Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis

A new series of quinoline hydrazone derivatives and their metal complexes have been synthesized and their biological properties have been evaluated against Mycobacterium tuberculosis (H37 RV strain). Most of the newly synthesized compounds displayed 100% inhibitory activity at a concentration of 6.2...

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Main Authors: Mustapha C. Mandewale, Bapu Thorat, Dnyaneshwar Shelke, Ramesh Yamgar
Format: Article
Language:English
Published: Wiley 2015-01-01
Series:Bioinorganic Chemistry and Applications
Online Access:http://dx.doi.org/10.1155/2015/153015
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author Mustapha C. Mandewale
Bapu Thorat
Dnyaneshwar Shelke
Ramesh Yamgar
author_facet Mustapha C. Mandewale
Bapu Thorat
Dnyaneshwar Shelke
Ramesh Yamgar
author_sort Mustapha C. Mandewale
collection DOAJ
description A new series of quinoline hydrazone derivatives and their metal complexes have been synthesized and their biological properties have been evaluated against Mycobacterium tuberculosis (H37 RV strain). Most of the newly synthesized compounds displayed 100% inhibitory activity at a concentration of 6.25–25 μg/mL, against Mycobacterium tuberculosis. Fluorescence properties of all the synthesized compounds have been studied.
format Article
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institution OA Journals
issn 1565-3633
1687-479X
language English
publishDate 2015-01-01
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record_format Article
series Bioinorganic Chemistry and Applications
spelling doaj-art-e0a70b4b5f25466dbdb9fd8618830e232025-08-20T02:21:29ZengWileyBioinorganic Chemistry and Applications1565-36331687-479X2015-01-01201510.1155/2015/153015153015Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosisMustapha C. Mandewale0Bapu Thorat1Dnyaneshwar Shelke2Ramesh Yamgar3P.G. and Research Centre, Department of Chemistry, Government of Maharashtra, Ismail Yusuf College of Arts, Science and Commerce, Jogeshwari (East), Mumbai 400 060, IndiaP.G. and Research Centre, Department of Chemistry, Government of Maharashtra, Ismail Yusuf College of Arts, Science and Commerce, Jogeshwari (East), Mumbai 400 060, IndiaP.G. and Research Centre, Department of Chemistry, Government of Maharashtra, Ismail Yusuf College of Arts, Science and Commerce, Jogeshwari (East), Mumbai 400 060, IndiaDepartment of Chemistry, Chikitsak Samuha’s Patkar-Varde College of Arts, Science and Commerce, Goregaon (West), Mumbai 400 062, IndiaA new series of quinoline hydrazone derivatives and their metal complexes have been synthesized and their biological properties have been evaluated against Mycobacterium tuberculosis (H37 RV strain). Most of the newly synthesized compounds displayed 100% inhibitory activity at a concentration of 6.25–25 μg/mL, against Mycobacterium tuberculosis. Fluorescence properties of all the synthesized compounds have been studied.http://dx.doi.org/10.1155/2015/153015
spellingShingle Mustapha C. Mandewale
Bapu Thorat
Dnyaneshwar Shelke
Ramesh Yamgar
Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
Bioinorganic Chemistry and Applications
title Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
title_full Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
title_fullStr Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
title_full_unstemmed Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
title_short Synthesis and Biological Evaluation of New Hydrazone Derivatives of Quinoline and Their Cu(II) and Zn(II) Complexes against Mycobacterium tuberculosis
title_sort synthesis and biological evaluation of new hydrazone derivatives of quinoline and their cu ii and zn ii complexes against mycobacterium tuberculosis
url http://dx.doi.org/10.1155/2015/153015
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