Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs

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Main Authors: Chungen Li, Yihan Chen, Weixue Huang, Yudi Qiu, Shengjie Huang, Yang Zhou, Fengtao Zhou, Jian Xu, Xiaomei Ren, Jinwei Zhang, Zhen Wang, Ming Ding, Ke Ding
Format: Article
Language:English
Published: American Chemical Society 2024-11-01
Series:JACS Au
Online Access:https://doi.org/10.1021/jacsau.4c00831
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author Chungen Li
Yihan Chen
Weixue Huang
Yudi Qiu
Shengjie Huang
Yang Zhou
Fengtao Zhou
Jian Xu
Xiaomei Ren
Jinwei Zhang
Zhen Wang
Ming Ding
Ke Ding
author_facet Chungen Li
Yihan Chen
Weixue Huang
Yudi Qiu
Shengjie Huang
Yang Zhou
Fengtao Zhou
Jian Xu
Xiaomei Ren
Jinwei Zhang
Zhen Wang
Ming Ding
Ke Ding
author_sort Chungen Li
collection DOAJ
format Article
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institution OA Journals
issn 2691-3704
language English
publishDate 2024-11-01
publisher American Chemical Society
record_format Article
series JACS Au
spelling doaj-art-e4af2f80ee094493919a955d9dfb9f562025-08-20T02:31:36ZengAmerican Chemical SocietyJACS Au2691-37042024-11-014124866488210.1021/jacsau.4c00831Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACsChungen Li0Yihan Chen1Weixue Huang2Yudi Qiu3Shengjie Huang4Yang Zhou5Fengtao Zhou6Jian Xu7Xiaomei Ren8Jinwei Zhang9Zhen Wang10Ming Ding11Ke Ding12State Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaKey Laboratory of Structure-Based Drugs Design and Discovery of Ministry of Education, Shengyang Pharmaceutical University, Shenyang, ChinaInternational Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Discovery of Chinese Ministry of Education (MOE), Guangzhou City Key Laboratory of Precision Chemical Drug Development, College of Pharmacy, Jinan University, Guangzhou, ChinaInternational Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Discovery of Chinese Ministry of Education (MOE), Guangzhou City Key Laboratory of Precision Chemical Drug Development, College of Pharmacy, Jinan University, Guangzhou, ChinaInternational Cooperative Laboratory of Traditional Chinese Medicine Modernization and Innovative Drug Discovery of Chinese Ministry of Education (MOE), Guangzhou City Key Laboratory of Precision Chemical Drug Development, College of Pharmacy, Jinan University, Guangzhou, ChinaLivzon Research Institute, Livzon Pharmaceutical Group Inc., Zhuhai, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, ChinaSchool of Life Science and Technology, China Pharmaceutical University, Nanjing, ChinaState Key Laboratory of Chemical Biology, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, Shanghai, Chinahttps://doi.org/10.1021/jacsau.4c00831
spellingShingle Chungen Li
Yihan Chen
Weixue Huang
Yudi Qiu
Shengjie Huang
Yang Zhou
Fengtao Zhou
Jian Xu
Xiaomei Ren
Jinwei Zhang
Zhen Wang
Ming Ding
Ke Ding
Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
JACS Au
title Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
title_full Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
title_fullStr Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
title_full_unstemmed Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
title_short Structure-Based Design of “Head-to-Tail” Macrocyclic PROTACs
title_sort structure based design of head to tail macrocyclic protacs
url https://doi.org/10.1021/jacsau.4c00831
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