Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo

Acute lung injury (ALI) is a clinical syndrome characterized by excessive inflammatory responses. Despite the exploration of various therapeutic approaches, no effective pharmacological treatment is currently available for ALI. In the current study, we investigated the role of SIRT3 in LPS-induced A...

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Main Authors: Jian Chen, Yang Cai, Xiaochun Peng, Yuanling Xu, Liying Chen, Xinxin Pan, Yingying Sun
Format: Article
Language:English
Published: Frontiers Media S.A. 2025-06-01
Series:Frontiers in Pharmacology
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Online Access:https://www.frontiersin.org/articles/10.3389/fphar.2025.1524219/full
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author Jian Chen
Jian Chen
Jian Chen
Yang Cai
Yang Cai
Yang Cai
Xiaochun Peng
Xiaochun Peng
Xiaochun Peng
Yuanling Xu
Yuanling Xu
Yuanling Xu
Liying Chen
Liying Chen
Liying Chen
Xinxin Pan
Xinxin Pan
Xinxin Pan
Yingying Sun
Yingying Sun
Yingying Sun
author_facet Jian Chen
Jian Chen
Jian Chen
Yang Cai
Yang Cai
Yang Cai
Xiaochun Peng
Xiaochun Peng
Xiaochun Peng
Yuanling Xu
Yuanling Xu
Yuanling Xu
Liying Chen
Liying Chen
Liying Chen
Xinxin Pan
Xinxin Pan
Xinxin Pan
Yingying Sun
Yingying Sun
Yingying Sun
author_sort Jian Chen
collection DOAJ
description Acute lung injury (ALI) is a clinical syndrome characterized by excessive inflammatory responses. Despite the exploration of various therapeutic approaches, no effective pharmacological treatment is currently available for ALI. In the current study, we investigated the role of SIRT3 in LPS-induced ALI and the potential protective effects of dexmedetomidine (Dex), an agent that activates α2-adrenergic receptors. Histological analysis showed extensive lung damage and increased inflammatory cells in LPS-treated lung samples, with elevated TUNEL+ cells indicating apoptosis (p < 0.05). SIRT3 mRNA and protein expression were significantly downregulated following LPS treatment, both in vivo and in vitro (p < 0.05). DEX administration restored protein SIRT3 levels and reduced inflammation, while the SIRT3 inhibitor 3-TYP negated these benefits (p < 0.05). Additionally, DEX reduced pro-inflammatory cytokine levels and oxidative stress, effects that were also diminished by 3-TYP (p < 0.05). Our findings suggest that DEX exerts its protective effects against LPS-induced ALI via modulation of the SIRT3/LKB1/AMPK signaling pathway, highlighting the critical role of SIRT3 in inflammatory and oxidative stress responses in ALI.
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issn 1663-9812
language English
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publisher Frontiers Media S.A.
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series Frontiers in Pharmacology
spelling doaj-art-a80149615246482491d77f61b33de5b22025-08-20T03:32:23ZengFrontiers Media S.A.Frontiers in Pharmacology1663-98122025-06-011610.3389/fphar.2025.15242191524219Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivoJian Chen0Jian Chen1Jian Chen2Yang Cai3Yang Cai4Yang Cai5Xiaochun Peng6Xiaochun Peng7Xiaochun Peng8Yuanling Xu9Yuanling Xu10Yuanling Xu11Liying Chen12Liying Chen13Liying Chen14Xinxin Pan15Xinxin Pan16Xinxin Pan17Yingying Sun18Yingying Sun19Yingying Sun20Department of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaDepartment of Anesthesiology, Anhui Provincial children’s Hospital, Anhui, ChinaThe Fifth Clinical Medical College of Anhui Medical University, Anhui, ChinaThe Children’s Medical Center of Anhui Medical University, Anhui, ChinaAcute lung injury (ALI) is a clinical syndrome characterized by excessive inflammatory responses. Despite the exploration of various therapeutic approaches, no effective pharmacological treatment is currently available for ALI. In the current study, we investigated the role of SIRT3 in LPS-induced ALI and the potential protective effects of dexmedetomidine (Dex), an agent that activates α2-adrenergic receptors. Histological analysis showed extensive lung damage and increased inflammatory cells in LPS-treated lung samples, with elevated TUNEL+ cells indicating apoptosis (p < 0.05). SIRT3 mRNA and protein expression were significantly downregulated following LPS treatment, both in vivo and in vitro (p < 0.05). DEX administration restored protein SIRT3 levels and reduced inflammation, while the SIRT3 inhibitor 3-TYP negated these benefits (p < 0.05). Additionally, DEX reduced pro-inflammatory cytokine levels and oxidative stress, effects that were also diminished by 3-TYP (p < 0.05). Our findings suggest that DEX exerts its protective effects against LPS-induced ALI via modulation of the SIRT3/LKB1/AMPK signaling pathway, highlighting the critical role of SIRT3 in inflammatory and oxidative stress responses in ALI.https://www.frontiersin.org/articles/10.3389/fphar.2025.1524219/fullacute lung injurysirt3dexmedetomidineinflammationoxidative stress
spellingShingle Jian Chen
Jian Chen
Jian Chen
Yang Cai
Yang Cai
Yang Cai
Xiaochun Peng
Xiaochun Peng
Xiaochun Peng
Yuanling Xu
Yuanling Xu
Yuanling Xu
Liying Chen
Liying Chen
Liying Chen
Xinxin Pan
Xinxin Pan
Xinxin Pan
Yingying Sun
Yingying Sun
Yingying Sun
Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
Frontiers in Pharmacology
acute lung injury
sirt3
dexmedetomidine
inflammation
oxidative stress
title Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
title_full Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
title_fullStr Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
title_full_unstemmed Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
title_short Dexmedetomidine reduces acute lung injury caused by LPS through the SIRT3 signaling pathway in vivo
title_sort dexmedetomidine reduces acute lung injury caused by lps through the sirt3 signaling pathway in vivo
topic acute lung injury
sirt3
dexmedetomidine
inflammation
oxidative stress
url https://www.frontiersin.org/articles/10.3389/fphar.2025.1524219/full
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