Development of ketobenzothiazole-based peptidomimetic TMPRSS13 inhibitors with low nanomolar potency by Alexandre Joushomme, Antoine Désilets, William Champagne, Malihe Hassanzadeh, Gabriel Lemieux, Alice Gravel-Trudeau, Matthieu Lepage, Sabrina Lafrenière, Ulrike Froehlich, Karin List, Pierre-Luc Boudreault, Richard Leduc

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Advancing the development of TRIP13 inhibitors: A high-throughput screening approach by Rae M. Sammons, Soma Ghosh, Lacin Yapindi, Eun Jeong Cho, Faye M. Johnson, Kevin N. Dalby

Subjects: “…High throughput compound screening…”
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Development of a live cell assay for real-time monitoring the interactions between the Hippo pathway components 14-3-3 and TAZ by Blaž Andlovic, Alexander Wolf, Malgorzata Hiltmann, Bert M. Klebl, Jan Eickhoff, Christian Ottmann

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Novel high throughput 3D ECM remodeling assay identifies MEK as key driver of fibrotic fibroblast activity by Chen-Yi Liao, Jasmijn H.M. Hundscheid, Justin Crawford, Peter ten Dijke, Beatrice Coornaert, Erik H.J. Danen

Subjects: “…High-throughput compound screening…”
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Malformin C preferentially kills glioblastoma stem‐like cells via concerted induction of proteotoxic stress and autophagic flux blockade by Emma Phillips, Sizèd vanEnk, Sara Kildgaard, Silja Schlue, Mona Göttmann, Victoria Jennings, Frederic Bethke, Gabriele Müller, Christel Herold‐Mende, Daniel Pastor‐Flores, Martin Schneider, Dominic Helm, Thomas Ostenfeld Larsen, Violaine Goidts

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Screening, docking, and molecular dynamics analysis of Mitragyna speciosa (Korth.) compounds for targeting HER2 in breast cancer by Nabila Hadiah Akbar, Farendina Suarantika, Taufik Muhammad Fakih, Ariranur Haniffadli, Khoirunnisa Muslimawati, Aditya Maulana Perdana Putra

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