Trimethyl Orthobenzoate as a1-C1-Phenyl-Synthon for Functionalization of 3-Unsubstituted Indoles
The methylindoles 2a and 2b are regioselectively functionalized with trimethyl orthobenzoate at C-3 by means of proton catalysis. The first stage is the formation of the key compounds, 3-indolyl-phenyl-methoxycarbenium ions 3. These can then be dealkylated under mild conditions using nucleophilic s...
Saved in:
| Main Authors: | , |
|---|---|
| Format: | Article |
| Language: | deu |
| Published: |
Swiss Chemical Society
1985-05-01
|
| Series: | CHIMIA |
| Online Access: | https://www.chimia.ch/chimia/article/view/9660 |
| Tags: |
Add Tag
No Tags, Be the first to tag this record!
|