Establishment and Evaluation of HepG2 Cell Insulin Resistance Model

Zixuan Meng,1 Yuehua Han,1 Linda Ruan,1 Chenming Xu,1 Mengxiao Zhang,1,2 Hao Liu1,2 1School of Pharmacy, Bengbu Medical University, Bengbu, People’s Republic of China; 2Anhui Province Engineering Technology Research Center of Biochemical Pharmaceutical, Bengbu, Anhui Province, People’s Republic of C...

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Main Authors: Meng Z, Han Y, Ruan L, Xu C, Zhang M, Liu H
Format: Article
Language:English
Published: Dove Medical Press 2025-07-01
Series:Diabetes, Metabolic Syndrome and Obesity
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Online Access:https://www.dovepress.com/establishment-and-evaluation-of-hepg2-cell-insulin-resistance-model-peer-reviewed-fulltext-article-DMSO
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author Meng Z
Han Y
Ruan L
Xu C
Zhang M
Liu H
author_facet Meng Z
Han Y
Ruan L
Xu C
Zhang M
Liu H
author_sort Meng Z
collection DOAJ
description Zixuan Meng,1 Yuehua Han,1 Linda Ruan,1 Chenming Xu,1 Mengxiao Zhang,1,2 Hao Liu1,2 1School of Pharmacy, Bengbu Medical University, Bengbu, People’s Republic of China; 2Anhui Province Engineering Technology Research Center of Biochemical Pharmaceutical, Bengbu, Anhui Province, People’s Republic of ChinaCorrespondence: Hao Liu, Email liuhao6886@bbmc.edu.cn Mengxiao Zhang, Email zhangmx@bbmc.edu.cnObjective: Establishing HepG2 cell insulin resistance models using glucosamine, high glucose with high insulin and palmitic acid and briefly evaluating them to provide reliable models for insulin resistance research.Methods: Three methods were used to induce insulin resistance in HepG2 cells, and glucose uptake and consumption, glucose metabolism-related mRNA and p-AKT/AKT protein levels and RNA-seq were detected to compare the three induction methods.Results: Glucose consumption capacity was reduced after glucosamine and palmitic acid induction and did not change significantly after high glucose with high insulin induction. Glucose uptake capacity was not significantly changed after glucosamine and high glucose with high insulin induction and was reduced after palmitic acid induction. After high insulin stimulation, p-AKT/AKT levels were elevated in glucosamine and high glucose with high insulin induction and did not change significantly in palmitic acid induction. G6pase, PC, and PCK1 were elevated after glucosamine and palmitic acid stimulation, and only PCK1 was elevated after high glucose with high insulin stimulation. The transcriptomes of cells induced by the three methods differed widely.Conclusion: Treatment with 0.2 mM palmitic acid for 24 h is a simple and stable method to induce insulin resistance in HepG2 cells.Keywords: HepG2 cells, insulin resistance model, palmitic acid
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publishDate 2025-07-01
publisher Dove Medical Press
record_format Article
series Diabetes, Metabolic Syndrome and Obesity
spelling doaj-art-b5ea48cd7cf34182b48ec4ec0f8af96a2025-08-20T03:31:33ZengDove Medical PressDiabetes, Metabolic Syndrome and Obesity1178-70072025-07-01Volume 18Issue 125732584105226Establishment and Evaluation of HepG2 Cell Insulin Resistance ModelMeng Z0Han YRuan L1Xu C2Zhang M3Liu H4college of pharmacycollege of pharmacycollege of pharmacySchool of PharmacyBengbu medical universityZixuan Meng,1 Yuehua Han,1 Linda Ruan,1 Chenming Xu,1 Mengxiao Zhang,1,2 Hao Liu1,2 1School of Pharmacy, Bengbu Medical University, Bengbu, People’s Republic of China; 2Anhui Province Engineering Technology Research Center of Biochemical Pharmaceutical, Bengbu, Anhui Province, People’s Republic of ChinaCorrespondence: Hao Liu, Email liuhao6886@bbmc.edu.cn Mengxiao Zhang, Email zhangmx@bbmc.edu.cnObjective: Establishing HepG2 cell insulin resistance models using glucosamine, high glucose with high insulin and palmitic acid and briefly evaluating them to provide reliable models for insulin resistance research.Methods: Three methods were used to induce insulin resistance in HepG2 cells, and glucose uptake and consumption, glucose metabolism-related mRNA and p-AKT/AKT protein levels and RNA-seq were detected to compare the three induction methods.Results: Glucose consumption capacity was reduced after glucosamine and palmitic acid induction and did not change significantly after high glucose with high insulin induction. Glucose uptake capacity was not significantly changed after glucosamine and high glucose with high insulin induction and was reduced after palmitic acid induction. After high insulin stimulation, p-AKT/AKT levels were elevated in glucosamine and high glucose with high insulin induction and did not change significantly in palmitic acid induction. G6pase, PC, and PCK1 were elevated after glucosamine and palmitic acid stimulation, and only PCK1 was elevated after high glucose with high insulin stimulation. The transcriptomes of cells induced by the three methods differed widely.Conclusion: Treatment with 0.2 mM palmitic acid for 24 h is a simple and stable method to induce insulin resistance in HepG2 cells.Keywords: HepG2 cells, insulin resistance model, palmitic acidhttps://www.dovepress.com/establishment-and-evaluation-of-hepg2-cell-insulin-resistance-model-peer-reviewed-fulltext-article-DMSOHepG2 cellsInsulin resistance modelPalmitic acid.
spellingShingle Meng Z
Han Y
Ruan L
Xu C
Zhang M
Liu H
Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
Diabetes, Metabolic Syndrome and Obesity
HepG2 cells
Insulin resistance model
Palmitic acid.
title Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
title_full Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
title_fullStr Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
title_full_unstemmed Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
title_short Establishment and Evaluation of HepG2 Cell Insulin Resistance Model
title_sort establishment and evaluation of hepg2 cell insulin resistance model
topic HepG2 cells
Insulin resistance model
Palmitic acid.
url https://www.dovepress.com/establishment-and-evaluation-of-hepg2-cell-insulin-resistance-model-peer-reviewed-fulltext-article-DMSO
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