Identification of low-molecular compounds that inhibit envelope formation of hepatitis B virus by Kosuke Sato, Jun Inoue, Masashi Ninomiya, Akitoshi Sano, Mio Tsuruoka, Masazumi Onuki, Satoko Sawahashi, Keishi Ouchi, Kotaro Doi, Kengo Watanabe, Atsushi Masamune

Subjects: Get full text

Development of a cell-based target engagement assay for pyruvate dehydrogenase kinase by Mya D. Gough, Matthew B. Robers, Cesear R. Corona, Ranjit K. Mehta, Mukesh K. Nyati, Peter L. Toogood

Subjects: Get full text

A simple method to generate stable cell lines for the analysis of transient protein-protein interactions by Emilia Elizabeth Savage, Denise Wootten, Arthur Christopoulos, Patrick Michael Sexton, Sebastian George Barton Furness

Subjects: “…BRET…”
Get full text

Problem of Periodization and Some Aspects of the Late Work of F. Bret Hart by A. B. Tanaseichuk, O. Yu. Osmukhina

Subjects: “…bret hart…”
Get full text

New heterocyclic A1/A3 adenosine receptor ligands through molecular simplification strategies by Letizia Crocetti, Abigail Pearce, Venkat S. Vege, Qi Xu, Jing Xu, Hannes Buthmann, Maria Paola Giovannoni, Gabriella Guerrini, Francesca Catarzi, Silvia Selleri, Xianglin Huang, Aneesh Chandran, Graham Ladds, Agostino Cilibrizzi

Subjects: Get full text

Biased antagonism of a series of bicyclic CXCR2 intracellular allosteric modulators by Brent Van Bosstraeten, Katrijn Boon, Max Van Hoof, Wim Dehaen, Martyna Szpakowska, Andy Chevigné, Dominique Schols, Steven De Jonghe, Tom Van Loy

Subjects: Get full text

Comparative evaluation of cell-based assay technologies for scoring drug-induced condensation of SARS-CoV-2 nucleocapsid protein by Rui Tong Quek, Cyna R. Shirazinejad, Christina L. Young, Kierra S. Hardy, Samuel Lim, Phillip J. Elms, David T. McSwiggen, Timothy J. Mitchison, Pamela A. Silver

Subjects: Get full text

Estrogenic activity of E2-conjugated GLP-1 is mediated by intracellular endolysosomal acidification and estrone metabolism by Callum Coupland, Na Sun, Ahmed Khalil, Özüm Ezgi Karaoglu, Arkadiusz Liskiewicz, Daniela Liskiewicz, Gerald Grandl, Seun Akindehin, Gandhari Maity, Bin Yang, Brian Finan, Patrick Knerr, Jonathan D. Douros, Axel Walch, Richard DiMarchi, Matthias H. Tschöp, Timo D. Müller, Aaron Novikoff

Subjects: “…Bioluminescence resonance energy transfer (BRET)…”
Get full text

Quantification of Wnt3a, Wnt5a and Wnt16 Binding to Multiple Frizzleds Under Physiological Conditions Using NanoBit/BRET by Janine Wesslowski, Sadia Safi, Michelle Rottmann, Melanie Rothley, Gary Davidson

Subjects: Get full text

Les origines de la critique de science-fiction : de Kepler à Wells by Arthur B. Evans

Subjects: Get full text

Small molecules targeting the eubacterial β-sliding clamp discovered by combined in silico and in vitro screening approaches by Alessia Caputo, Gian Marco Elisi, Elisabetta Levati, Giulia Barotti, Sara Sartini, Jerome Wagner, Dominique Y. Burnouf, Simone Ottonello, Silvia Rivara, Barbara Montanini

Subjects: “…yeast Bioluminescence Resonance Energy Transfer (yBRET)…”
Get full text

Unraveling ER dimerization dynamics in endocrine disruption based on a BRET-focused approach by Soomin Yum, Haksoo Lee, Yong-Kook Kwon, Gunyoung Lee, Hye-Young Lee, HyeSook Youn, BuHyun Youn

Subjects: “…bioluminescence resonance energy transfer (BRET)…”
Get full text

Dual compartment utility of BRET-based biosensors for PPP2R5A/B56α, a cancer-associated B regulatory subunit of PP2A by Hirofumi Yamauchi, Atsuro Oishi, Masahiko Ajiro, Atsuhito Nakayama, Kazuki Nishimura, Michiko Kurikawa, Mina Yoshida, Rei Kudo, Minori Koizumi, Takuya Izumi-Tamura, Miki Nagase, Natsuko Shinohara, Mayumi Hanzawa, Marimu Sakumoto, Takahiro Nishino, Ryoichi Maenosono, Asuka Kawachi, Junko Mukohyama, Shingo Yano, Tomoya Muto, Akihide Yoshimi

Subjects: “…bioluminescence resonance energy transfer (BRET)…”
Get full text

The cell adhesion molecule CD44 acts as a modulator of 5-HT7 receptor functions by Saskia Borsdorf, Andre Zeug, Yuxin Wu, Elena Mitroshina, Maria Vedunova, Supriya A. Gaitonde, Michel Bouvier, Michael C. Wehr, Josephine Labus, Evgeni Ponimaskin

Subjects: “…Bioluminescence Resonance Energy Transfer (BRET)…”
Get full text