Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer

Abstract Colorectal cancer (CRC) treatment remains challenging due to genetic heterogeneity and resistance mechanisms. To address this, we developed a drug discovery pipeline using patient-derived primary CRC cultures with diverse genomic profiles. These cultures closely resemble certain molecular c...

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Main Authors: Marcin Duleba, Eliza Zimoląg, Joanna Szuszkiewicz, Marcin Serocki, Joanna Szklarczyk, Olga Dracz, Alexander Kurzejamski, Izabella Więckowska, Marcelina Chmiel, Barbara Lipert, Katarzyna Sarad, Joanna Krawczyk, Oleksii Bryzghalov, Agata Stachowicz-Wałaszek, Karolina Pyziak, Joanna Drozdowska, Krzysztof Baczyński, Konrad Wojtowicz, Maurycy Chronowski, Krzysztof Rataj, Magdalena Otrocka, Michał Mikula, Paula Feliksiak, Rafał Dziadziuszko, Tomasz Rzymski, Andrew Thomason, Krzysztof Brzózka, Andrzej Mazan
Format: Article
Language:English
Published: Nature Portfolio 2025-07-01
Series:Scientific Reports
Online Access:https://doi.org/10.1038/s41598-025-08649-0
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author Marcin Duleba
Eliza Zimoląg
Joanna Szuszkiewicz
Marcin Serocki
Joanna Szklarczyk
Olga Dracz
Alexander Kurzejamski
Izabella Więckowska
Marcelina Chmiel
Barbara Lipert
Katarzyna Sarad
Joanna Krawczyk
Oleksii Bryzghalov
Agata Stachowicz-Wałaszek
Karolina Pyziak
Joanna Drozdowska
Krzysztof Baczyński
Konrad Wojtowicz
Maurycy Chronowski
Krzysztof Rataj
Magdalena Otrocka
Michał Mikula
Paula Feliksiak
Rafał Dziadziuszko
Tomasz Rzymski
Andrew Thomason
Krzysztof Brzózka
Andrzej Mazan
author_facet Marcin Duleba
Eliza Zimoląg
Joanna Szuszkiewicz
Marcin Serocki
Joanna Szklarczyk
Olga Dracz
Alexander Kurzejamski
Izabella Więckowska
Marcelina Chmiel
Barbara Lipert
Katarzyna Sarad
Joanna Krawczyk
Oleksii Bryzghalov
Agata Stachowicz-Wałaszek
Karolina Pyziak
Joanna Drozdowska
Krzysztof Baczyński
Konrad Wojtowicz
Maurycy Chronowski
Krzysztof Rataj
Magdalena Otrocka
Michał Mikula
Paula Feliksiak
Rafał Dziadziuszko
Tomasz Rzymski
Andrew Thomason
Krzysztof Brzózka
Andrzej Mazan
author_sort Marcin Duleba
collection DOAJ
description Abstract Colorectal cancer (CRC) treatment remains challenging due to genetic heterogeneity and resistance mechanisms. To address this, we developed a drug discovery pipeline using patient-derived primary CRC cultures with diverse genomic profiles. These cultures closely resemble certain molecular characteristics of primary and metastatic CRC, highlighting their promise as a translational platform for therapeutic evaluation. Importantly, our engineered model and patient-derived cells reflect the complexity and heterogeneity of primary tumors, not observed with standard immortalized cell lines, offering a more clinically relevant system, although further validation is needed. High-throughput screening (HTS) of 4255 compounds identified 33 with selective efficacy against CRC cells, sparing normal, healthy epithelial cells. Among the tested combinations, everolimus (mTOR inhibitor) and uprosertib (AKT inhibitor) demonstrated promising synergy at clinically relevant concentrations, with favorable therapeutic windows confirmed across tested patient-derived cultures. Notably, this synergy, revealed through advanced models, might have been overlooked in traditional immortalized cell lines, highlighting the translational advantage of patient-derived systems. Furthermore, the integration of machine learning into the HTS pipeline significantly improved scalability, cost-efficiency, and predictive accuracy. Our findings underscore the potential of patient-derived materials combined with machine learning-enhanced drug discovery to advance personalized therapies. Specifically, mTOR-AKT inhibition emerges as a promising strategy for CRC treatment, paving the way for more effective and targeted therapeutic approaches.
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institution Kabale University
issn 2045-2322
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publishDate 2025-07-01
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spelling doaj-art-bc69b090faef47cab3295ed7913b386e2025-08-20T04:02:45ZengNature PortfolioScientific Reports2045-23222025-07-0115111710.1038/s41598-025-08649-0Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancerMarcin Duleba0Eliza Zimoląg1Joanna Szuszkiewicz2Marcin Serocki3Joanna Szklarczyk4Olga Dracz5Alexander Kurzejamski6Izabella Więckowska7Marcelina Chmiel8Barbara Lipert9Katarzyna Sarad10Joanna Krawczyk11Oleksii Bryzghalov12Agata Stachowicz-Wałaszek13Karolina Pyziak14Joanna Drozdowska15Krzysztof Baczyński16Konrad Wojtowicz17Maurycy Chronowski18Krzysztof Rataj19Magdalena Otrocka20Michał Mikula21Paula Feliksiak22Rafał Dziadziuszko23Tomasz Rzymski24Andrew Thomason25Krzysztof Brzózka26Andrzej Mazan27Ryvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsArdigenArdigenArdigenArdigenMaria Skłodowska-Curie National Research Institute of OncologyMedical University of GdańskMedical University of GdańskRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsRyvu TherapeuticsAbstract Colorectal cancer (CRC) treatment remains challenging due to genetic heterogeneity and resistance mechanisms. To address this, we developed a drug discovery pipeline using patient-derived primary CRC cultures with diverse genomic profiles. These cultures closely resemble certain molecular characteristics of primary and metastatic CRC, highlighting their promise as a translational platform for therapeutic evaluation. Importantly, our engineered model and patient-derived cells reflect the complexity and heterogeneity of primary tumors, not observed with standard immortalized cell lines, offering a more clinically relevant system, although further validation is needed. High-throughput screening (HTS) of 4255 compounds identified 33 with selective efficacy against CRC cells, sparing normal, healthy epithelial cells. Among the tested combinations, everolimus (mTOR inhibitor) and uprosertib (AKT inhibitor) demonstrated promising synergy at clinically relevant concentrations, with favorable therapeutic windows confirmed across tested patient-derived cultures. Notably, this synergy, revealed through advanced models, might have been overlooked in traditional immortalized cell lines, highlighting the translational advantage of patient-derived systems. Furthermore, the integration of machine learning into the HTS pipeline significantly improved scalability, cost-efficiency, and predictive accuracy. Our findings underscore the potential of patient-derived materials combined with machine learning-enhanced drug discovery to advance personalized therapies. Specifically, mTOR-AKT inhibition emerges as a promising strategy for CRC treatment, paving the way for more effective and targeted therapeutic approaches.https://doi.org/10.1038/s41598-025-08649-0
spellingShingle Marcin Duleba
Eliza Zimoląg
Joanna Szuszkiewicz
Marcin Serocki
Joanna Szklarczyk
Olga Dracz
Alexander Kurzejamski
Izabella Więckowska
Marcelina Chmiel
Barbara Lipert
Katarzyna Sarad
Joanna Krawczyk
Oleksii Bryzghalov
Agata Stachowicz-Wałaszek
Karolina Pyziak
Joanna Drozdowska
Krzysztof Baczyński
Konrad Wojtowicz
Maurycy Chronowski
Krzysztof Rataj
Magdalena Otrocka
Michał Mikula
Paula Feliksiak
Rafał Dziadziuszko
Tomasz Rzymski
Andrew Thomason
Krzysztof Brzózka
Andrzej Mazan
Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
Scientific Reports
title Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
title_full Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
title_fullStr Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
title_full_unstemmed Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
title_short Integrated transcriptomic and functional modeling reveals AKT and mTOR synergy in colorectal cancer
title_sort integrated transcriptomic and functional modeling reveals akt and mtor synergy in colorectal cancer
url https://doi.org/10.1038/s41598-025-08649-0
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