Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia

Relieving hypoxia in the tumor microenvironment (TME) promotes innate and adaptive immunity. Our previous research demonstrated that reoxygenation of the TME promotes the phagocytosis and tumor-killing functions of tumor-associated macrophages (TAMs) by upregulating pyruvate carboxylase (PCB). Howev...

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Main Authors: Shu Yuxin, Zhou Linmin, Qian Jinqin, Zhu Wei-Guo
Format: Article
Language:English
Published: China Science Publishing & Media Ltd. 2025-01-01
Series:Acta Biochimica et Biophysica Sinica
Subjects:
Online Access:https://www.sciengine.com/doi/10.3724/abbs.2025011
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author Shu Yuxin
Zhou Linmin
Qian Jinqin
Zhu Wei-Guo
author_facet Shu Yuxin
Zhou Linmin
Qian Jinqin
Zhu Wei-Guo
author_sort Shu Yuxin
collection DOAJ
description Relieving hypoxia in the tumor microenvironment (TME) promotes innate and adaptive immunity. Our previous research demonstrated that reoxygenation of the TME promotes the phagocytosis and tumor-killing functions of tumor-associated macrophages (TAMs) by upregulating pyruvate carboxylase (PCB). However, the mechanism remains obscure. In the present study, we find that versican derived from melanoma cells binds to TLR2 and activates the downstream transcription factor RelB, which transcribes PCB under normoxia. Blocking the versican-TLR2-MyD88-RelB axis not only reverses the upregulation of PCB in TAMs but also hinders the clearance of tumor cells by TAMs. Our work suggests a pathway that modulates the functions of TAMs under normoxia, which could be harnessed for strengthening anti-tumor immunity.
format Article
id doaj-art-e2c83d1b21b34cc4b3b6db28e0177ce2
institution Kabale University
issn 1672-9145
language English
publishDate 2025-01-01
publisher China Science Publishing & Media Ltd.
record_format Article
series Acta Biochimica et Biophysica Sinica
spelling doaj-art-e2c83d1b21b34cc4b3b6db28e0177ce22025-08-20T03:30:03ZengChina Science Publishing & Media Ltd.Acta Biochimica et Biophysica Sinica1672-91452025-01-015787187810.3724/abbs.202501120d259ccMelanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxiaShu Yuxin0Zhou Linmin1Qian Jinqin2Zhu Wei-Guo3["International Cancer Center, Guangdong Key Laboratory of Genome Instability and Human Disease Prevention, Department of Biochemistry and Molecular Biology, Shenzhen University Medical School, Shenzhen 518060, China","School of Basic Medical Sciences, Wannan Medical College, Wuhu 241002, China"]["School of Pharmaceutical Sciences, Shenzhen University Health Science Center, Shenzhen 518055, China"]["Department of Urology, Peking University First Hospital; Institute of Urology, Peking University; National Urological Cancer Center of China, Beijing 100034, China"]["International Cancer Center, Guangdong Key Laboratory of Genome Instability and Human Disease Prevention, Department of Biochemistry and Molecular Biology, Shenzhen University Medical School, Shenzhen 518060, China","School of Basic Medical Sciences, Wannan Medical College, Wuhu 241002, China"]Relieving hypoxia in the tumor microenvironment (TME) promotes innate and adaptive immunity. Our previous research demonstrated that reoxygenation of the TME promotes the phagocytosis and tumor-killing functions of tumor-associated macrophages (TAMs) by upregulating pyruvate carboxylase (PCB). However, the mechanism remains obscure. In the present study, we find that versican derived from melanoma cells binds to TLR2 and activates the downstream transcription factor RelB, which transcribes PCB under normoxia. Blocking the versican-TLR2-MyD88-RelB axis not only reverses the upregulation of PCB in TAMs but also hinders the clearance of tumor cells by TAMs. Our work suggests a pathway that modulates the functions of TAMs under normoxia, which could be harnessed for strengthening anti-tumor immunity.https://www.sciengine.com/doi/10.3724/abbs.2025011pyruvate carboxylasephagocytosisRelBtumor-associated macrophagesversican
spellingShingle Shu Yuxin
Zhou Linmin
Qian Jinqin
Zhu Wei-Guo
Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
Acta Biochimica et Biophysica Sinica
pyruvate carboxylase
phagocytosis
RelB
tumor-associated macrophages
versican
title Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
title_full Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
title_fullStr Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
title_full_unstemmed Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
title_short Melanoma-derived versican reactivates tumor-associated macrophages by upregulating pyruvate carboxylase through TLR2-MyD88-RelB axis under normoxia
title_sort melanoma derived versican reactivates tumor associated macrophages by upregulating pyruvate carboxylase through tlr2 myd88 relb axis under normoxia
topic pyruvate carboxylase
phagocytosis
RelB
tumor-associated macrophages
versican
url https://www.sciengine.com/doi/10.3724/abbs.2025011
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AT zhoulinmin melanomaderivedversicanreactivatestumorassociatedmacrophagesbyupregulatingpyruvatecarboxylasethroughtlr2myd88relbaxisundernormoxia
AT qianjinqin melanomaderivedversicanreactivatestumorassociatedmacrophagesbyupregulatingpyruvatecarboxylasethroughtlr2myd88relbaxisundernormoxia
AT zhuweiguo melanomaderivedversicanreactivatestumorassociatedmacrophagesbyupregulatingpyruvatecarboxylasethroughtlr2myd88relbaxisundernormoxia