Synthesis and Biological Activity of Glycosyl Thiazolyl Disulfides Based on Thiacarpine, an Analogue of the Cytotoxic Alkaloid Polycarpine from the Ascidian <i>Polycarpa aurata</i> by Dmitry N. Pelageev, Yuri E. Sabutski, Svetlana M. Kovach, Nadezhda N. Balaneva, Ekaterina S. Menchinskaya, Ekaterina A. Chingizova, Anna L. Burylova, Victor Ph. Anufriev

“…Based on this assumption, and to increase the selectivity of action, glycosyl disulfide conjugates of thiacarpine derivatives with thioglucose and thioxylose were synthesized and screened for their cytotoxic and antimicrobial activities. …”
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The effectiveness of eplerenone in clinical practice from the standpoint of evidence-based medicine (twenty years on the guard of life) by A. G. Evdokimova, R. I. Stryuk, V. V. Evdokimov, A. K. Kaptaeva

“…The article focuses on the negative role of hyperaldosteronism in cardiovascular diseases and the possibility of its control when using a selective mineralocorticoid receptor antagonist – eplerenone. …”
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Focused Ultrasound (FUS) for Chronic Pain Management: Approved and Potential Applications by Lazzaro di Biase, Emma Falato, Maria Letizia Caminiti, Pasquale Maria Pecoraro, Flavia Narducci, Vincenzo Di Lazzaro

“…FUS at nonablative dosage, LILFUS, has potential reversible and tissue-selective effects. FUS applications at nonablative doses currently are at a research stage. …”
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ADCY4 inhibits cAMP-induced growth of breast cancer by inactivating FAK/AKT and ERK signaling but is frequently silenced by DNA methylation by Guangrui Pan, Mingquan Huang, Shaozhi Fu, Yu Wang, Lijia He, Bin Wu, Jinping Yang, Sheng Lin, Yu Fan

“…Abstract Local increases in cyclic adenosine monophosphate (cAMP) caused by specific adenylyl cyclases (ACs) can selectively modulate related proteins. AC-selective drugs have an advantage in side effect control, and the specific AC may finally be considered as a therapeutic target. …”
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Influence of asphaltene precipitation on development effect of typical heavy oil reservoirs in eastern South China Sea by TU Yi, DAI Jianwen, YANG Jiao, WANG Yahui, MIAO Yun, ZHONG Xulin

“…The asphaltene molecules in crude oil precipitate through the cores if the formation pressures drop below the precipitation pressures of asphaltene. They first block small pores and throats and then block large throats and medium-large pores. …”
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Non-therapeutic play to overcome negative emotional symptoms and improve emotional intelligence in children aged 3–7: a systematic review by Alexander N. Veraksa, Valeriya A. Plotnikova, Vera L. Sukhikh, Dmitry S. Kornienko, Natalia A. Rudnova

“…Using the PRISMA method, we selected 33 articles for qualitative analysis from the 9,639 published articles over the past 5 years found through PubMed, ScienceDirect, and Scopus. …”
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Multi-factor consideration sample assignment for oriented tiny object detection by Jun Miao, Peng Liu, Yuanhua Qiao

“…Initially, we craft a dynamic prior block (DPB) to facilitate the dynamic alignment of priors with objects. …”
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A sleep staging model based on adversarial domain generalized residual attention network by Pengwei Zhang, Sijia Xiang, Kailei Hu, Jialing He, Jingxia Chen

“…In the feature extractor part, the channel attention network is combined with the residual block to selectively enhance the important features and the correlation between multi-channel physiological signals. …”
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RESULTS OF OPTIMIZATION OF PARAMETERS AND OPERATING MODES OF THE DISK PNEUMATIC SOWING DEVICE by V. V. Golubev, A. S. Firsov, D. M. Rula

“…The major studied factors were selected and levels of their variation were established. …”
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Respons Pertumbuhan Aren (Arenga pinnata Merr.) Fase TBM Umur 4 Tahun terhadap Aplikasi Variasi Dosis Pupuk Tunggal dan Majemuk by Fatimah Az Zahra, Mira Ariyanti

“…This study highlights the importance of selecting the appropriate type and dosage of fertilizer to improve sugar palm cultivation efficiency and provides valuable insights for optimizing practices during the immature phase.…”
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Green Tea Catechin, EGCG, Suppresses PCB 102-Induced Proliferation in Estrogen-Sensitive Breast Cancer Cells by Kimberly Mantzke Baker, Angela C. Bauer

“…Furthermore, the proliferative effects of PCB 102 were mediated by ERα and could be abrogated by the selective ERα antagonist MPP. EGCG (10–50 μM) caused a dose-dependent inhibition of PCB 102-induced cell proliferation, with nearly complete inhibition at 25 μM EGCG. …”
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ABOUT DATA MODELING SUBJECT DOMAINS PRACTICE-ORIENTED DIRECTION FOR UNIVERSAL SYSTEM OF STORAGE AND PROCESSING DATA by L. V. Rudikova, E. V. Zhavnerko

“…Using complex system, which can work with some information sources and represent data in convenient view for users will in-demand for analysis data selected subject domains and determination of possible relationships.…”
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PERBEDAAN HASIL BELAJAR SISWA YANG DIAJARKAN DENGAN MODEL PEMBELAJARAN KOOPERATIF TIPE THINK PAIR SHARE DAN MODEL PEMBELAJARAN KONVENSIONAL by Nilam Wally, Juliana Selvina Molle, Christina Martha Laamena

“…The population in this study were all eighth grade students of Ambon-Wathan High School with 100 students and the sample in this study was 40 students, selected using purposive sampling. The instrument used in this study was in the form of test questions which consisted of question details for the final test. …”
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RESPONSE OF SOME HERBACEOUS PLANTS TO DIFFERENT GROWING MEDIA AND POTASSIUM SILICATE FOLIAR SPRAYING IN (LWS) by A. M. S. Zalzala, S. A. Abdul Latif

“… This study was aimed to conduct one of the vertical garden systems , selecting suitable plant species that with stand the climate conditions of Baghdad city in outer space to determine the appropriate growing medium for the (LWS), and to assess the impact of spraying with potassium silicate on the resistance of the cultivated plants to heat stresses . …”
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Rate and Spraying Frequency Determination of Propiconazole Fungicide for the Management of Garlic Rust at Woreilu District, Northeastern Ethiopia by Admasie Kassaw, Aderajew Mihretie, Abebe Ayalew

“…A field experiment was conducted at Kabe and Segno Kebeles of Woreilu District in 2019 to determine the appropriate rate and spraying frequency of propiconazole fungicide and select cost-effective management options of garlic rust. …”
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Active faults paragenesis and the state of crustal stresses in the Late Cenozoic in Central Mongolia by V. A. Sankov, A. V. Parfeevets, A. I. Miroshnichenko, A. V. Sankov, A. Bayasgalan, D. Battogtokh

“…The study results show that faults activation during the Late Cenozoic stage was selective, and a cluster pattern of active faults is typical for the study region. …”
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<i>DSW-YOLO</i>-Based Green Pepper Detection Method Under Complex Environments by Yukuan Han, Gaifeng Ren, Jiarui Zhang, Yuxin Du, Guoqiang Bao, Lijun Cheng, Hongwen Yan

“…After comparing mainstream lightweight models (<i>YOLOv5n</i>, <i>YOLOv6n</i>, <i>YOLOv8n</i>, <i>YOLOv9t</i> and <i>YOLOv10n</i>), <i>YOLOv10n</i> with the best performance was selected as the baseline. The <i>DWRR</i> block was then designed and integrated with the <i>C2f</i> module to form <i>C2f</i>-<i>DWRR</i>, replacing the original <i>C2f</i> blocks in the backbone. …”
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Analgesic efficacy and safety of methylene blue combined with cocktail for periarticular infiltration following total knee arthroplasty: a prospective, randomized, controlled study by Yijiang Deng, Yong Yang, Feng Zhu, Wenzhi Liu, Jiarui Chen, Guangmin Xu

“…At the end of the surgery, the M group received a 0.05% methylene blue combined cocktail for periarticular infiltration block, while the C group received a conventional cocktail infiltration block. …”
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Research and Application of Evaluation Methods for Functional Characteristics of Oil-Based Drilling Fluid in Shale Gas Wells by Dewei Gao, Jiajun Xie, Shengming Huang, Shenyao Wu, Pengcheng Wu, Weian Huang

“…The new methods were used to evaluate the oil-based drilling fluid used in 4 wells in the Changning block. It was found that the drilling fluid of CN209H2 well adhered to the steel column with at least 0.41 g of cuttings; the recovery rate of the drilling fluid resistance of CN209H1 was up to 87.70%, and YX1200 oil-based drilling fluid plugging agent was selected through the microporous membrane experiment. …”
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Lactational performance of dairy cows fed diets based on corn silages varying in ruminal degradability of starch and fiber by S.F. Cueva, L.F. Martins, N. Stepanchenko, D.E. Wasson, Greg W. Roth, A.N. Hristov

“…The study was a randomized complete block design where cows within a block were randomly assigned to treatment diets. …”
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