Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives

Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-one and benzo[<i>e</i>][1,3]thiazin-4-one derivatives, as significant sulfur- and nitrogen-containing heterocyclic compounds, are prevalent in natural products, pharmaceuticals, and food items. In recent years, a variety of i...

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Main Authors: Yongli He, Dan Yuan, Ke Yang, Bindong Li
Format: Article
Language:English
Published: MDPI AG 2025-05-01
Series:Molecules
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Online Access:https://www.mdpi.com/1420-3049/30/10/2099
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author Yongli He
Dan Yuan
Ke Yang
Bindong Li
author_facet Yongli He
Dan Yuan
Ke Yang
Bindong Li
author_sort Yongli He
collection DOAJ
description Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-one and benzo[<i>e</i>][1,3]thiazin-4-one derivatives, as significant sulfur- and nitrogen-containing heterocyclic compounds, are prevalent in natural products, pharmaceuticals, and food items. In recent years, a variety of innovative synthetic methodologies for these compounds have been developed. In this review, we will comprehensively introduce the major advances in the synthesis of benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-one and benzo[<i>e</i>][1,3]thiazin-4-one derivatives via both intramolecular and intermolecular pathways from 2012 to the present.
format Article
id doaj-art-ba55bb886b8d4964a412a9c0589303ce
institution OA Journals
issn 1420-3049
language English
publishDate 2025-05-01
publisher MDPI AG
record_format Article
series Molecules
spelling doaj-art-ba55bb886b8d4964a412a9c0589303ce2025-08-20T01:56:41ZengMDPI AGMolecules1420-30492025-05-013010209910.3390/molecules30102099Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One DerivativesYongli He0Dan Yuan1Ke Yang2Bindong Li3School of Chemistry and Chemical Engineering, Nanjing University of Science and Technology, Nanjing 210094, ChinaJiangsu Key Laboratory of Advanced Catalytic Materials & Technology, School of Petrochemical Engineering, Changzhou University, Changzhou 213164, ChinaJiangsu Key Laboratory of Advanced Catalytic Materials & Technology, School of Petrochemical Engineering, Changzhou University, Changzhou 213164, ChinaSchool of Chemistry and Chemical Engineering, Nanjing University of Science and Technology, Nanjing 210094, ChinaBenzo[<i>d</i>]isothiazol-3(2<i>H</i>)-one and benzo[<i>e</i>][1,3]thiazin-4-one derivatives, as significant sulfur- and nitrogen-containing heterocyclic compounds, are prevalent in natural products, pharmaceuticals, and food items. In recent years, a variety of innovative synthetic methodologies for these compounds have been developed. In this review, we will comprehensively introduce the major advances in the synthesis of benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-one and benzo[<i>e</i>][1,3]thiazin-4-one derivatives via both intramolecular and intermolecular pathways from 2012 to the present.https://www.mdpi.com/1420-3049/30/10/2099benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-onesbenzo[<i>e</i>][1,3]thiazin-4-onesorganic synthesis
spellingShingle Yongli He
Dan Yuan
Ke Yang
Bindong Li
Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
Molecules
benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-ones
benzo[<i>e</i>][1,3]thiazin-4-ones
organic synthesis
title Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
title_full Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
title_fullStr Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
title_full_unstemmed Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
title_short Recent Advances in the Synthesis of Benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-One and Benzo[<i>e</i>][1,3]Thiazin-4-One Derivatives
title_sort recent advances in the synthesis of benzo i d i isothiazol 3 2 i h i one and benzo i e i 1 3 thiazin 4 one derivatives
topic benzo[<i>d</i>]isothiazol-3(2<i>H</i>)-ones
benzo[<i>e</i>][1,3]thiazin-4-ones
organic synthesis
url https://www.mdpi.com/1420-3049/30/10/2099
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