Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level

Adenomyosis is a gynecological disorder characterized by the invasion of endometrial tissue into the myometrium, leading to chronic inflammation and pelvic pain. Interleukin 8 (IL-8) plays a key role in inflammation and pain sensitization in adenomyosis. Metformin, an antidiabetic agent, exerts ant...

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Main Authors: Damas Hendriansyah, Nusratuddin Abdullah, Rudy B. Leonardy, Mardiah Tahir, Samrichard Rambulangi, Firdaus Hamid
Format: Article
Language:English
Published: PAGEPress Publications 2025-04-01
Series:Italian Journal of Medicine
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Online Access:https://www.italjmed.org/ijm/article/view/1940
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author Damas Hendriansyah
Nusratuddin Abdullah
Rudy B. Leonardy
Mardiah Tahir
Samrichard Rambulangi
Firdaus Hamid
author_facet Damas Hendriansyah
Nusratuddin Abdullah
Rudy B. Leonardy
Mardiah Tahir
Samrichard Rambulangi
Firdaus Hamid
author_sort Damas Hendriansyah
collection DOAJ
description Adenomyosis is a gynecological disorder characterized by the invasion of endometrial tissue into the myometrium, leading to chronic inflammation and pelvic pain. Interleukin 8 (IL-8) plays a key role in inflammation and pain sensitization in adenomyosis. Metformin, an antidiabetic agent, exerts anti-inflammatory effects by activating adenosine monophosphate-activated protein kinase, inhibiting IL-8 production, and reducing inflammatory cell infiltration. This cohort-prospective study evaluates the effects of metformin on IL-8 levels and pain in adenomyosis patients. This cohort-prospective study in Makassar, Indonesia, included 40 women diagnosed with adenomyosis via physical examination and ultrasound examination in a polyclinic at Hasanuddin University Teaching Hospital. Participants were divided into two groups: 20 received metformin 500 mg and ibuprofen 400 mg every 8 hours for 30 days, while 20 only received ibuprofen. All statistical analyses were conducted using the Statistical Program for Social Sciences (IBM, Chicago, IL, USA). IL-8 levels increased in both groups (p=0.45). Visual Analog Scale (VAS) significantly decreased in the metformin group (p<0.001) but was not significant in the control group (p=0.06). Comparison of changes in IL-8 (p=0.13) and VAS (p=0.09) levels between the metformin and control groups was not statistically significant. This study suggests that the anti-diabetic drug metformin can also be used as an anti-inflammatory drug in adenomyosis patients as an adjunctive therapy. Further clinical trials need to be done on metformin drugs.
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spelling doaj-art-e29080d0f8bd425f8d1fe452770739452025-08-20T03:14:53ZengPAGEPress PublicationsItalian Journal of Medicine1877-93441877-93522025-04-0110.4081/itjm.2025.1940Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 levelDamas Hendriansyah0Nusratuddin Abdullah1Rudy B. Leonardy2Mardiah Tahir3Samrichard Rambulangi4Firdaus Hamid5Department of Obstetrics and Gynecology, Faculty of Medicine, Hasanuddin University, MakassarDepartment of Obstetrics and Gynecology, Faculty of Medicine, Hasanuddin University, MakassarDepartment of Obstetrics and Gynecology, Faculty of Medicine, Hasanuddin University, MakassarDepartment of Obstetrics and Gynecology, Faculty of Medicine, Hasanuddin University, MakassarDepartment of Obstetrics and Gynecology, Faculty of Medicine, Hasanuddin University, MakassarDepartment of Microbiology, Faculty of Medicine, Hasanuddin University, Makassar Adenomyosis is a gynecological disorder characterized by the invasion of endometrial tissue into the myometrium, leading to chronic inflammation and pelvic pain. Interleukin 8 (IL-8) plays a key role in inflammation and pain sensitization in adenomyosis. Metformin, an antidiabetic agent, exerts anti-inflammatory effects by activating adenosine monophosphate-activated protein kinase, inhibiting IL-8 production, and reducing inflammatory cell infiltration. This cohort-prospective study evaluates the effects of metformin on IL-8 levels and pain in adenomyosis patients. This cohort-prospective study in Makassar, Indonesia, included 40 women diagnosed with adenomyosis via physical examination and ultrasound examination in a polyclinic at Hasanuddin University Teaching Hospital. Participants were divided into two groups: 20 received metformin 500 mg and ibuprofen 400 mg every 8 hours for 30 days, while 20 only received ibuprofen. All statistical analyses were conducted using the Statistical Program for Social Sciences (IBM, Chicago, IL, USA). IL-8 levels increased in both groups (p=0.45). Visual Analog Scale (VAS) significantly decreased in the metformin group (p<0.001) but was not significant in the control group (p=0.06). Comparison of changes in IL-8 (p=0.13) and VAS (p=0.09) levels between the metformin and control groups was not statistically significant. This study suggests that the anti-diabetic drug metformin can also be used as an anti-inflammatory drug in adenomyosis patients as an adjunctive therapy. Further clinical trials need to be done on metformin drugs. https://www.italjmed.org/ijm/article/view/1940Adenomyosisinterleukin 8metformininflammationpain
spellingShingle Damas Hendriansyah
Nusratuddin Abdullah
Rudy B. Leonardy
Mardiah Tahir
Samrichard Rambulangi
Firdaus Hamid
Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
Italian Journal of Medicine
Adenomyosis
interleukin 8
metformin
inflammation
pain
title Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
title_full Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
title_fullStr Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
title_full_unstemmed Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
title_short Metformin’s therapeutic potential in adenomyosis: insights from interleukin 8 level
title_sort metformin s therapeutic potential in adenomyosis insights from interleukin 8 level
topic Adenomyosis
interleukin 8
metformin
inflammation
pain
url https://www.italjmed.org/ijm/article/view/1940
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AT mardiahtahir metforminstherapeuticpotentialinadenomyosisinsightsfrominterleukin8level
AT samrichardrambulangi metforminstherapeuticpotentialinadenomyosisinsightsfrominterleukin8level
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