Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide

Aryl iodides, bromides and vinyl-triflates are usually converted in high to excellent yields into the corresponding carboxylic acids through a parallel palladium-catalyzed hydroxycarbonylation using lithium formate and acetic anhydride as external condensed source of carbon monoxide.

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Main Authors: Antonia Iazzetti, Giancarlo Fabrizi, Yuri Gazzilli, Antonella Goggiamani, Federico Marrone, Chen Shen, Roberta Zoppoli
Format: Article
Language:English
Published: MDPI AG 2025-08-01
Series:Molecules
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Online Access:https://www.mdpi.com/1420-3049/30/15/3298
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author Antonia Iazzetti
Giancarlo Fabrizi
Yuri Gazzilli
Antonella Goggiamani
Federico Marrone
Chen Shen
Roberta Zoppoli
author_facet Antonia Iazzetti
Giancarlo Fabrizi
Yuri Gazzilli
Antonella Goggiamani
Federico Marrone
Chen Shen
Roberta Zoppoli
author_sort Antonia Iazzetti
collection DOAJ
description Aryl iodides, bromides and vinyl-triflates are usually converted in high to excellent yields into the corresponding carboxylic acids through a parallel palladium-catalyzed hydroxycarbonylation using lithium formate and acetic anhydride as external condensed source of carbon monoxide.
format Article
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institution Kabale University
issn 1420-3049
language English
publishDate 2025-08-01
publisher MDPI AG
record_format Article
series Molecules
spelling doaj-art-d2ac81f36feb446ab337d4e51985a06d2025-08-20T03:36:22ZengMDPI AGMolecules1420-30492025-08-013015329810.3390/molecules30153298Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon MonoxideAntonia Iazzetti0Giancarlo Fabrizi1Yuri Gazzilli2Antonella Goggiamani3Federico Marrone4Chen Shen5Roberta Zoppoli6Dipartimento di Scienze Biotecnologiche di Base, Cliniche Intensivologiche e Perioperatorie, Università Cattolica del Sacro Cuore, L. go Francesco Vito 1, 00168 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyDipartimento di Chimica e Tecnologie del Farmaco, Sapienza, Università di Roma, P. le A. Moro 5, 00185 Rome, ItalyAryl iodides, bromides and vinyl-triflates are usually converted in high to excellent yields into the corresponding carboxylic acids through a parallel palladium-catalyzed hydroxycarbonylation using lithium formate and acetic anhydride as external condensed source of carbon monoxide.https://www.mdpi.com/1420-3049/30/15/3298palladium catalysiscarbon monoxidecarboxylic acidcombinatorial chemistry
spellingShingle Antonia Iazzetti
Giancarlo Fabrizi
Yuri Gazzilli
Antonella Goggiamani
Federico Marrone
Chen Shen
Roberta Zoppoli
Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
Molecules
palladium catalysis
carbon monoxide
carboxylic acid
combinatorial chemistry
title Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
title_full Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
title_fullStr Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
title_full_unstemmed Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
title_short Parallel Palladium-Catalyzed Synthesis of Carboxylic Acids from Aryl Iodides, Bromides, and Vinyl Triflates Using Acetic Anhydride and Formate Anion as an External Condensed Source of Carbon Monoxide
title_sort parallel palladium catalyzed synthesis of carboxylic acids from aryl iodides bromides and vinyl triflates using acetic anhydride and formate anion as an external condensed source of carbon monoxide
topic palladium catalysis
carbon monoxide
carboxylic acid
combinatorial chemistry
url https://www.mdpi.com/1420-3049/30/15/3298
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