<i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration

<b>Background/Objectives</b>: <i>Corema album</i> berries are edible fruits from the Iberian Atlantic coast, characterized by a rich polyphenolic composition, which endows their juice with potential protective effects against neurodegeneration. This study aimed to evaluate th...

Full description

Saved in:
Bibliographic Details
Main Authors: Antonio Canoyra, Carmen Martín-Cordero, Dolores Muñoz-Mingarro, Antonio J. León-González, Richard B. Parsons, Nuria Acero
Format: Article
Language:English
Published: MDPI AG 2024-11-01
Series:Pharmaceuticals
Subjects:
Online Access:https://www.mdpi.com/1424-8247/17/11/1535
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850267166763384832
author Antonio Canoyra
Carmen Martín-Cordero
Dolores Muñoz-Mingarro
Antonio J. León-González
Richard B. Parsons
Nuria Acero
author_facet Antonio Canoyra
Carmen Martín-Cordero
Dolores Muñoz-Mingarro
Antonio J. León-González
Richard B. Parsons
Nuria Acero
author_sort Antonio Canoyra
collection DOAJ
description <b>Background/Objectives</b>: <i>Corema album</i> berries are edible fruits from the Iberian Atlantic coast, characterized by a rich polyphenolic composition, which endows their juice with potential protective effects against neurodegeneration. This study aimed to evaluate the potential of the relatively lesser-known <i>C. album</i> berries as a novel neuroprotective agent against neurodegenerative diseases. <b>Methods</b>: The phenolic compounds of the juice were characterized using UHPLC-HRMS (Orbitrap). The SH-SY5Y neuroblastoma line was used to determine the preventive effect of the juice against H<sub>2</sub>O<sub>2</sub>-induced oxidative stress. Furthermore, neuronal cells were differentiated into dopaminergic and cholinergic lines and exposed to 6-hydroxydopamine and okadaic acid, respectively, to simulate in vitro models of Parkinson’s disease and Alzheimer’s disease. The ability of the juice to enhance neuronal viability under toxic conditions was examined. Additionally, its inhibitory effects on neuroprotective-related enzymes, including MAO-A and MAO-B, were assessed in vitro. <b>Results:</b> Phytochemical characterization reveals that 5-<i>O</i>-caffeoylquinic acid constitutes 80% of the total phenolic compounds. Higher concentrations of the juice effectively protected both differentiated and undifferentiated SH-SY5Y cells from H<sub>2</sub>O<sub>2</sub>-induced oxidative damage, reducing oxidative stress by approximately 20% and suggesting a dose-dependent mechanism. Moreover, the presence of the juice significantly enhanced the viability of dopaminergic and cholinergic cells exposed to neurotoxic agents. In vitro, the juice inhibited the activity of MAO-A (IC<sub>50</sub> = 87.21 µg/mL) and MAO-B (IC<sub>50</sub> = 56.50 µg/mL). <b>Conclusions</b>: While these findings highlight <i>C. album</i> berries as a promising neuroprotective agent, further research is required to elucidate its neuroprotective mechanisms in cell and animal models and, ultimately, in human trials.
format Article
id doaj-art-d1f50cfc5a7d4e1fa82cf727de734445
institution OA Journals
issn 1424-8247
language English
publishDate 2024-11-01
publisher MDPI AG
record_format Article
series Pharmaceuticals
spelling doaj-art-d1f50cfc5a7d4e1fa82cf727de7344452025-08-20T01:53:54ZengMDPI AGPharmaceuticals1424-82472024-11-011711153510.3390/ph17111535<i>Corema album</i> Berry Juice as a Protective Agent Against NeurodegenerationAntonio Canoyra0Carmen Martín-Cordero1Dolores Muñoz-Mingarro2Antonio J. León-González3Richard B. Parsons4Nuria Acero5Pharmaceutical and Health Science Department, Pharmacy Faculty, San Pablo-CEU University, CEU Universities, Urbanización Montepríncipe Boadilla del Monte, 28660 Madrid, SpainDepartment of Pharmacology, Faculty of Pharmacy, University of Seville, C/P. García González, 2, 41012 Seville, SpainChemistry and Biochemistry Department, Pharmacy Faculty, San Pablo-CEU University, CEU Universities, Urbanización Montepríncipe, Boadilla del Monte, 28668 Madrid, SpainDepartment of Pharmacology, Faculty of Pharmacy, University of Seville, C/P. García González, 2, 41012 Seville, SpainKing’s College London, Institute of Pharmaceutical Sciences, 150 Stamford Street, London SE1 9NH, UKPharmaceutical and Health Science Department, Pharmacy Faculty, San Pablo-CEU University, CEU Universities, Urbanización Montepríncipe Boadilla del Monte, 28660 Madrid, Spain<b>Background/Objectives</b>: <i>Corema album</i> berries are edible fruits from the Iberian Atlantic coast, characterized by a rich polyphenolic composition, which endows their juice with potential protective effects against neurodegeneration. This study aimed to evaluate the potential of the relatively lesser-known <i>C. album</i> berries as a novel neuroprotective agent against neurodegenerative diseases. <b>Methods</b>: The phenolic compounds of the juice were characterized using UHPLC-HRMS (Orbitrap). The SH-SY5Y neuroblastoma line was used to determine the preventive effect of the juice against H<sub>2</sub>O<sub>2</sub>-induced oxidative stress. Furthermore, neuronal cells were differentiated into dopaminergic and cholinergic lines and exposed to 6-hydroxydopamine and okadaic acid, respectively, to simulate in vitro models of Parkinson’s disease and Alzheimer’s disease. The ability of the juice to enhance neuronal viability under toxic conditions was examined. Additionally, its inhibitory effects on neuroprotective-related enzymes, including MAO-A and MAO-B, were assessed in vitro. <b>Results:</b> Phytochemical characterization reveals that 5-<i>O</i>-caffeoylquinic acid constitutes 80% of the total phenolic compounds. Higher concentrations of the juice effectively protected both differentiated and undifferentiated SH-SY5Y cells from H<sub>2</sub>O<sub>2</sub>-induced oxidative damage, reducing oxidative stress by approximately 20% and suggesting a dose-dependent mechanism. Moreover, the presence of the juice significantly enhanced the viability of dopaminergic and cholinergic cells exposed to neurotoxic agents. In vitro, the juice inhibited the activity of MAO-A (IC<sub>50</sub> = 87.21 µg/mL) and MAO-B (IC<sub>50</sub> = 56.50 µg/mL). <b>Conclusions</b>: While these findings highlight <i>C. album</i> berries as a promising neuroprotective agent, further research is required to elucidate its neuroprotective mechanisms in cell and animal models and, ultimately, in human trials.https://www.mdpi.com/1424-8247/17/11/1535<i>Corema album</i>oxidative stressneuroprotectiveberriesphenolsAlzheimer’s disease
spellingShingle Antonio Canoyra
Carmen Martín-Cordero
Dolores Muñoz-Mingarro
Antonio J. León-González
Richard B. Parsons
Nuria Acero
<i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
Pharmaceuticals
<i>Corema album</i>
oxidative stress
neuroprotective
berries
phenols
Alzheimer’s disease
title <i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
title_full <i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
title_fullStr <i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
title_full_unstemmed <i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
title_short <i>Corema album</i> Berry Juice as a Protective Agent Against Neurodegeneration
title_sort i corema album i berry juice as a protective agent against neurodegeneration
topic <i>Corema album</i>
oxidative stress
neuroprotective
berries
phenols
Alzheimer’s disease
url https://www.mdpi.com/1424-8247/17/11/1535
work_keys_str_mv AT antoniocanoyra icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration
AT carmenmartincordero icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration
AT doloresmunozmingarro icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration
AT antoniojleongonzalez icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration
AT richardbparsons icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration
AT nuriaacero icoremaalbumiberryjuiceasaprotectiveagentagainstneurodegeneration