Exploring covalent inhibitors of SARS-CoV-2 main protease: from peptidomimetics to novel scaffolds by Noor Atatreh, Radwa E. Mahgoub, Mohammad A. Ghattas

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Bicyclic peptide-enhanced covalent inhibitor of SARS-CoV-2 3CL protease by Qian Wang, Yanhui Wang, Jian Li, Hong Liu, Shiyu Chen

Subjects: “…protease covalent inhibitor…”
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Unanticipated mechanisms of covalent inhibitor and synthetic ligand cobinding to PPARγ by Jinsai Shang, Douglas J Kojetin

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Advancements, challenges, and future frontiers in covalent inhibitors and covalent drugs: A review by Muhammad Salman Hameed, Hongxuan Cao, Li Guo, Lei Zeng, Yanliang Ren

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Boronic acid inhibitors of penicillin-binding protein 1b: serine and lysine labelling agents by Levente Kollár, Katarina Grabrijan, Martina Hrast Rambaher, Krištof Bozovičar, Tímea Imre, György G. Ferenczy, Stanislav Gobec, György M. Keserű

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Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX by Aivaras Vaškevičius, Denis Baronas, Janis Leitans, Agnė Kvietkauskaitė, Audronė Rukšėnaitė, Elena Manakova, Zigmantas Toleikis, Algirdas Kaupinis, Andris Kazaks, Marius Gedgaudas, Aurelija Mickevičiūtė, Vaida Juozapaitienė, Helgi B Schiöth, Kristaps Jaudzems, Mindaugas Valius, Kaspars Tars, Saulius Gražulis, Franz-Josef Meyer-Almes, Jurgita Matulienė, Asta Zubrienė, Virginija Dudutienė, Daumantas Matulis

Subjects: “…targeted covalent inhibitors…”
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Miniaturized Modular Click Chemistry‐enabled Rapid Discovery of Unique SARS‐CoV‐2 Mpro Inhibitors With Robust Potency and Drug‐like Profile by Mianling Yang, Myoung Kyu Lee, Shenghua Gao, Letian Song, Hye‐Yeon Jang, Inseong Jo, Chun‐Chiao Yang, Katharina Sylvester, Chunkyu Ko, Shuo Wang, Bing Ye, Kai Tang, Junyi Li, Manyu Gu, Christa E. Müller, Norbert Sträter, Xinyong Liu, Meehyein Kim, Peng Zhan

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