Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach

Objectives. We hereby describe an improvement of a previously developed quantification technique for polysorbate 80 in biopharmaceutical formulations (darbepoetin alfa and eculizumab) and report the validation of the new approach.Methods. Polysorbate was isolated from analyte samples by protein prec...

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Main Authors: A. S. Seregin, N. V. Orlova, A. D. Askretkov, D. I. Zybin, Yu. A. Seregin
Format: Article
Language:Russian
Published: MIREA - Russian Technological University 2020-07-01
Series:Тонкие химические технологии
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Online Access:https://www.finechem-mirea.ru/jour/article/view/1625
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author A. S. Seregin
N. V. Orlova
A. D. Askretkov
D. I. Zybin
Yu. A. Seregin
author_facet A. S. Seregin
N. V. Orlova
A. D. Askretkov
D. I. Zybin
Yu. A. Seregin
author_sort A. S. Seregin
collection DOAJ
description Objectives. We hereby describe an improvement of a previously developed quantification technique for polysorbate 80 in biopharmaceutical formulations (darbepoetin alfa and eculizumab) and report the validation of the new approach.Methods. Polysorbate was isolated from analyte samples by protein precipitation using an organic solvent, followed by supernatant evaporation in vacuum. Polysorbate was derivatized using a ferric thiocyanate reagent and extracted into an organic phase; the relevant optical density measurements were performed.Results. We established the optimal conditions for each step of the analysis procedure. The accuracy was 97–102% in the tested analytical range, the relative standard deviation did not exceed 5%, and the limit of quantification was 0.01 mg/mL.Conclusions. The reported approach is highly sensitive; polysorbate isolation and quantification do not depend on the matrix or, most importantly, the protein.
format Article
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institution DOAJ
issn 2410-6593
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language Russian
publishDate 2020-07-01
publisher MIREA - Russian Technological University
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series Тонкие химические технологии
spelling doaj-art-c06d532a15bc476a8561ddd4150b60922025-08-20T03:23:07ZrusMIREA - Russian Technological UniversityТонкие химические технологии2410-65932686-75752020-07-01153707710.32362/2410-6593-2020-15-3-70-771596Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approachA. S. Seregin0N. V. Orlova1A. D. Askretkov2D. I. Zybin3Yu. A. Seregin4Scientific Center “Kurchatov Institute,” Research Institute for Genetics and Selection of Industrial MicroorganismsScientific Center “Kurchatov Institute,” Research Institute for Genetics and Selection of Industrial MicroorganismsPHARMAPARKPHARMAPARKScientific Center “Kurchatov Institute,” Research Institute for Genetics and Selection of Industrial MicroorganismsObjectives. We hereby describe an improvement of a previously developed quantification technique for polysorbate 80 in biopharmaceutical formulations (darbepoetin alfa and eculizumab) and report the validation of the new approach.Methods. Polysorbate was isolated from analyte samples by protein precipitation using an organic solvent, followed by supernatant evaporation in vacuum. Polysorbate was derivatized using a ferric thiocyanate reagent and extracted into an organic phase; the relevant optical density measurements were performed.Results. We established the optimal conditions for each step of the analysis procedure. The accuracy was 97–102% in the tested analytical range, the relative standard deviation did not exceed 5%, and the limit of quantification was 0.01 mg/mL.Conclusions. The reported approach is highly sensitive; polysorbate isolation and quantification do not depend on the matrix or, most importantly, the protein.https://www.finechem-mirea.ru/jour/article/view/1625validationdarbepoetin alfaeculizumabpolysorbateprecipitationferric thiocyanate
spellingShingle A. S. Seregin
N. V. Orlova
A. D. Askretkov
D. I. Zybin
Yu. A. Seregin
Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
Тонкие химические технологии
validation
darbepoetin alfa
eculizumab
polysorbate
precipitation
ferric thiocyanate
title Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
title_full Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
title_fullStr Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
title_full_unstemmed Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
title_short Quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
title_sort quantification of polysorbate 80 in biopharmaceutical formulations implementing an optimized colorimetric approach
topic validation
darbepoetin alfa
eculizumab
polysorbate
precipitation
ferric thiocyanate
url https://www.finechem-mirea.ru/jour/article/view/1625
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AT adaskretkov quantificationofpolysorbate80inbiopharmaceuticalformulationsimplementinganoptimizedcolorimetricapproach
AT dizybin quantificationofpolysorbate80inbiopharmaceuticalformulationsimplementinganoptimizedcolorimetricapproach
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