Inhibition of Activated Coagulation Factor XII by the Phosphodiesterase-4 Inhibitor Roflumilast: In Vitro and In Silico Studies

Background: This study aimed to evaluate the effects of selected phosphodiesterase-4 inhibitors (PDE-4 inhibitors)—roflumilast, ibudilast, and crisaborole—on the activity of blood coagulation factor XII (FXII). In the intrinsic coagulation pathway, FXII is known to initiate the ka...

Full description

Saved in:
Bibliographic Details
Main Authors: Hassan A. Madkhali, Mohd Nazam Ansari, Mubarak A. Alamri
Format: Article
Language:English
Published: IMR Press 2025-05-01
Series:Frontiers in Bioscience-Landmark
Subjects:
Online Access:https://www.imrpress.com/journal/FBL/30/5/10.31083/FBL38395
Tags: Add Tag
No Tags, Be the first to tag this record!