NMR Data Analysis of Acarbose

Acarbose, an α-glucosidase inhibitor, has been widely used in the treatment of type-II diabetes due to its unique mechanism of action. In this study, comprehensive and accurate 1H and 13C NMR data of acarbose in DMSO-d6, including 1H NMR data of all hydroxyl groups of acarbose as well as 1H and 13C...

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Main Authors: LI Yujiang, ZHAO Wei, TAO Le, LU Bohua, ZHENG Guo, ZHANG Haiyan, GUO Xiaohe, ZHAO Tianzeng
Format: Article
Language:zho
Published: Science Press 2025-06-01
Series:Chinese Journal of Magnetic Resonance
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Online Access:http://121.43.60.238/bpxzz/article/2025/1000-4556/1000-4556-42-2-184.shtml
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author LI Yujiang
ZHAO Wei
TAO Le
LU Bohua
ZHENG Guo
ZHANG Haiyan
GUO Xiaohe
ZHAO Tianzeng
author_facet LI Yujiang
ZHAO Wei
TAO Le
LU Bohua
ZHENG Guo
ZHANG Haiyan
GUO Xiaohe
ZHAO Tianzeng
author_sort LI Yujiang
collection DOAJ
description Acarbose, an α-glucosidase inhibitor, has been widely used in the treatment of type-II diabetes due to its unique mechanism of action. In this study, comprehensive and accurate 1H and 13C NMR data of acarbose in DMSO-d6, including 1H NMR data of all hydroxyl groups of acarbose as well as 1H and 13C NMR data of the dual signal of C-ring α and β, were reported for the first time. The assignment of 1H and 13C NMR data was conducted using DEPT-135, 1H-1H COSY, 1H-13C HSQC, and 1H-13C HMBC techniques. The molecular structure of acarbose was confirmed, providing a reliable data basis for the safety and quality control of acarbose drugs.
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institution Kabale University
issn 1000-4556
language zho
publishDate 2025-06-01
publisher Science Press
record_format Article
series Chinese Journal of Magnetic Resonance
spelling doaj-art-d943443c07254bf5a3c7ddec2bf0c5632025-08-20T03:45:10ZzhoScience PressChinese Journal of Magnetic Resonance1000-45562025-06-0142218419410.11938/cjmr20243125NMR Data Analysis of AcarboseLI Yujiang0ZHAO Wei1TAO Le2LU Bohua3ZHENG Guo4ZHANG Haiyan5GUO Xiaohe6ZHAO Tianzeng7High&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, ChinaHigh&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, ChinaHigh&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, ChinaHigh&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, ChinaHigh&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, ChinaKey Laboratory of Natural Products, Henan Academy of Sciences, Zhengzhou, 450002, ChinaHigh&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, China1. High&New Technology Research Center of Henan Academy of Sciences, Zhengzhou, 450002, China 2. Key Laboratory of Natural Products, Henan Academy of Sciences, Zhengzhou, 450002, ChinaAcarbose, an α-glucosidase inhibitor, has been widely used in the treatment of type-II diabetes due to its unique mechanism of action. In this study, comprehensive and accurate 1H and 13C NMR data of acarbose in DMSO-d6, including 1H NMR data of all hydroxyl groups of acarbose as well as 1H and 13C NMR data of the dual signal of C-ring α and β, were reported for the first time. The assignment of 1H and 13C NMR data was conducted using DEPT-135, 1H-1H COSY, 1H-13C HSQC, and 1H-13C HMBC techniques. The molecular structure of acarbose was confirmed, providing a reliable data basis for the safety and quality control of acarbose drugs.http://121.43.60.238/bpxzz/article/2025/1000-4556/1000-4556-42-2-184.shtmlliquid-state nmrstructural assignment2d nmracarbose
spellingShingle LI Yujiang
ZHAO Wei
TAO Le
LU Bohua
ZHENG Guo
ZHANG Haiyan
GUO Xiaohe
ZHAO Tianzeng
NMR Data Analysis of Acarbose
Chinese Journal of Magnetic Resonance
liquid-state nmr
structural assignment
2d nmr
acarbose
title NMR Data Analysis of Acarbose
title_full NMR Data Analysis of Acarbose
title_fullStr NMR Data Analysis of Acarbose
title_full_unstemmed NMR Data Analysis of Acarbose
title_short NMR Data Analysis of Acarbose
title_sort nmr data analysis of acarbose
topic liquid-state nmr
structural assignment
2d nmr
acarbose
url http://121.43.60.238/bpxzz/article/2025/1000-4556/1000-4556-42-2-184.shtml
work_keys_str_mv AT liyujiang nmrdataanalysisofacarbose
AT zhaowei nmrdataanalysisofacarbose
AT taole nmrdataanalysisofacarbose
AT lubohua nmrdataanalysisofacarbose
AT zhengguo nmrdataanalysisofacarbose
AT zhanghaiyan nmrdataanalysisofacarbose
AT guoxiaohe nmrdataanalysisofacarbose
AT zhaotianzeng nmrdataanalysisofacarbose