Synthesis, biological evaluation and clinical trials of Cereblon-based PROTACs

Abstract PROteolysis-Targeting Chimeras (PROTACs) are an emerging class of molecules capable of inducing a forced approximation between a protein of interest (POI) and an E3 ligase enzyme (e.g., Cereblon), leading to the degradation of the POI by the cell’s own machinery. Although in early stages of...

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Bibliographic Details
Main Authors: André T. S. Vicente, Sara P. S. P. Moura, Jorge A. R. Salvador
Format: Article
Language:English
Published: Nature Portfolio 2025-07-01
Series:Communications Chemistry
Online Access:https://doi.org/10.1038/s42004-025-01598-9
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