Pharmacogenetics or predictive genetics? APOE testing blurs the lines

The integration of pharmacogenetics into personalized medicine enables the optimization of drug selection and dosage, maximizing therapeutic benefits while minimizing the risk of adverse drug reactions. The association between APOE alleles and ARIA, a known adverse reaction in Alzheimer’s disease pa...

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Main Authors: Stefania Zampatti, Cristina Peconi, Juliette Farro, Fabrizio Piras, Clelia Pellicano, Carlo Caltagirone, Emiliano Giardina
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-07-01
Series:Frontiers in Pharmacology
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Online Access:https://www.frontiersin.org/articles/10.3389/fphar.2025.1627239/full
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author Stefania Zampatti
Cristina Peconi
Juliette Farro
Fabrizio Piras
Clelia Pellicano
Carlo Caltagirone
Emiliano Giardina
Emiliano Giardina
author_facet Stefania Zampatti
Cristina Peconi
Juliette Farro
Fabrizio Piras
Clelia Pellicano
Carlo Caltagirone
Emiliano Giardina
Emiliano Giardina
author_sort Stefania Zampatti
collection DOAJ
description The integration of pharmacogenetics into personalized medicine enables the optimization of drug selection and dosage, maximizing therapeutic benefits while minimizing the risk of adverse drug reactions. The association between APOE alleles and ARIA, a known adverse reaction in Alzheimer’s disease patients treated with anti-amyloid monoclonal antibodies, has led to the inclusion of APOE genotyping among conventional pharmacogenetic tests. Given the dual role of APOE alleles, the widespread implementation of this genetic test requires caution and should be accompanied by appropriate genetic counselling. APOE genotyping is uniquely positioned at the intersection of pharmacogenetics and germline testing: it provides insight not only into drug safety (specifically the risk of Amyloid-Related Imaging Abnormalities) but also into familial risk for developing Alzheimer’s disease. Carriers of risk alleles, especially homozygotes, face the highest risk and require close monitoring. While APOE genotyping can inform treatment decisions, it also raises ethical concerns due to the broader implications of disclosing genetic risk information for neurodegenerative diseases. Identifying a high-risk APOE genotype in a patient substantially impacts family members. Therefore, patients considered for treatment with anti-amyloid monoclonal antibodies should receive comprehensive pre- and post-test genetic counseling that goes beyond traditional standards, as currently provided for other peculiar tests. Such counseling ensures that patients are adequately informed about potential outcomes, psychological impacts, and familial implications. It also supports ethical decision-making and facilitates truly informed consent, helping to prevent deterministic or overly simplistic interpretations of genetic risk.
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spelling doaj-art-d3f242b07f2a471a939a3c747ea6e0542025-08-20T03:28:13ZengFrontiers Media S.A.Frontiers in Pharmacology1663-98122025-07-011610.3389/fphar.2025.16272391627239Pharmacogenetics or predictive genetics? APOE testing blurs the linesStefania Zampatti0Cristina Peconi1Juliette Farro2Fabrizio Piras3Clelia Pellicano4Carlo Caltagirone5Emiliano Giardina6Emiliano Giardina7Genomic Medicine Laboratory UILDM, IRCCS Santa Lucia Foundation, Rome, ItalyGenomic Medicine Laboratory UILDM, IRCCS Santa Lucia Foundation, Rome, ItalyGenomic Medicine Laboratory UILDM, IRCCS Santa Lucia Foundation, Rome, ItalyNeuropsychiatry Laboratory, Department of Clinical Neuroscience and Neurorehabilitation, IRCCS Santa Lucia Foundation, Rome, ItalyNeuropsychiatry Laboratory, Department of Clinical Neuroscience and Neurorehabilitation, IRCCS Santa Lucia Foundation, Rome, ItalyDepartment of Clinical and Behavioral Neurology, IRCCS Fondazione Santa Lucia, Rome, ItalyGenomic Medicine Laboratory UILDM, IRCCS Santa Lucia Foundation, Rome, ItalyDepartment of Biomedicine and Prevention, Tor Vergata University, Rome, ItalyThe integration of pharmacogenetics into personalized medicine enables the optimization of drug selection and dosage, maximizing therapeutic benefits while minimizing the risk of adverse drug reactions. The association between APOE alleles and ARIA, a known adverse reaction in Alzheimer’s disease patients treated with anti-amyloid monoclonal antibodies, has led to the inclusion of APOE genotyping among conventional pharmacogenetic tests. Given the dual role of APOE alleles, the widespread implementation of this genetic test requires caution and should be accompanied by appropriate genetic counselling. APOE genotyping is uniquely positioned at the intersection of pharmacogenetics and germline testing: it provides insight not only into drug safety (specifically the risk of Amyloid-Related Imaging Abnormalities) but also into familial risk for developing Alzheimer’s disease. Carriers of risk alleles, especially homozygotes, face the highest risk and require close monitoring. While APOE genotyping can inform treatment decisions, it also raises ethical concerns due to the broader implications of disclosing genetic risk information for neurodegenerative diseases. Identifying a high-risk APOE genotype in a patient substantially impacts family members. Therefore, patients considered for treatment with anti-amyloid monoclonal antibodies should receive comprehensive pre- and post-test genetic counseling that goes beyond traditional standards, as currently provided for other peculiar tests. Such counseling ensures that patients are adequately informed about potential outcomes, psychological impacts, and familial implications. It also supports ethical decision-making and facilitates truly informed consent, helping to prevent deterministic or overly simplistic interpretations of genetic risk.https://www.frontiersin.org/articles/10.3389/fphar.2025.1627239/fullpharmacogeneticspredictive testgenetic counsellingalzheimer diseasemonoclonal antibodiesAPOE
spellingShingle Stefania Zampatti
Cristina Peconi
Juliette Farro
Fabrizio Piras
Clelia Pellicano
Carlo Caltagirone
Emiliano Giardina
Emiliano Giardina
Pharmacogenetics or predictive genetics? APOE testing blurs the lines
Frontiers in Pharmacology
pharmacogenetics
predictive test
genetic counselling
alzheimer disease
monoclonal antibodies
APOE
title Pharmacogenetics or predictive genetics? APOE testing blurs the lines
title_full Pharmacogenetics or predictive genetics? APOE testing blurs the lines
title_fullStr Pharmacogenetics or predictive genetics? APOE testing blurs the lines
title_full_unstemmed Pharmacogenetics or predictive genetics? APOE testing blurs the lines
title_short Pharmacogenetics or predictive genetics? APOE testing blurs the lines
title_sort pharmacogenetics or predictive genetics apoe testing blurs the lines
topic pharmacogenetics
predictive test
genetic counselling
alzheimer disease
monoclonal antibodies
APOE
url https://www.frontiersin.org/articles/10.3389/fphar.2025.1627239/full
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