Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery

In recent decades, nose-to-brain drug delivery has shown effectiveness in treating many central nervous system diseases. Intranasally administered drugs can be delivered to the brain through the olfactory and trigeminal pathways that bypass the blood–brain barrier. However, nose-to-brain drug delive...

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Main Authors: Thi-Thao-Linh Nguyen, Van-An Duong
Format: Article
Language:English
Published: MDPI AG 2025-04-01
Series:Pharmaceuticals
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Online Access:https://www.mdpi.com/1424-8247/18/5/615
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author Thi-Thao-Linh Nguyen
Van-An Duong
author_facet Thi-Thao-Linh Nguyen
Van-An Duong
author_sort Thi-Thao-Linh Nguyen
collection DOAJ
description In recent decades, nose-to-brain drug delivery has shown effectiveness in treating many central nervous system diseases. Intranasally administered drugs can be delivered to the brain through the olfactory and trigeminal pathways that bypass the blood–brain barrier. However, nose-to-brain drug delivery is challenging due to the inadequate nasal mucosa absorption of drugs and the short retention time of the intranasal formulations. These problems can be minimized through the use of nano-drug delivery systems, such as micelles, polymeric nanoparticles, nanoemulsions, liposomes, solid lipid nanoparticles, and nanostructured lipid carriers. They can enhance the drug’s bioavailability in the brain via increases in drug solubility, permeation, and stability. Nose-to-brain nano-drug delivery systems have been evaluated in vivo by a number of research groups. This review aims to provide an overview of nose-to-brain delivery and recent advances in the development of nano-drug delivery systems for delivering drugs from the nose to the brain to improve the treatment of some central nervous system diseases.
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spelling doaj-art-fa56c6a2d0c84e51b85303663550e9082025-08-20T03:14:36ZengMDPI AGPharmaceuticals1424-82472025-04-0118561510.3390/ph18050615Advancements in Nanocarrier Systems for Nose-to-Brain Drug DeliveryThi-Thao-Linh Nguyen0Van-An Duong1Institute of Pharmaceutical Education and Research, Binh Duong University, Thu Dau Mot City 820000, Binh Duong, VietnamThe Institute of Molecular Medicine, The University of Texas Health Science Center at Houston, Houston, TX 77030, USAIn recent decades, nose-to-brain drug delivery has shown effectiveness in treating many central nervous system diseases. Intranasally administered drugs can be delivered to the brain through the olfactory and trigeminal pathways that bypass the blood–brain barrier. However, nose-to-brain drug delivery is challenging due to the inadequate nasal mucosa absorption of drugs and the short retention time of the intranasal formulations. These problems can be minimized through the use of nano-drug delivery systems, such as micelles, polymeric nanoparticles, nanoemulsions, liposomes, solid lipid nanoparticles, and nanostructured lipid carriers. They can enhance the drug’s bioavailability in the brain via increases in drug solubility, permeation, and stability. Nose-to-brain nano-drug delivery systems have been evaluated in vivo by a number of research groups. This review aims to provide an overview of nose-to-brain delivery and recent advances in the development of nano-drug delivery systems for delivering drugs from the nose to the brain to improve the treatment of some central nervous system diseases.https://www.mdpi.com/1424-8247/18/5/615nose-to-brainnanoparticlesmicellesemulsionsliposomesSLNs
spellingShingle Thi-Thao-Linh Nguyen
Van-An Duong
Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
Pharmaceuticals
nose-to-brain
nanoparticles
micelles
emulsions
liposomes
SLNs
title Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
title_full Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
title_fullStr Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
title_full_unstemmed Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
title_short Advancements in Nanocarrier Systems for Nose-to-Brain Drug Delivery
title_sort advancements in nanocarrier systems for nose to brain drug delivery
topic nose-to-brain
nanoparticles
micelles
emulsions
liposomes
SLNs
url https://www.mdpi.com/1424-8247/18/5/615
work_keys_str_mv AT thithaolinhnguyen advancementsinnanocarriersystemsfornosetobraindrugdelivery
AT vananduong advancementsinnanocarriersystemsfornosetobraindrugdelivery