Mitochondrial metabolism and cancer therapeutic innovation

Abstract Mitochondria are dynamic organelles that are essential for cellular energy generation, metabolic regulation, and signal transduction. Their structural complexity enables adaptive responses to diverse physiological demands. In cancer, mitochondria orchestrate multiple cellular processes crit...

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Main Authors: Hongxiang Du, Tianhan Xu, Sihui Yu, Sufang Wu, Jiawen Zhang
Format: Article
Language:English
Published: Nature Publishing Group 2025-08-01
Series:Signal Transduction and Targeted Therapy
Online Access:https://doi.org/10.1038/s41392-025-02311-x
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author Hongxiang Du
Tianhan Xu
Sihui Yu
Sufang Wu
Jiawen Zhang
author_facet Hongxiang Du
Tianhan Xu
Sihui Yu
Sufang Wu
Jiawen Zhang
author_sort Hongxiang Du
collection DOAJ
description Abstract Mitochondria are dynamic organelles that are essential for cellular energy generation, metabolic regulation, and signal transduction. Their structural complexity enables adaptive responses to diverse physiological demands. In cancer, mitochondria orchestrate multiple cellular processes critical to tumor development. Metabolic reprogramming enables cancer cells to exploit aerobic glycolysis, glutamine metabolism, and lipid alterations, supporting uncontrolled growth, survival, and treatment resistance. Genetic and epigenetic alterations in mitochondrial and nuclear DNA disrupt oxidative phosphorylation, tricarboxylic acid cycle dynamics, and redox homeostasis, driving oncogenic progression. Mitochondrial dysfunction in tumors is highly heterogeneous, influencing disease phenotypes and treatment responses across cancer types. Within the tumor microenvironment, mitochondria profoundly impact immune responses by modulating T-cell survival and function, macrophage polarization, NK cell cytotoxicity, and neutrophil activation. They also mediate stromal cell functions, particularly in cancer-associated fibroblasts and tumor endothelial cells. Although targeting mitochondrial function represents a promising therapeutic strategy, mitochondrial heterogeneity and adaptive resistance mechanisms complicate interventional approaches. Advances in mitochondrial genome editing, proteomics, and circulating mitochondrial DNA analysis have enhanced tumor diagnostic precision. This review synthesizes the developmental landscape of mitochondrial research in cancer, comprehensively summarizing mitochondrial structural dynamics, metabolic plasticity, signaling networks, and interactions with the tumor microenvironment. Finally, we discuss the translational challenges in developing effective mitochondria-based cancer interventions.
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spelling doaj-art-c6dfb240c0984f23876af14046fbaea02025-08-20T03:06:09ZengNature Publishing GroupSignal Transduction and Targeted Therapy2059-36352025-08-0110113710.1038/s41392-025-02311-xMitochondrial metabolism and cancer therapeutic innovationHongxiang Du0Tianhan Xu1Sihui Yu2Sufang Wu3Jiawen Zhang4Department of Obstetrics and Gynecology, Shanghai General Hospital, Shanghai Jiao Tong University School of MedicineDepartment of Obstetrics and Gynecology, Shanghai General Hospital, Shanghai Jiao Tong University School of MedicineDepartment of Obstetrics and Gynecology, Zhongshan Hospital, Fudan UniversityDepartment of Obstetrics and Gynecology, Shanghai General Hospital, Shanghai Jiao Tong University School of MedicineDepartment of Obstetrics and Gynecology, Shanghai General Hospital, Shanghai Jiao Tong University School of MedicineAbstract Mitochondria are dynamic organelles that are essential for cellular energy generation, metabolic regulation, and signal transduction. Their structural complexity enables adaptive responses to diverse physiological demands. In cancer, mitochondria orchestrate multiple cellular processes critical to tumor development. Metabolic reprogramming enables cancer cells to exploit aerobic glycolysis, glutamine metabolism, and lipid alterations, supporting uncontrolled growth, survival, and treatment resistance. Genetic and epigenetic alterations in mitochondrial and nuclear DNA disrupt oxidative phosphorylation, tricarboxylic acid cycle dynamics, and redox homeostasis, driving oncogenic progression. Mitochondrial dysfunction in tumors is highly heterogeneous, influencing disease phenotypes and treatment responses across cancer types. Within the tumor microenvironment, mitochondria profoundly impact immune responses by modulating T-cell survival and function, macrophage polarization, NK cell cytotoxicity, and neutrophil activation. They also mediate stromal cell functions, particularly in cancer-associated fibroblasts and tumor endothelial cells. Although targeting mitochondrial function represents a promising therapeutic strategy, mitochondrial heterogeneity and adaptive resistance mechanisms complicate interventional approaches. Advances in mitochondrial genome editing, proteomics, and circulating mitochondrial DNA analysis have enhanced tumor diagnostic precision. This review synthesizes the developmental landscape of mitochondrial research in cancer, comprehensively summarizing mitochondrial structural dynamics, metabolic plasticity, signaling networks, and interactions with the tumor microenvironment. Finally, we discuss the translational challenges in developing effective mitochondria-based cancer interventions.https://doi.org/10.1038/s41392-025-02311-x
spellingShingle Hongxiang Du
Tianhan Xu
Sihui Yu
Sufang Wu
Jiawen Zhang
Mitochondrial metabolism and cancer therapeutic innovation
Signal Transduction and Targeted Therapy
title Mitochondrial metabolism and cancer therapeutic innovation
title_full Mitochondrial metabolism and cancer therapeutic innovation
title_fullStr Mitochondrial metabolism and cancer therapeutic innovation
title_full_unstemmed Mitochondrial metabolism and cancer therapeutic innovation
title_short Mitochondrial metabolism and cancer therapeutic innovation
title_sort mitochondrial metabolism and cancer therapeutic innovation
url https://doi.org/10.1038/s41392-025-02311-x
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AT jiawenzhang mitochondrialmetabolismandcancertherapeuticinnovation