Solvent-free and eco-friendly green protocol for N-Boc Protection of amines using picric acid as a catalyst

We have developed an environmentally conscious green protocol to protect amine functional groups in drug discovery and the total synthesis of biologically active natural products. This method utilizes di-tert-butyl dicarbonate ((Boc)2O) to protect aromatic and aliphatic amines, with readily availabl...

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Bibliographic Details
Main Authors: Ramesha Thongolla, Ummareddy Venkata Subba Reddy, Sailam Sri Gogula, Empati Raja Sekhar, Puchakayala Muralidhar Reddy, Anren Hu
Format: Article
Language:English
Published: Elsevier 2025-06-01
Series:Tetrahedron Green Chem
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Online Access:http://www.sciencedirect.com/science/article/pii/S2773223124000268
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