Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations

Somatic activating mutations in PIK3CA are common drivers of vascular and lymphatic malformations. Despite common biophysical signatures of tissues susceptible to lesion formation, including compliant extracellular matrix and low rates of perfusion, lesions vary in clinical presentation from localiz...

Full description

Saved in:
Bibliographic Details
Main Authors: Wen Yih Aw, Aanya Sawhney, Mitesh Rathod, Chloe P. Whitworth, Elizabeth L. Doherty, Ethan Madden, Jingming Lu, Kaden Westphal, Ryan Stack, William J. Polacheck
Format: Article
Language:English
Published: AIP Publishing LLC 2025-03-01
Series:APL Bioengineering
Online Access:http://dx.doi.org/10.1063/5.0234507
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849739327046680576
author Wen Yih Aw
Aanya Sawhney
Mitesh Rathod
Chloe P. Whitworth
Elizabeth L. Doherty
Ethan Madden
Jingming Lu
Kaden Westphal
Ryan Stack
William J. Polacheck
author_facet Wen Yih Aw
Aanya Sawhney
Mitesh Rathod
Chloe P. Whitworth
Elizabeth L. Doherty
Ethan Madden
Jingming Lu
Kaden Westphal
Ryan Stack
William J. Polacheck
author_sort Wen Yih Aw
collection DOAJ
description Somatic activating mutations in PIK3CA are common drivers of vascular and lymphatic malformations. Despite common biophysical signatures of tissues susceptible to lesion formation, including compliant extracellular matrix and low rates of perfusion, lesions vary in clinical presentation from localized cystic dilatation to diffuse and infiltrative vascular dysplasia. The mechanisms driving the differences in disease severity and variability in clinical presentation and the role of the biophysical microenvironment in potentiating progression are poorly understood. Here, we investigate the role of hemodynamic forces and the biophysical microenvironment in the pathophysiology of vascular malformations (VMs), and we identify hemodynamic shear stress and defective endothelial cell mechanotransduction as key regulators of lesion progression. We found that constitutive PI3K activation impaired flow-mediated endothelial cell alignment and barrier function. We show that defective shear stress sensing in PIK3CAE542K endothelial cells is associated with reduced myosin light chain phosphorylation, junctional instability, and defective recruitment of vinculin to cell–cell junctions. Using three dimensional (3D) microfluidic models of the vasculature, we demonstrate that PIK3CAE542K microvessels apply reduced traction forces and are unaffected by flow interruption. We further found that draining transmural flow resulted in increased sprouting and invasion responses in PIK3CAE542K microvessels. Mechanistically, constitutive PI3K activation decreased cellular and nuclear elasticity resulting in defective cellular tensional homeostasis in endothelial cells which may underlie vascular dilation, tissue hyperplasia, and hypersprouting in PIK3CA-driven venous and lymphatic malformations. Together, these results suggest that defective nuclear mechanics, impaired cellular mechanotransduction, and maladaptive hemodynamic responses contribute to the development and progression of PIK3CA-driven vascular malformations.
format Article
id doaj-art-b42fcde7aba444d98db75feac8e275d2
institution DOAJ
issn 2473-2877
language English
publishDate 2025-03-01
publisher AIP Publishing LLC
record_format Article
series APL Bioengineering
spelling doaj-art-b42fcde7aba444d98db75feac8e275d22025-08-20T03:06:17ZengAIP Publishing LLCAPL Bioengineering2473-28772025-03-0191016106016106-2010.1063/5.0234507Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformationsWen Yih Aw0Aanya Sawhney1Mitesh Rathod2Chloe P. Whitworth3Elizabeth L. Doherty4Ethan Madden5Jingming Lu6Kaden Westphal7Ryan Stack8William J. Polacheck9 Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Department of Genetics and Molecular Biology, University of North Carolina at Chapel Hill School of Medicine, Chapel Hill, North Carolina 27599, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USA Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill and North Carolina State University, Chapel Hill, North Carolina 27514, USASomatic activating mutations in PIK3CA are common drivers of vascular and lymphatic malformations. Despite common biophysical signatures of tissues susceptible to lesion formation, including compliant extracellular matrix and low rates of perfusion, lesions vary in clinical presentation from localized cystic dilatation to diffuse and infiltrative vascular dysplasia. The mechanisms driving the differences in disease severity and variability in clinical presentation and the role of the biophysical microenvironment in potentiating progression are poorly understood. Here, we investigate the role of hemodynamic forces and the biophysical microenvironment in the pathophysiology of vascular malformations (VMs), and we identify hemodynamic shear stress and defective endothelial cell mechanotransduction as key regulators of lesion progression. We found that constitutive PI3K activation impaired flow-mediated endothelial cell alignment and barrier function. We show that defective shear stress sensing in PIK3CAE542K endothelial cells is associated with reduced myosin light chain phosphorylation, junctional instability, and defective recruitment of vinculin to cell–cell junctions. Using three dimensional (3D) microfluidic models of the vasculature, we demonstrate that PIK3CAE542K microvessels apply reduced traction forces and are unaffected by flow interruption. We further found that draining transmural flow resulted in increased sprouting and invasion responses in PIK3CAE542K microvessels. Mechanistically, constitutive PI3K activation decreased cellular and nuclear elasticity resulting in defective cellular tensional homeostasis in endothelial cells which may underlie vascular dilation, tissue hyperplasia, and hypersprouting in PIK3CA-driven venous and lymphatic malformations. Together, these results suggest that defective nuclear mechanics, impaired cellular mechanotransduction, and maladaptive hemodynamic responses contribute to the development and progression of PIK3CA-driven vascular malformations.http://dx.doi.org/10.1063/5.0234507
spellingShingle Wen Yih Aw
Aanya Sawhney
Mitesh Rathod
Chloe P. Whitworth
Elizabeth L. Doherty
Ethan Madden
Jingming Lu
Kaden Westphal
Ryan Stack
William J. Polacheck
Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
APL Bioengineering
title Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
title_full Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
title_fullStr Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
title_full_unstemmed Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
title_short Dysfunctional mechanotransduction regulates the progression of PIK3CA-driven vascular malformations
title_sort dysfunctional mechanotransduction regulates the progression of pik3ca driven vascular malformations
url http://dx.doi.org/10.1063/5.0234507
work_keys_str_mv AT wenyihaw dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT aanyasawhney dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT miteshrathod dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT chloepwhitworth dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT elizabethldoherty dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT ethanmadden dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT jingminglu dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT kadenwestphal dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT ryanstack dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations
AT williamjpolacheck dysfunctionalmechanotransductionregulatestheprogressionofpik3cadrivenvascularmalformations