#Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1

Influenza virus flu A H1N1 still remains a target for its inhibition with small molecules. Fleeting nitrosocarbonyl intermediates are at work in a short-cut synthesis of carbocyclic nucleoside analogues. The strategy of the synthetic approaches is presented along with the in vitro antiviral tests. T...

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Main Authors: Dalya Al-Saad, Misal Giuseppe Memeo, Paolo Quadrelli
Format: Article
Language:English
Published: Wiley 2014-01-01
Series:The Scientific World Journal
Online Access:http://dx.doi.org/10.1155/2014/472373
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author Dalya Al-Saad
Misal Giuseppe Memeo
Paolo Quadrelli
author_facet Dalya Al-Saad
Misal Giuseppe Memeo
Paolo Quadrelli
author_sort Dalya Al-Saad
collection DOAJ
description Influenza virus flu A H1N1 still remains a target for its inhibition with small molecules. Fleeting nitrosocarbonyl intermediates are at work in a short-cut synthesis of carbocyclic nucleoside analogues. The strategy of the synthetic approaches is presented along with the in vitro antiviral tests. The nucleoside derivatives were tested for their inhibitory activity against a variety of viruses. Promising antiviral activities were found for specific compounds in the case of flu A H1N1.
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publishDate 2014-01-01
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series The Scientific World Journal
spelling doaj-art-ec83b3e50d8d4476a8ea892e289edfc02025-08-20T02:21:49ZengWileyThe Scientific World Journal2356-61401537-744X2014-01-01201410.1155/2014/472373472373#Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1Dalya Al-Saad0Misal Giuseppe Memeo1Paolo Quadrelli2Department of Chemistry, University of Pavia, Viale Taramelli 12, 27100 Pavia, ItalyDepartment of Chemistry, University of Pavia, Viale Taramelli 12, 27100 Pavia, ItalyDepartment of Chemistry, University of Pavia, Viale Taramelli 12, 27100 Pavia, ItalyInfluenza virus flu A H1N1 still remains a target for its inhibition with small molecules. Fleeting nitrosocarbonyl intermediates are at work in a short-cut synthesis of carbocyclic nucleoside analogues. The strategy of the synthetic approaches is presented along with the in vitro antiviral tests. The nucleoside derivatives were tested for their inhibitory activity against a variety of viruses. Promising antiviral activities were found for specific compounds in the case of flu A H1N1.http://dx.doi.org/10.1155/2014/472373
spellingShingle Dalya Al-Saad
Misal Giuseppe Memeo
Paolo Quadrelli
#Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
The Scientific World Journal
title #Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
title_full #Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
title_fullStr #Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
title_full_unstemmed #Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
title_short #Nitrosocarbonyls 1: Antiviral Activity of N-(4-Hydroxycyclohex-2-en-1-yl)quinoline-2-carboxamide against the Influenza A Virus H1N1
title_sort nitrosocarbonyls 1 antiviral activity of n 4 hydroxycyclohex 2 en 1 yl quinoline 2 carboxamide against the influenza a virus h1n1
url http://dx.doi.org/10.1155/2014/472373
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