Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development

Rheumatoid arthritis (RA) is a chronic systemic autoimmune disease with severe complications. Ferroptosis, an iron-dependent form of apoptosis, encompasses mechanisms including iron overload, lipid peroxidation, redox homeostasis, and reactive oxygen species accumulation, all of which are closely re...

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Main Authors: Zhuoling Wang, Xinyue Bai, Huahua Zhang, Min Yang, Meilin Liu, Tingyu Nie, Tianjiao Li, Mingru Zhang, Xingdan Wang, Jin Wang, Jiming Han, Xiaolong Liu
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-06-01
Series:Frontiers in Immunology
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Online Access:https://www.frontiersin.org/articles/10.3389/fimmu.2025.1610121/full
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author Zhuoling Wang
Xinyue Bai
Huahua Zhang
Min Yang
Meilin Liu
Tingyu Nie
Tianjiao Li
Mingru Zhang
Xingdan Wang
Jin Wang
Jiming Han
Xiaolong Liu
author_facet Zhuoling Wang
Xinyue Bai
Huahua Zhang
Min Yang
Meilin Liu
Tingyu Nie
Tianjiao Li
Mingru Zhang
Xingdan Wang
Jin Wang
Jiming Han
Xiaolong Liu
author_sort Zhuoling Wang
collection DOAJ
description Rheumatoid arthritis (RA) is a chronic systemic autoimmune disease with severe complications. Ferroptosis, an iron-dependent form of apoptosis, encompasses mechanisms including iron overload, lipid peroxidation, redox homeostasis, and reactive oxygen species accumulation, all of which are closely related to RA pathogenesis. This study focused on the mechanism of ferroptosis and RA, detailing their relationship and outlining the reported roles of ferroptosis inhibitors in RA treatment to provide a useful research basis in drug discovery and development and for clinicians.
format Article
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institution OA Journals
issn 1664-3224
language English
publishDate 2025-06-01
publisher Frontiers Media S.A.
record_format Article
series Frontiers in Immunology
spelling doaj-art-e9088e65d5ce4688b5f914ba1a2a17c32025-08-20T02:08:46ZengFrontiers Media S.A.Frontiers in Immunology1664-32242025-06-011610.3389/fimmu.2025.16101211610121Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor developmentZhuoling Wang0Xinyue Bai1Huahua Zhang2Min Yang3Meilin Liu4Tingyu Nie5Tianjiao Li6Mingru Zhang7Xingdan Wang8Jin Wang9Jiming Han10Xiaolong Liu11Medical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaNursing Department of Yan’an University Affiliated Hospital, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaMedical Research and Experiment Center, Yan’an Medical College of Yan’an University, Yan’an, ChinaRheumatoid arthritis (RA) is a chronic systemic autoimmune disease with severe complications. Ferroptosis, an iron-dependent form of apoptosis, encompasses mechanisms including iron overload, lipid peroxidation, redox homeostasis, and reactive oxygen species accumulation, all of which are closely related to RA pathogenesis. This study focused on the mechanism of ferroptosis and RA, detailing their relationship and outlining the reported roles of ferroptosis inhibitors in RA treatment to provide a useful research basis in drug discovery and development and for clinicians.https://www.frontiersin.org/articles/10.3389/fimmu.2025.1610121/fullferroptosisrheumatoid arthritislipid peroxidationnatural medicinenanomedicine
spellingShingle Zhuoling Wang
Xinyue Bai
Huahua Zhang
Min Yang
Meilin Liu
Tingyu Nie
Tianjiao Li
Mingru Zhang
Xingdan Wang
Jin Wang
Jiming Han
Xiaolong Liu
Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
Frontiers in Immunology
ferroptosis
rheumatoid arthritis
lipid peroxidation
natural medicine
nanomedicine
title Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
title_full Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
title_fullStr Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
title_full_unstemmed Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
title_short Targeting the ferroptosis pathway for rheumatoid arthritis: molecular mechanisms and prospects for inhibitor development
title_sort targeting the ferroptosis pathway for rheumatoid arthritis molecular mechanisms and prospects for inhibitor development
topic ferroptosis
rheumatoid arthritis
lipid peroxidation
natural medicine
nanomedicine
url https://www.frontiersin.org/articles/10.3389/fimmu.2025.1610121/full
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