MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION

The review is devoted to modern pharmaceutical treatment of pulmonary arterial hypertension (PAH). In 1970-80s, it was based on high-dose calcium antagonists, CAs (e.g., nifedipine 240 mg/d), which were effective only in some patients with primary (idiopathic) PAH. CAs were combined with digoxin, in...

Full description

Saved in:
Bibliographic Details
Main Authors: D. V. Preobrazhensky, B. A. Sidorenko, S. A. Pataraya, T. A. Batyraliev, Z. A. Niyazova-Karben, Mesut Ishlek
Format: Article
Language:Russian
Published: «FIRMA «SILICEA» LLC 2009-12-01
Series:Российский кардиологический журнал
Subjects:
Online Access:https://russjcardiol.elpub.ru/jour/article/view/1409
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849341478851051520
author D. V. Preobrazhensky
B. A. Sidorenko
S. A. Pataraya
T. A. Batyraliev
Z. A. Niyazova-Karben
Mesut Ishlek
author_facet D. V. Preobrazhensky
B. A. Sidorenko
S. A. Pataraya
T. A. Batyraliev
Z. A. Niyazova-Karben
Mesut Ishlek
author_sort D. V. Preobrazhensky
collection DOAJ
description The review is devoted to modern pharmaceutical treatment of pulmonary arterial hypertension (PAH). In 1970-80s, it was based on high-dose calcium antagonists, CAs (e.g., nifedipine 240 mg/d), which were effective only in some patients with primary (idiopathic) PAH. CAs were combined with digoxin, indirect anticoagulants and oxygen. In 1990s, PAH therapy included prostanoids, endothelin receptor (ER) blockers and phosphodiesterase (PDE) inhibitors, which are more selective pulmonary vasodilatators than CAs, and therefore are safer for long-term treatment. Prospective studies have demonstrated that continuous intravenous infusion of epoprostenol and ET receptor blocker bosentan treatment improve survival of PAH patients receiving traditional therapy. Clinical effectiveness of epoprostenol is similar to that of subcutaneously administered trepostinil, and bosentan is similar to PDE inhibitor Type 5 sildenafil. Bosentan increases the effectiveness of intravenous epoprostenol and inhaled trepostinil.
format Article
id doaj-art-be849ca8d18d45629d9bfb4c7d225b54
institution Kabale University
issn 1560-4071
2618-7620
language Russian
publishDate 2009-12-01
publisher «FIRMA «SILICEA» LLC
record_format Article
series Российский кардиологический журнал
spelling doaj-art-be849ca8d18d45629d9bfb4c7d225b542025-08-20T03:43:37Zrus«FIRMA «SILICEA» LLCРоссийский кардиологический журнал1560-40712618-76202009-12-010669791197MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSIOND. V. Preobrazhensky0B. A. Sidorenko1S. A. Pataraya2T. A. Batyraliev3Z. A. Niyazova-Karben4Mesut Ishlek5Учебно-научный медицинский центр Управления делами Президента Российской Федерации, МоскваУчебно-научный медицинский центр Управления делами Президента Российской Федерации, МоскваУчебно-научный медицинский центр Управления делами Президента Российской Федерации, МоскваМедицинский центр имени Сани Конукоглы и Университет, Газиантеп, ТурцияМедицинский центр имени Сани Конукоглы и Университет, Газиантеп, ТурцияМедицинский центр имени Сани Конукоглы и Университет, Газиантеп, ТурцияThe review is devoted to modern pharmaceutical treatment of pulmonary arterial hypertension (PAH). In 1970-80s, it was based on high-dose calcium antagonists, CAs (e.g., nifedipine 240 mg/d), which were effective only in some patients with primary (idiopathic) PAH. CAs were combined with digoxin, indirect anticoagulants and oxygen. In 1990s, PAH therapy included prostanoids, endothelin receptor (ER) blockers and phosphodiesterase (PDE) inhibitors, which are more selective pulmonary vasodilatators than CAs, and therefore are safer for long-term treatment. Prospective studies have demonstrated that continuous intravenous infusion of epoprostenol and ET receptor blocker bosentan treatment improve survival of PAH patients receiving traditional therapy. Clinical effectiveness of epoprostenol is similar to that of subcutaneously administered trepostinil, and bosentan is similar to PDE inhibitor Type 5 sildenafil. Bosentan increases the effectiveness of intravenous epoprostenol and inhaled trepostinil.https://russjcardiol.elpub.ru/jour/article/view/1409calcium antagonistsprostanoidsepoprostenoltrepostinililoprostbosentansildenafil
spellingShingle D. V. Preobrazhensky
B. A. Sidorenko
S. A. Pataraya
T. A. Batyraliev
Z. A. Niyazova-Karben
Mesut Ishlek
MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
Российский кардиологический журнал
calcium antagonists
prostanoids
epoprostenol
trepostinil
iloprost
bosentan
sildenafil
title MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
title_full MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
title_fullStr MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
title_full_unstemmed MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
title_short MODERN PHARMACEUTICAL TREATMENT OF PULMONARY ARTERIAL HYPERTENSION
title_sort modern pharmaceutical treatment of pulmonary arterial hypertension
topic calcium antagonists
prostanoids
epoprostenol
trepostinil
iloprost
bosentan
sildenafil
url https://russjcardiol.elpub.ru/jour/article/view/1409
work_keys_str_mv AT dvpreobrazhensky modernpharmaceuticaltreatmentofpulmonaryarterialhypertension
AT basidorenko modernpharmaceuticaltreatmentofpulmonaryarterialhypertension
AT sapataraya modernpharmaceuticaltreatmentofpulmonaryarterialhypertension
AT tabatyraliev modernpharmaceuticaltreatmentofpulmonaryarterialhypertension
AT zaniyazovakarben modernpharmaceuticaltreatmentofpulmonaryarterialhypertension
AT mesutishlek modernpharmaceuticaltreatmentofpulmonaryarterialhypertension