Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway

Abstract Breast cancer is a prevalent and deadly disease affecting women worldwide. Recent studies have shown that γ-glutamyl cyclotransferase (GGCT), an enzyme involved in glutathione metabolism, is consistently upregulated in various cancers. However, its specific role in breast cancer remains poo...

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Main Authors: De He, Weiheng Cui, Xijiao Pang, Jiale Dong, Quanwei Qiu, Hongmei Dong, Ruijun Zhao
Format: Article
Language:English
Published: Nature Portfolio 2025-06-01
Series:Scientific Reports
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Online Access:https://doi.org/10.1038/s41598-025-04500-8
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author De He
Weiheng Cui
Xijiao Pang
Jiale Dong
Quanwei Qiu
Hongmei Dong
Ruijun Zhao
author_facet De He
Weiheng Cui
Xijiao Pang
Jiale Dong
Quanwei Qiu
Hongmei Dong
Ruijun Zhao
author_sort De He
collection DOAJ
description Abstract Breast cancer is a prevalent and deadly disease affecting women worldwide. Recent studies have shown that γ-glutamyl cyclotransferase (GGCT), an enzyme involved in glutathione metabolism, is consistently upregulated in various cancers. However, its specific role in breast cancer remains poorly understood. This study aimed to investigate the functional role of GGCT in breast cancer. Bioinformatics, immunohistochemistry and immunoblotting analysis revealed that GGCT is significantly upregulated in breast cancer tissues, and its high expression is associated with poor survival outcomes. The knockdown of GGCT significantly suppressed MCF-7 and SKBR-3 cell activities. Cell proliferation decreased by 29.4–45.9%, and colony formation reduced by 51.5–56.6%. Migratory ability diminished by 36.8–49.1%, while invasion capability declined by 35.2–55.0%. Moreover, GGCT silencing reduced epithelial-mesenchymal transition (EMT) and inhibited the PI3K/AKT/mTOR signaling pathway. Notably, E-cadherin expression significantly increased in MCF-7 and SKBR-3-shGGCT cells, with changes ranging from 2.1-fold to 5.4-fold. Conversely, N-cadherin expression decreased by 54.2–84.2% in both cell lines. Vimentin expression also decreased significantly, with reductions of 58.8–83.0%. Further analyses indicated that p-AKT expression in MCF-7 and SKBR-3-shGGCT cells decreased by 51.4–84.8%. Additionally, p-mTOR expression was reduced by 71.2–87.2% in both cell lines, compared to shCtrl. Our data highlights the crucial role of GGCT in regulating EMT and the progression of breast cancer. The findings suggest that GGCT not only serves as a valuable prognostic marker but also represents a potential target for therapeutic interventions in breast cancer patients.
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spelling doaj-art-0be8c79a77b44c71aab7ffc636e02ecb2025-08-20T02:05:38ZengNature PortfolioScientific Reports2045-23222025-06-0115111110.1038/s41598-025-04500-8Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathwayDe He0Weiheng Cui1Xijiao Pang2Jiale Dong3Quanwei Qiu4Hongmei Dong5Ruijun Zhao6Department of Thyroid and Breast Surgery, PingXiang People’s HospitalInstitute of Precision Cancer Medicine and Pathology, Department of Pathology, School of Medicine, Jinan UniversityHenan key laboratory of tumor molecular biology medicine, First People’s Hospital of NanyangSchool of Nursing and Rehabilitation, Xi’an FANYI UniversityTumor Division, Anhui Anke Biotechnology (Group) Co.,LtdInstitute of Precision Cancer Medicine and Pathology, Department of Pathology, School of Medicine, Jinan UniversityDepartment of Breast Surgery, Nanchang People’s HospitalAbstract Breast cancer is a prevalent and deadly disease affecting women worldwide. Recent studies have shown that γ-glutamyl cyclotransferase (GGCT), an enzyme involved in glutathione metabolism, is consistently upregulated in various cancers. However, its specific role in breast cancer remains poorly understood. This study aimed to investigate the functional role of GGCT in breast cancer. Bioinformatics, immunohistochemistry and immunoblotting analysis revealed that GGCT is significantly upregulated in breast cancer tissues, and its high expression is associated with poor survival outcomes. The knockdown of GGCT significantly suppressed MCF-7 and SKBR-3 cell activities. Cell proliferation decreased by 29.4–45.9%, and colony formation reduced by 51.5–56.6%. Migratory ability diminished by 36.8–49.1%, while invasion capability declined by 35.2–55.0%. Moreover, GGCT silencing reduced epithelial-mesenchymal transition (EMT) and inhibited the PI3K/AKT/mTOR signaling pathway. Notably, E-cadherin expression significantly increased in MCF-7 and SKBR-3-shGGCT cells, with changes ranging from 2.1-fold to 5.4-fold. Conversely, N-cadherin expression decreased by 54.2–84.2% in both cell lines. Vimentin expression also decreased significantly, with reductions of 58.8–83.0%. Further analyses indicated that p-AKT expression in MCF-7 and SKBR-3-shGGCT cells decreased by 51.4–84.8%. Additionally, p-mTOR expression was reduced by 71.2–87.2% in both cell lines, compared to shCtrl. Our data highlights the crucial role of GGCT in regulating EMT and the progression of breast cancer. The findings suggest that GGCT not only serves as a valuable prognostic marker but also represents a potential target for therapeutic interventions in breast cancer patients.https://doi.org/10.1038/s41598-025-04500-8Breast cancerγ-Glutamyl cyclotransferaseProliferationMigrationInvasionPrognosis
spellingShingle De He
Weiheng Cui
Xijiao Pang
Jiale Dong
Quanwei Qiu
Hongmei Dong
Ruijun Zhao
Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
Scientific Reports
Breast cancer
γ-Glutamyl cyclotransferase
Proliferation
Migration
Invasion
Prognosis
title Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
title_full Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
title_fullStr Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
title_full_unstemmed Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
title_short Depletion of γ-glutamyl cyclotransferase suppresses the proliferation, migration and invasion of breast cancer cells accompanied by the activation of PI3K/AKT/mTOR pathway
title_sort depletion of γ glutamyl cyclotransferase suppresses the proliferation migration and invasion of breast cancer cells accompanied by the activation of pi3k akt mtor pathway
topic Breast cancer
γ-Glutamyl cyclotransferase
Proliferation
Migration
Invasion
Prognosis
url https://doi.org/10.1038/s41598-025-04500-8
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