Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC

Abstract Background Despite extensive research on hypoxia in hepatocellular carcinoma (HCC), previous studies have relied on pre-existing hypoxia gene sets, limiting their specificity. We developed a novel approach using direct comparison of hypoxic versus normoxic HCC cell lines to establish a more...

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Main Authors: Min Su, Haibo Duan, Yu Gu, Jianfu Zhao
Format: Article
Language:English
Published: Springer 2025-06-01
Series:Discover Oncology
Subjects:
Online Access:https://doi.org/10.1007/s12672-025-02923-3
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author Min Su
Haibo Duan
Yu Gu
Jianfu Zhao
author_facet Min Su
Haibo Duan
Yu Gu
Jianfu Zhao
author_sort Min Su
collection DOAJ
description Abstract Background Despite extensive research on hypoxia in hepatocellular carcinoma (HCC), previous studies have relied on pre-existing hypoxia gene sets, limiting their specificity. We developed a novel approach using direct comparison of hypoxic versus normoxic HCC cell lines to establish a more precise hypoxia signature. Methods Through differential gene expression analysis of HCC cells under controlled oxygen conditions (GSE185969) and integration with TCGA-LIHC data, we identified and validated a highly specific 29-gene hypoxia signature. We performed comprehensive immune profiling and genomic instability analyses using multi-omics approaches. Results Our HCC-specific hypoxia signature demonstrated superior prognostic value (AUC: 0.805, 0.805, 0.748 at 1/3/5 years) compared to conventional hypoxia markers. High-risk tumors showed distinct immunosuppressive features including reduced CD8 + T cells and elevated Th2 cells, along with significantly increased expression of immune checkpoints CD274 (PD-1, p < 0.05) and CD276 (B7-H3, r = 0.62, p < 0.001). Notably, we uncovered an unexpected inverse relationship between hypoxia-induced genomic instability and PARP inhibitor sensitivity, challenging current therapeutic paradigms. Conclusion Our methodology establishes a more precise hypoxia signature specific to HCC, advancing beyond traditional approaches. The paradoxical finding of reduced PARP inhibitor sensitivity in genomically unstable tumors reveals new complexities in hypoxia-driven treatment resistance, suggesting the need for alternative therapeutic strategies in hypoxic HCC.
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spelling doaj-art-ecf1a7c334eb42ad8febc43d1184df5b2025-08-20T03:22:50ZengSpringerDiscover Oncology2730-60112025-06-0116111410.1007/s12672-025-02923-3Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCCMin Su0Haibo Duan1Yu Gu2Jianfu Zhao3Department of Oncology, Cancer Diagnosis and Therapy Research Center, The First Affiliated Hospital of Jinan UniversityDepartment of Oncology, Cancer Diagnosis and Therapy Research Center, The First Affiliated Hospital of Jinan UniversityGuangzhou Institute of Cancer Research, Affiliated Cancer Hospital,Guangzhou Medical UniversityDepartment of Oncology, Cancer Diagnosis and Therapy Research Center, The First Affiliated Hospital of Jinan UniversityAbstract Background Despite extensive research on hypoxia in hepatocellular carcinoma (HCC), previous studies have relied on pre-existing hypoxia gene sets, limiting their specificity. We developed a novel approach using direct comparison of hypoxic versus normoxic HCC cell lines to establish a more precise hypoxia signature. Methods Through differential gene expression analysis of HCC cells under controlled oxygen conditions (GSE185969) and integration with TCGA-LIHC data, we identified and validated a highly specific 29-gene hypoxia signature. We performed comprehensive immune profiling and genomic instability analyses using multi-omics approaches. Results Our HCC-specific hypoxia signature demonstrated superior prognostic value (AUC: 0.805, 0.805, 0.748 at 1/3/5 years) compared to conventional hypoxia markers. High-risk tumors showed distinct immunosuppressive features including reduced CD8 + T cells and elevated Th2 cells, along with significantly increased expression of immune checkpoints CD274 (PD-1, p < 0.05) and CD276 (B7-H3, r = 0.62, p < 0.001). Notably, we uncovered an unexpected inverse relationship between hypoxia-induced genomic instability and PARP inhibitor sensitivity, challenging current therapeutic paradigms. Conclusion Our methodology establishes a more precise hypoxia signature specific to HCC, advancing beyond traditional approaches. The paradoxical finding of reduced PARP inhibitor sensitivity in genomically unstable tumors reveals new complexities in hypoxia-driven treatment resistance, suggesting the need for alternative therapeutic strategies in hypoxic HCC.https://doi.org/10.1007/s12672-025-02923-3Hepatocellular carcinomaHypoxiaGenomic instabilityTumor immune microenvironmentPrognostic signature
spellingShingle Min Su
Haibo Duan
Yu Gu
Jianfu Zhao
Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
Discover Oncology
Hepatocellular carcinoma
Hypoxia
Genomic instability
Tumor immune microenvironment
Prognostic signature
title Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
title_full Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
title_fullStr Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
title_full_unstemmed Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
title_short Hypoxia-related signatures predicts survival, immunosuppression and PARP inhibitor resistance in HCC
title_sort hypoxia related signatures predicts survival immunosuppression and parp inhibitor resistance in hcc
topic Hepatocellular carcinoma
Hypoxia
Genomic instability
Tumor immune microenvironment
Prognostic signature
url https://doi.org/10.1007/s12672-025-02923-3
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AT haiboduan hypoxiarelatedsignaturespredictssurvivalimmunosuppressionandparpinhibitorresistanceinhcc
AT yugu hypoxiarelatedsignaturespredictssurvivalimmunosuppressionandparpinhibitorresistanceinhcc
AT jianfuzhao hypoxiarelatedsignaturespredictssurvivalimmunosuppressionandparpinhibitorresistanceinhcc