The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential

The global prevalence of type 2 diabetes mellitus (T2DM) necessitates the exploration of novel therapeutic approaches to mitigate its complex molecular pathogenesis. This review investigates the potential role of genistein, a prominent isoflavone derived from soybeans, in the management of T2DM. Rec...

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Main Authors: Mateusz Kciuk, Weronika Kruczkowska, Katarzyna Wanke, Julia Gałęziewska, Damian Kołat, Somdutt Mujwar, Renata Kontek
Format: Article
Language:English
Published: MDPI AG 2025-02-01
Series:Molecules
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Online Access:https://www.mdpi.com/1420-3049/30/5/1068
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author Mateusz Kciuk
Weronika Kruczkowska
Katarzyna Wanke
Julia Gałęziewska
Damian Kołat
Somdutt Mujwar
Renata Kontek
author_facet Mateusz Kciuk
Weronika Kruczkowska
Katarzyna Wanke
Julia Gałęziewska
Damian Kołat
Somdutt Mujwar
Renata Kontek
author_sort Mateusz Kciuk
collection DOAJ
description The global prevalence of type 2 diabetes mellitus (T2DM) necessitates the exploration of novel therapeutic approaches to mitigate its complex molecular pathogenesis. This review investigates the potential role of genistein, a prominent isoflavone derived from soybeans, in the management of T2DM. Recognized for its selective estrogen receptor modulator (SERM) activity, genistein exerts a multifaceted influence on key intracellular signaling pathways, which are crucial in regulating cell proliferation, apoptosis, and insulin signaling. Genistein’s anti-inflammatory, anti-oxidant, and metabolic regulatory properties position it as a promising candidate for T2DM intervention. This review synthesizes current research spanning preclinical studies and clinical trials, emphasizing genistein’s impact on insulin sensitivity, glucose metabolism, and inflammatory markers. Additionally, this review addresses genistein’s bioavailability, safety, and potential influence on gut microbiota composition. By consolidating these findings, this review aims to provide a comprehensive understanding of genistein’s therapeutic potential in T2DM management, offering valuable insights for future research and clinical practice.
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series Molecules
spelling doaj-art-cf3dc13bc8e54c5bb5bab4bdb383cba42025-08-20T02:06:12ZengMDPI AGMolecules1420-30492025-02-01305106810.3390/molecules30051068The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic PotentialMateusz Kciuk0Weronika Kruczkowska1Katarzyna Wanke2Julia Gałęziewska3Damian Kołat4Somdutt Mujwar5Renata Kontek6Department of Molecular Biotechnology and Genetics, Univeristy of Lodz, Banacha 12/16, 90-237 Lodz, PolandDepartment of Functional Genomics, Faculty of Medicine, Medical University of Lodz, Żeligowskiego 7/9, 90-752 Lodz, PolandDepartment of Molecular Biotechnology and Genetics, Univeristy of Lodz, Banacha 12/16, 90-237 Lodz, PolandDepartment of Functional Genomics, Faculty of Medicine, Medical University of Lodz, Żeligowskiego 7/9, 90-752 Lodz, PolandDepartment of Functional Genomics, Faculty of Medicine, Medical University of Lodz, Żeligowskiego 7/9, 90-752 Lodz, PolandChitkara College of Pharmacy, Chitkara University, Rajpura 140401, Punjab, IndiaDepartment of Molecular Biotechnology and Genetics, Univeristy of Lodz, Banacha 12/16, 90-237 Lodz, PolandThe global prevalence of type 2 diabetes mellitus (T2DM) necessitates the exploration of novel therapeutic approaches to mitigate its complex molecular pathogenesis. This review investigates the potential role of genistein, a prominent isoflavone derived from soybeans, in the management of T2DM. Recognized for its selective estrogen receptor modulator (SERM) activity, genistein exerts a multifaceted influence on key intracellular signaling pathways, which are crucial in regulating cell proliferation, apoptosis, and insulin signaling. Genistein’s anti-inflammatory, anti-oxidant, and metabolic regulatory properties position it as a promising candidate for T2DM intervention. This review synthesizes current research spanning preclinical studies and clinical trials, emphasizing genistein’s impact on insulin sensitivity, glucose metabolism, and inflammatory markers. Additionally, this review addresses genistein’s bioavailability, safety, and potential influence on gut microbiota composition. By consolidating these findings, this review aims to provide a comprehensive understanding of genistein’s therapeutic potential in T2DM management, offering valuable insights for future research and clinical practice.https://www.mdpi.com/1420-3049/30/5/1068anti-oxidantbioavailabilitygenisteinmetabolic diseasenatural producttype 2 diabetes mellitus
spellingShingle Mateusz Kciuk
Weronika Kruczkowska
Katarzyna Wanke
Julia Gałęziewska
Damian Kołat
Somdutt Mujwar
Renata Kontek
The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
Molecules
anti-oxidant
bioavailability
genistein
metabolic disease
natural product
type 2 diabetes mellitus
title The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
title_full The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
title_fullStr The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
title_full_unstemmed The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
title_short The Role of Genistein in Type 2 Diabetes and Beyond: Mechanisms and Therapeutic Potential
title_sort role of genistein in type 2 diabetes and beyond mechanisms and therapeutic potential
topic anti-oxidant
bioavailability
genistein
metabolic disease
natural product
type 2 diabetes mellitus
url https://www.mdpi.com/1420-3049/30/5/1068
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