Binding and Activating of Analgesic Crotalphine with Human TRPA1

TRPA1 (Transient Receptor Potential Ankyrin 1), a cation channel predominantly expressed in sensory neurons, plays a critical role in detecting noxious stimuli and mediating pain signal transmission. As a key player in nociceptive signaling pathways, TRPA1 has emerged as a promising therapeutic targ...

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Bibliographic Details
Main Authors: Mingmin Kang, Yanming Zhang, Xiufang Ding, Jianfu Xu, Xiaoyun Pang
Format: Article
Language:English
Published: MDPI AG 2025-06-01
Series:Membranes
Subjects:
Online Access:https://www.mdpi.com/2077-0375/15/6/187
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