Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI

Abstract Third-generation epidermal growth factor receptor-tyrosine kinase inhibitors (EGFR-TKIs) are the latest and a vital treatment option for non-small cell lung cancer (NSCLC) patients. Although EGFR-sensitive mutations are an indication for third-generation EGFR-TKI therapy, 30% of NSCLC patie...

Full description

Saved in:
Bibliographic Details
Main Authors: Ning Lou, Ruyun Gao, Yuankai Shi, Xiaohong Han
Format: Article
Language:English
Published: Nature Portfolio 2024-12-01
Series:Scientific Data
Online Access:https://doi.org/10.1038/s41597-024-04169-0
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1850244528725819392
author Ning Lou
Ruyun Gao
Yuankai Shi
Xiaohong Han
author_facet Ning Lou
Ruyun Gao
Yuankai Shi
Xiaohong Han
author_sort Ning Lou
collection DOAJ
description Abstract Third-generation epidermal growth factor receptor-tyrosine kinase inhibitors (EGFR-TKIs) are the latest and a vital treatment option for non-small cell lung cancer (NSCLC) patients. Although EGFR-sensitive mutations are an indication for third-generation EGFR-TKI therapy, 30% of NSCLC patients lack response and all patients inevitably progress. There is a lack of biomarkers to predict the efficacy of EGFR-TKI therapy. In this report, we performed comprehensive plasma metabolomic profiling on 186 baseline and 20 post-treatment samples, analyzing 1,019 metabolites using four ultrahigh performance liquid chromatography-tandem mass spectroscopy (UPLC-MS/MS) methods. The dataset contains detailed clinical and metabolic information for 186 patients. Rigorous quality control measures were implemented. No significant differences in body mass index and biochemical metabolic parameters were observed between responders and non-responders. The datasets were utilized to characterize the responsive metabolic traits of third-generation EGFR-TKI therapy. All datasets are available for download on the OMIX website. We anticipate that these datasets will serve as valuable resources for future studies investigating NSCLC metabolism and for the development of personalized therapeutic strategies.
format Article
id doaj-art-a7444eef336e47c49daa474401304eda
institution OA Journals
issn 2052-4463
language English
publishDate 2024-12-01
publisher Nature Portfolio
record_format Article
series Scientific Data
spelling doaj-art-a7444eef336e47c49daa474401304eda2025-08-20T01:59:43ZengNature PortfolioScientific Data2052-44632024-12-011111710.1038/s41597-024-04169-0Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKINing Lou0Ruyun Gao1Yuankai Shi2Xiaohong Han3Clinical Pharmacology Research Center, Peking Union Medical College Hospital, State Key Laboratory of Complex Severe and Rare Diseases, NMPA Key Laboratory for Clinical Research and Evaluation of Drug, Beijing Key Laboratory of Clinical PK & PD Investigation for Innovative Drugs, Chinese Academy of Medical Sciences & Peking Union Medical College; No.1, Shuaifuyuan, Dongcheng DistrictDepartment of Medical Oncology, National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital, Chinese Academy of Medical Sciences & Peking Union Medical College, Beijing Key Laboratory of Clinical Study on Anticancer Molecular Targeted Drugs; No. 17 Panjiayuan Nanli, Chaoyang DistrictDepartment of Medical Oncology, National Cancer Center/National Clinical Research Center for Cancer/Cancer Hospital, Chinese Academy of Medical Sciences & Peking Union Medical College, Beijing Key Laboratory of Clinical Study on Anticancer Molecular Targeted Drugs; No. 17 Panjiayuan Nanli, Chaoyang DistrictClinical Pharmacology Research Center, Peking Union Medical College Hospital, State Key Laboratory of Complex Severe and Rare Diseases, NMPA Key Laboratory for Clinical Research and Evaluation of Drug, Beijing Key Laboratory of Clinical PK & PD Investigation for Innovative Drugs, Chinese Academy of Medical Sciences & Peking Union Medical College; No.1, Shuaifuyuan, Dongcheng DistrictAbstract Third-generation epidermal growth factor receptor-tyrosine kinase inhibitors (EGFR-TKIs) are the latest and a vital treatment option for non-small cell lung cancer (NSCLC) patients. Although EGFR-sensitive mutations are an indication for third-generation EGFR-TKI therapy, 30% of NSCLC patients lack response and all patients inevitably progress. There is a lack of biomarkers to predict the efficacy of EGFR-TKI therapy. In this report, we performed comprehensive plasma metabolomic profiling on 186 baseline and 20 post-treatment samples, analyzing 1,019 metabolites using four ultrahigh performance liquid chromatography-tandem mass spectroscopy (UPLC-MS/MS) methods. The dataset contains detailed clinical and metabolic information for 186 patients. Rigorous quality control measures were implemented. No significant differences in body mass index and biochemical metabolic parameters were observed between responders and non-responders. The datasets were utilized to characterize the responsive metabolic traits of third-generation EGFR-TKI therapy. All datasets are available for download on the OMIX website. We anticipate that these datasets will serve as valuable resources for future studies investigating NSCLC metabolism and for the development of personalized therapeutic strategies.https://doi.org/10.1038/s41597-024-04169-0
spellingShingle Ning Lou
Ruyun Gao
Yuankai Shi
Xiaohong Han
Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
Scientific Data
title Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
title_full Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
title_fullStr Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
title_full_unstemmed Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
title_short Plasma metabolomics profiling of EGFR-mutant NSCLC patients treated with third-generation EGFR-TKI
title_sort plasma metabolomics profiling of egfr mutant nsclc patients treated with third generation egfr tki
url https://doi.org/10.1038/s41597-024-04169-0
work_keys_str_mv AT ninglou plasmametabolomicsprofilingofegfrmutantnsclcpatientstreatedwiththirdgenerationegfrtki
AT ruyungao plasmametabolomicsprofilingofegfrmutantnsclcpatientstreatedwiththirdgenerationegfrtki
AT yuankaishi plasmametabolomicsprofilingofegfrmutantnsclcpatientstreatedwiththirdgenerationegfrtki
AT xiaohonghan plasmametabolomicsprofilingofegfrmutantnsclcpatientstreatedwiththirdgenerationegfrtki