Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.

<h4>Background</h4>Cutaneous leishmaniasis (CL) is treated with parenteral drugs for decades with decreasing rate cures. Miltefosine is an oral medication with anti-leishmania activity and may increase the cure rates and improve compliance.<h4>Methodology/principal findings</h4&...

Full description

Saved in:
Bibliographic Details
Main Authors: Paulo R Machado, Julia Ampuero, Luiz H Guimarães, Leonardo Villasboas, Ana T Rocha, Albert Schriefer, Rosana S Sousa, Anette Talhari, Gerson Penna, Edgar M Carvalho
Format: Article
Language:English
Published: Public Library of Science (PLoS) 2010-12-01
Series:PLoS Neglected Tropical Diseases
Online Access:https://journals.plos.org/plosntds/article/file?id=10.1371/journal.pntd.0000912&type=printable
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850025412741038080
author Paulo R Machado
Julia Ampuero
Luiz H Guimarães
Leonardo Villasboas
Ana T Rocha
Albert Schriefer
Rosana S Sousa
Anette Talhari
Gerson Penna
Edgar M Carvalho
author_facet Paulo R Machado
Julia Ampuero
Luiz H Guimarães
Leonardo Villasboas
Ana T Rocha
Albert Schriefer
Rosana S Sousa
Anette Talhari
Gerson Penna
Edgar M Carvalho
author_sort Paulo R Machado
collection DOAJ
description <h4>Background</h4>Cutaneous leishmaniasis (CL) is treated with parenteral drugs for decades with decreasing rate cures. Miltefosine is an oral medication with anti-leishmania activity and may increase the cure rates and improve compliance.<h4>Methodology/principal findings</h4>This study is a randomized, open-label, controlled clinical trial aimed to evaluate the efficacy and safety of miltefosine versus pentavalent antimony (Sb(v)) in the treatment of patients with CL caused by Leishmania braziliensis in Bahia, Brazil. A total of 90 patients were enrolled in the trial; 60 were assigned to receive miltefosine and 30 to receive Sb(v). Six months after treatment, in the intention-to-treat analyses, the definitive cure rate was 53.3% in the Sb(v) group and 75% in the miltefosine group (difference of 21.7%, 95% CI 0.08% to 42.7%, p = 0.04). Miltefosine was more effective than Sb(v) in the age group of 13-65 years-old compared to 2-12 years-old group (78.9% versus 45% p = 0.02; 68.2% versus 70% p = 1.0, respectively). The incidence of adverse events was similar in the Sb(v) and miltefosine groups (76.7% vs. 78.3%). Vomiting (41.7%), nausea (40%), and abdominal pain (23.3%) were significantly more frequent in the miltefosine group while arthralgias (20.7%), mialgias (20.7%) and fever (23.3%) were significantly more frequent in the Sb(v) group.<h4>Conclusions</h4>This study demonstrates that miltefosine therapy is more effective than standard Sb(v) and safe for the treatment of CL caused by Leishmania braziliensis in Bahia, Brazil.<h4>Trial registration</h4>Clinicaltrials.gov Identifier NCT00600548.
format Article
id doaj-art-fed5a58e5fb04ecead71ad89bc5a3d97
institution DOAJ
issn 1935-2727
1935-2735
language English
publishDate 2010-12-01
publisher Public Library of Science (PLoS)
record_format Article
series PLoS Neglected Tropical Diseases
spelling doaj-art-fed5a58e5fb04ecead71ad89bc5a3d972025-08-20T03:00:51ZengPublic Library of Science (PLoS)PLoS Neglected Tropical Diseases1935-27271935-27352010-12-01412e91210.1371/journal.pntd.0000912Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.Paulo R MachadoJulia AmpueroLuiz H GuimarãesLeonardo VillasboasAna T RochaAlbert SchrieferRosana S SousaAnette TalhariGerson PennaEdgar M Carvalho<h4>Background</h4>Cutaneous leishmaniasis (CL) is treated with parenteral drugs for decades with decreasing rate cures. Miltefosine is an oral medication with anti-leishmania activity and may increase the cure rates and improve compliance.<h4>Methodology/principal findings</h4>This study is a randomized, open-label, controlled clinical trial aimed to evaluate the efficacy and safety of miltefosine versus pentavalent antimony (Sb(v)) in the treatment of patients with CL caused by Leishmania braziliensis in Bahia, Brazil. A total of 90 patients were enrolled in the trial; 60 were assigned to receive miltefosine and 30 to receive Sb(v). Six months after treatment, in the intention-to-treat analyses, the definitive cure rate was 53.3% in the Sb(v) group and 75% in the miltefosine group (difference of 21.7%, 95% CI 0.08% to 42.7%, p = 0.04). Miltefosine was more effective than Sb(v) in the age group of 13-65 years-old compared to 2-12 years-old group (78.9% versus 45% p = 0.02; 68.2% versus 70% p = 1.0, respectively). The incidence of adverse events was similar in the Sb(v) and miltefosine groups (76.7% vs. 78.3%). Vomiting (41.7%), nausea (40%), and abdominal pain (23.3%) were significantly more frequent in the miltefosine group while arthralgias (20.7%), mialgias (20.7%) and fever (23.3%) were significantly more frequent in the Sb(v) group.<h4>Conclusions</h4>This study demonstrates that miltefosine therapy is more effective than standard Sb(v) and safe for the treatment of CL caused by Leishmania braziliensis in Bahia, Brazil.<h4>Trial registration</h4>Clinicaltrials.gov Identifier NCT00600548.https://journals.plos.org/plosntds/article/file?id=10.1371/journal.pntd.0000912&type=printable
spellingShingle Paulo R Machado
Julia Ampuero
Luiz H Guimarães
Leonardo Villasboas
Ana T Rocha
Albert Schriefer
Rosana S Sousa
Anette Talhari
Gerson Penna
Edgar M Carvalho
Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
PLoS Neglected Tropical Diseases
title Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
title_full Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
title_fullStr Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
title_full_unstemmed Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
title_short Miltefosine in the treatment of cutaneous leishmaniasis caused by Leishmania braziliensis in Brazil: a randomized and controlled trial.
title_sort miltefosine in the treatment of cutaneous leishmaniasis caused by leishmania braziliensis in brazil a randomized and controlled trial
url https://journals.plos.org/plosntds/article/file?id=10.1371/journal.pntd.0000912&type=printable
work_keys_str_mv AT paulormachado miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT juliaampuero miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT luizhguimaraes miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT leonardovillasboas miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT anatrocha miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT albertschriefer miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT rosanassousa miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT anettetalhari miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT gersonpenna miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial
AT edgarmcarvalho miltefosineinthetreatmentofcutaneousleishmaniasiscausedbyleishmaniabraziliensisinbrazilarandomizedandcontrolledtrial