Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology

AMP-activated protein kinase (AMPK) is a central regulator of cellular energy homeostasis, integrating metabolic, mitochondrial, and oxidative stress responses. In the heart, an organ with high and dynamically fluctuating energy demands, AMPK is essential for maintaining metabolic balance, particula...

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Main Authors: Ani Rakoubian, Julia Khinchin, Johnathan Yarbro, Satoru Kobayashi, Qiangrong Liang
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-08-01
Series:Frontiers in Cardiovascular Medicine
Subjects:
Online Access:https://www.frontiersin.org/articles/10.3389/fcvm.2025.1638515/full
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author Ani Rakoubian
Julia Khinchin
Johnathan Yarbro
Satoru Kobayashi
Qiangrong Liang
author_facet Ani Rakoubian
Julia Khinchin
Johnathan Yarbro
Satoru Kobayashi
Qiangrong Liang
author_sort Ani Rakoubian
collection DOAJ
description AMP-activated protein kinase (AMPK) is a central regulator of cellular energy homeostasis, integrating metabolic, mitochondrial, and oxidative stress responses. In the heart, an organ with high and dynamically fluctuating energy demands, AMPK is essential for maintaining metabolic balance, particularly during conditions such as exercise, ischemia, hypertrophy, and heart failure. The AMPK complex comprises a catalytic α subunit and regulatory β and γ subunits, each with multiple isoforms (α1, α2; β1, β2; γ1, γ2, γ3) that confer tissue-specific distribution and functional specialization. This review highlights the isoform-specific roles of AMPK in the heart, emphasizing their distinct contributions to myocardial energy metabolism, contractile function, and cardiac remodeling across diverse physiological and pathological conditions.
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institution Kabale University
issn 2297-055X
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publishDate 2025-08-01
publisher Frontiers Media S.A.
record_format Article
series Frontiers in Cardiovascular Medicine
spelling doaj-art-b1773bf22be34b6db60db174d7ba86bc2025-08-20T03:38:55ZengFrontiers Media S.A.Frontiers in Cardiovascular Medicine2297-055X2025-08-011210.3389/fcvm.2025.16385151638515Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiologyAni RakoubianJulia KhinchinJohnathan YarbroSatoru KobayashiQiangrong LiangAMP-activated protein kinase (AMPK) is a central regulator of cellular energy homeostasis, integrating metabolic, mitochondrial, and oxidative stress responses. In the heart, an organ with high and dynamically fluctuating energy demands, AMPK is essential for maintaining metabolic balance, particularly during conditions such as exercise, ischemia, hypertrophy, and heart failure. The AMPK complex comprises a catalytic α subunit and regulatory β and γ subunits, each with multiple isoforms (α1, α2; β1, β2; γ1, γ2, γ3) that confer tissue-specific distribution and functional specialization. This review highlights the isoform-specific roles of AMPK in the heart, emphasizing their distinct contributions to myocardial energy metabolism, contractile function, and cardiac remodeling across diverse physiological and pathological conditions.https://www.frontiersin.org/articles/10.3389/fcvm.2025.1638515/fullAMPKisoform-specificenergy metabolismmitochondria quality controlcardiac remodeling
spellingShingle Ani Rakoubian
Julia Khinchin
Johnathan Yarbro
Satoru Kobayashi
Qiangrong Liang
Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
Frontiers in Cardiovascular Medicine
AMPK
isoform-specific
energy metabolism
mitochondria quality control
cardiac remodeling
title Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
title_full Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
title_fullStr Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
title_full_unstemmed Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
title_short Isoform-specific roles of AMP-activated protein kinase in cardiac physiology and pathophysiology
title_sort isoform specific roles of amp activated protein kinase in cardiac physiology and pathophysiology
topic AMPK
isoform-specific
energy metabolism
mitochondria quality control
cardiac remodeling
url https://www.frontiersin.org/articles/10.3389/fcvm.2025.1638515/full
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AT satorukobayashi isoformspecificrolesofampactivatedproteinkinaseincardiacphysiologyandpathophysiology
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