Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer

Halal hard shell capsules are importantly needed by Indonesian consumers, who are predominantly Muslim, to substitute mostly used and commercially available products made from non-halal ingredients such as gelatin. The objective of this study is to prepare, characterize, and evaluate halal hard shel...

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Main Authors: Tri Susanti, Siti Wafiroh, Esti Hendradi, Pratiwi Pudjiastuti
Format: Article
Language:English
Published: Universitas Airlangga 2020-06-01
Series:Journal of Halal Product and Research
Subjects:
Online Access:https://e-journal.unair.ac.id/JHPR/article/view/19586
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author Tri Susanti
Siti Wafiroh
Esti Hendradi
Pratiwi Pudjiastuti
author_facet Tri Susanti
Siti Wafiroh
Esti Hendradi
Pratiwi Pudjiastuti
author_sort Tri Susanti
collection DOAJ
description Halal hard shell capsules are importantly needed by Indonesian consumers, who are predominantly Muslim, to substitute mostly used and commercially available products made from non-halal ingredients such as gelatin. The objective of this study is to prepare, characterize, and evaluate halal hard shell capsules made from k-carrageenan-xanthan gum with sorbitol as the plasticizer with diclofenac sodium as the model drug. Hardshell capsules were prepared with combinations of κ-carrageenan-xanthan gum at a weight ratio of 4:2 with the addition of 70% sorbitol, which added at a varied volume of 0.25; 0.50; 0.75; and 1.00 mL. Characterization of halal hard shell capsules includes swelling degree, tensile strength, Fourier Transformed Infrared (FTIR) and Scanning Electron Microscope (SEM), as well as disintegration test. The diclofenac sodium profile release was evaluated through the dissolution test at pH 6.8. The best physical characteristics were obtained by preparing capsule shells with a mixture of carrageenan-xanthan gum at a weight ratio of 4:2 with the addition of 0.25 mL sorbitol. The evaluation of Halal hard shell capsules showed that it had a swelling rate of 3.46% in water media, stress modulus of 28.6 MPa, strain modulus of 4.3 MPa, and modulus young of 362,3%, as well as disintegration time of capsules, was 51.8 minutes at pH 6.8. The dissolution test showed that diclofenac sodium was released at a level of 2.7% for 16 minutes. Based on this data, it can be concluded that the Halal hard shell capsule of κ-carrageenan-xanthan gum with the addition of sorbitol can be used as an alternative for the gelatin capsule with more controlled release.
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spelling doaj-art-a5d4aa9f759a4e6e904bb25978e5fc982025-08-20T02:36:38ZengUniversitas AirlanggaJournal of Halal Product and Research2654-94092654-97782020-06-01311810.20473/jhpr.vol.3-issue.1.1-816001Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizerTri Susanti0Siti Wafiroh1Esti Hendradi2Pratiwi Pudjiastuti3Departemen Kimia, Fakultas Sains danTeknologi,Universitas Airlangga, Surabaya, IndonesiaDepartemen Kimia, Fakultas Sains danTeknologi,Universitas Airlangga, Surabaya, IndonesiaDepartemen Farmasetika, Fakultas Farmasi, Universitas Airlangga, Surabaya, IndonesiaDepartemen Kimia, Fakultas Sains danTeknologi,Universitas Airlangga, Surabaya, IndonesiaHalal hard shell capsules are importantly needed by Indonesian consumers, who are predominantly Muslim, to substitute mostly used and commercially available products made from non-halal ingredients such as gelatin. The objective of this study is to prepare, characterize, and evaluate halal hard shell capsules made from k-carrageenan-xanthan gum with sorbitol as the plasticizer with diclofenac sodium as the model drug. Hardshell capsules were prepared with combinations of κ-carrageenan-xanthan gum at a weight ratio of 4:2 with the addition of 70% sorbitol, which added at a varied volume of 0.25; 0.50; 0.75; and 1.00 mL. Characterization of halal hard shell capsules includes swelling degree, tensile strength, Fourier Transformed Infrared (FTIR) and Scanning Electron Microscope (SEM), as well as disintegration test. The diclofenac sodium profile release was evaluated through the dissolution test at pH 6.8. The best physical characteristics were obtained by preparing capsule shells with a mixture of carrageenan-xanthan gum at a weight ratio of 4:2 with the addition of 0.25 mL sorbitol. The evaluation of Halal hard shell capsules showed that it had a swelling rate of 3.46% in water media, stress modulus of 28.6 MPa, strain modulus of 4.3 MPa, and modulus young of 362,3%, as well as disintegration time of capsules, was 51.8 minutes at pH 6.8. The dissolution test showed that diclofenac sodium was released at a level of 2.7% for 16 minutes. Based on this data, it can be concluded that the Halal hard shell capsule of κ-carrageenan-xanthan gum with the addition of sorbitol can be used as an alternative for the gelatin capsule with more controlled release.https://e-journal.unair.ac.id/JHPR/article/view/19586characterizationdiclofenac sodiumrelease profileîº-carrageenan-xanthan gumhalal hardhell capsule
spellingShingle Tri Susanti
Siti Wafiroh
Esti Hendradi
Pratiwi Pudjiastuti
Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
Journal of Halal Product and Research
characterization
diclofenac sodium
release profile
îº-carrageenan-xanthan gum
halal hardhell capsule
title Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
title_full Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
title_fullStr Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
title_full_unstemmed Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
title_short Characterization and release profile of sodium diclofenac halal hard shell capsules made from k-carrageenan and xanthan gum with sorbitol plasticizer
title_sort characterization and release profile of sodium diclofenac halal hard shell capsules made from k carrageenan and xanthan gum with sorbitol plasticizer
topic characterization
diclofenac sodium
release profile
îº-carrageenan-xanthan gum
halal hardhell capsule
url https://e-journal.unair.ac.id/JHPR/article/view/19586
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AT sitiwafiroh characterizationandreleaseprofileofsodiumdiclofenachalalhardshellcapsulesmadefromkcarrageenanandxanthangumwithsorbitolplasticizer
AT estihendradi characterizationandreleaseprofileofsodiumdiclofenachalalhardshellcapsulesmadefromkcarrageenanandxanthangumwithsorbitolplasticizer
AT pratiwipudjiastuti characterizationandreleaseprofileofsodiumdiclofenachalalhardshellcapsulesmadefromkcarrageenanandxanthangumwithsorbitolplasticizer