synthesis of planar chiral ferrocenes enabled by gold(I)-catalyzed hydroarylation. By using this protocol, a variety of planar chiral ferrocenopyridin-2(1H)-ones were obtained in good yields and excellent enantioselectivities (up to 96 % ee).
format Article
id doaj-art-57928d9b22d34f5e900a0fc60ac24099
institution Kabale University
issn 2666-5549
language English
publishDate 2025-05-01
publisher KeAi Communications Co. Ltd.
record_format Article
series Green Synthesis and Catalysis
spelling doaj-art-57928d9b22d34f5e900a0fc60ac240992025-08-20T03:29:10ZengKeAi Communications Co. Ltd.Green Synthesis and Catalysis2666-55492025-05-016219820110.1016/j.gresc.2024.02.007Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamidesQian Zhou0Lulin Qiao1An-An Zhang2Lu Li3Tuan-Jie Meng4Baomin Fan5Yuan-Yuan Gao6Lantao Liu7College of Chemistry, Zhengzhou University, Zhengzhou 450001, China; Henan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, ChinaHenan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, China; Key Laboratory of Chemistry in Ethnic Medicinal Resources, Yunnan Minzu University, Kunming 650500, ChinaHenan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, ChinaHenan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, ChinaHenan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, ChinaKey Laboratory of Chemistry in Ethnic Medicinal Resources, Yunnan Minzu University, Kunming 650500, China; Corresponding author. Key Laboratory of Chemistry in Ethnic Medicinal Resources, Yunnan Minzu University, Kunming 650500, China.Henan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, China; Corresponding author. College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, China.College of Chemistry, Zhengzhou University, Zhengzhou 450001, China; Henan Engineering Laboratory of Green Synthesis for Pharmaceuticals, College of Chemistry and Chemical Engineering, Shangqiu Normal University, Shangqiu 476000, China; Corresponding author. College of Chemistry, Zhengzhou University, Zhengzhou 450001, China.Herein, we report an intramolecular 6-endo-dig cyclization of N-ferrocenyl propiolamides for the synthesis of planar chiral ferrocenes enabled by gold(I)-catalyzed hydroarylation. By using this protocol, a variety of planar chiral ferrocenopyridin-2(1H)-ones were obtained in good yields and excellent enantioselectivities (up to 96 % ee).http://www.sciencedirect.com/science/article/pii/S2666554924000279Planar chiral ferrocenesEnantioselective synthesisGold(I)-catalyzed hydroarylation6-endo-dig cyclizationN-ferrocenyl propiolamides
spellingShingle Qian Zhou
Lulin Qiao
An-An Zhang
Lu Li
Tuan-Jie Meng
Baomin Fan
Yuan-Yuan Gao
Lantao Liu
Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
Green Synthesis and Catalysis
Planar chiral ferrocenes
Enantioselective synthesis
Gold(I)-catalyzed hydroarylation
6-endo-dig cyclization
N-ferrocenyl propiolamides
title Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
title_full Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
title_fullStr Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
title_full_unstemmed Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
title_short Enantioselective synthesis of planar chiral ferrocenes via gold(I)-catalyzed hydroarylation of N-ferrocenyl propiolamides
title_sort enantioselective synthesis of planar chiral ferrocenes via gold i catalyzed hydroarylation of n ferrocenyl propiolamides
topic Planar chiral ferrocenes
Enantioselective synthesis
Gold(I)-catalyzed hydroarylation
6-endo-dig cyclization
N-ferrocenyl propiolamides
url http://www.sciencedirect.com/science/article/pii/S2666554924000279
work_keys_str_mv AT qianzhou enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT lulinqiao enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT ananzhang enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT luli enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT tuanjiemeng enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT baominfan enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT yuanyuangao enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides
AT lantaoliu enantioselectivesynthesisofplanarchiralferrocenesviagoldicatalyzedhydroarylationofnferrocenylpropiolamides