TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life

TrYbe® is an Fc-free therapeutic antibody format, capable of engaging up to three targets simultaneously, with long in vivo half-life conferred by albumin binding. This format is shown by small-angle X-ray scattering to be conformationally flexible with favorable ‘reach’ properties. We demonstrate t...

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Main Authors: Emma Davé, Oliver Durrant, Neha Dhami, Joanne Compson, Janice Broadbridge, Sophie Archer, Asher Maroof, Kevin Whale, Karelle Menochet, Pierre Bonnaillie, Emily Barry, Gavin Wild, Claude Peerboom, Pallavi Bhatta, Mark Ellis, Matthew Hinchliffe, David P. Humphreys, Sam P. Heywood
Format: Article
Language:English
Published: Taylor & Francis Group 2023-12-01
Series:mAbs
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Online Access:https://www.tandfonline.com/doi/10.1080/19420862.2022.2160229
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author Emma Davé
Oliver Durrant
Neha Dhami
Joanne Compson
Janice Broadbridge
Sophie Archer
Asher Maroof
Kevin Whale
Karelle Menochet
Pierre Bonnaillie
Emily Barry
Gavin Wild
Claude Peerboom
Pallavi Bhatta
Mark Ellis
Matthew Hinchliffe
David P. Humphreys
Sam P. Heywood
author_facet Emma Davé
Oliver Durrant
Neha Dhami
Joanne Compson
Janice Broadbridge
Sophie Archer
Asher Maroof
Kevin Whale
Karelle Menochet
Pierre Bonnaillie
Emily Barry
Gavin Wild
Claude Peerboom
Pallavi Bhatta
Mark Ellis
Matthew Hinchliffe
David P. Humphreys
Sam P. Heywood
author_sort Emma Davé
collection DOAJ
description TrYbe® is an Fc-free therapeutic antibody format, capable of engaging up to three targets simultaneously, with long in vivo half-life conferred by albumin binding. This format is shown by small-angle X-ray scattering to be conformationally flexible with favorable ‘reach’ properties. We demonstrate the format’s broad functionality by co-targeting of soluble and cell surface antigens. The benefit of monovalent target binding is illustrated by the lack of formation of large immune complexes when co-targeting multivalent antigens. TrYbes® are manufactured using standard mammalian cell culture and protein A affinity capture processes. TrYbes® have been formulated at high concentrations and have favorable drug-like properties, including stability, solubility, and low viscosity. The unique functionality and inherent developability of the TrYbe® makes it a promising multi-specific antibody fragment format for antibody therapy.
format Article
id doaj-art-da5a5f25917d459295f40b2ca83010e7
institution Kabale University
issn 1942-0862
1942-0870
language English
publishDate 2023-12-01
publisher Taylor & Francis Group
record_format Article
series mAbs
spelling doaj-art-da5a5f25917d459295f40b2ca83010e72025-08-20T03:25:53ZengTaylor & Francis GroupmAbs1942-08621942-08702023-12-0115110.1080/19420862.2022.2160229TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-lifeEmma Davé0Oliver Durrant1Neha Dhami2Joanne Compson3Janice Broadbridge4Sophie Archer5Asher Maroof6Kevin Whale7Karelle Menochet8Pierre Bonnaillie9Emily Barry10Gavin Wild11Claude Peerboom12Pallavi Bhatta13Mark Ellis14Matthew Hinchliffe15David P. Humphreys16Sam P. Heywood17Early Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKPV Supply and Technology Solutions, UCB Biopharma UK, Slough, UKPV Supply and Technology Solutions, UCB Biopharma SRL, Braine-l'Alleud, Belgium, EUEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKEarly Solutions, UCB Biopharma UK, Slough, UKTrYbe® is an Fc-free therapeutic antibody format, capable of engaging up to three targets simultaneously, with long in vivo half-life conferred by albumin binding. This format is shown by small-angle X-ray scattering to be conformationally flexible with favorable ‘reach’ properties. We demonstrate the format’s broad functionality by co-targeting of soluble and cell surface antigens. The benefit of monovalent target binding is illustrated by the lack of formation of large immune complexes when co-targeting multivalent antigens. TrYbes® are manufactured using standard mammalian cell culture and protein A affinity capture processes. TrYbes® have been formulated at high concentrations and have favorable drug-like properties, including stability, solubility, and low viscosity. The unique functionality and inherent developability of the TrYbe® makes it a promising multi-specific antibody fragment format for antibody therapy.https://www.tandfonline.com/doi/10.1080/19420862.2022.2160229TrYbe®multi-specificmonovalentFc-freetargetingmultivalent antigen
spellingShingle Emma Davé
Oliver Durrant
Neha Dhami
Joanne Compson
Janice Broadbridge
Sophie Archer
Asher Maroof
Kevin Whale
Karelle Menochet
Pierre Bonnaillie
Emily Barry
Gavin Wild
Claude Peerboom
Pallavi Bhatta
Mark Ellis
Matthew Hinchliffe
David P. Humphreys
Sam P. Heywood
TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
mAbs
TrYbe®
multi-specific
monovalent
Fc-free
targeting
multivalent antigen
title TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
title_full TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
title_fullStr TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
title_full_unstemmed TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
title_short TRYBE®: an Fc-free antibody format with three monovalent targeting arms engineered for long in vivo half-life
title_sort trybe r an fc free antibody format with three monovalent targeting arms engineered for long in vivo half life
topic TrYbe®
multi-specific
monovalent
Fc-free
targeting
multivalent antigen
url https://www.tandfonline.com/doi/10.1080/19420862.2022.2160229
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