Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting

The Philippines has a high diversity of venomous snake species, but there is minimal information on their envenomation effects. This is evidenced by the small number of case reports, the poor reporting of envenomation cases, and the absence of specific antivenoms apart from one against the Philippin...

Full description

Saved in:
Bibliographic Details
Main Authors: Daniel Albert E. Castillo, Lorenzo Seneci, Abhinandan Chowdhury, Marilyn G. Rimando, Bryan G. Fry
Format: Article
Language:English
Published: MDPI AG 2025-04-01
Series:Toxins
Subjects:
Online Access:https://www.mdpi.com/2072-6651/17/4/185
Tags: Add Tag
No Tags, Be the first to tag this record!
_version_ 1849714040430919680
author Daniel Albert E. Castillo
Lorenzo Seneci
Abhinandan Chowdhury
Marilyn G. Rimando
Bryan G. Fry
author_facet Daniel Albert E. Castillo
Lorenzo Seneci
Abhinandan Chowdhury
Marilyn G. Rimando
Bryan G. Fry
author_sort Daniel Albert E. Castillo
collection DOAJ
description The Philippines has a high diversity of venomous snake species, but there is minimal information on their envenomation effects. This is evidenced by the small number of case reports, the poor reporting of envenomation cases, and the absence of specific antivenoms apart from one against the Philippine cobra (<i>Naja philippinensis</i>). This study sought to profile the action of selected Philippine pit viper venoms on blood coagulation and to investigate whether commercially available non-specific antivenoms can provide adequate protection against these venoms. Venom from the pit vipers <i>Trimeresurus flavomaculatus</i> and <i>Trimeresurus mcgregori</i> were subjected to coagulation assays, antivenom cross-neutralization tests, and thromboelastography. Venoms from both species were able to clot human plasma and isolated human fibrinogen. Consistent with pseudo-procoagulant/thrombin-like activity, the resulting fibrin clots were weak and transient, thereby contributing to net anticoagulation through the depletion of fibrinogen levels. Clotting factors fIXa and fXa were also inhibited by the venoms, further contributing to the net anticoagulant activity. Monovalent and polyvalent antivenoms from the Thai Red Cross Society were effective against both venoms, indicating cross-neutralization of venom toxins; the polyvalent antivenom was able to rescue fibrinogen clotting to a greater degree than the monovalent antivenom. Our findings highlight the coagulopathic effects of these pit viper venoms and suggest the utility of procuring the non-specific antivenoms for areas in the Philippines with a high risk for pit viper envenomation.
format Article
id doaj-art-a5669ebc85e64116aa33decccdcfe80e
institution DOAJ
issn 2072-6651
language English
publishDate 2025-04-01
publisher MDPI AG
record_format Article
series Toxins
spelling doaj-art-a5669ebc85e64116aa33decccdcfe80e2025-08-20T03:13:48ZengMDPI AGToxins2072-66512025-04-0117418510.3390/toxins17040185Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood ClottingDaniel Albert E. Castillo0Lorenzo Seneci1Abhinandan Chowdhury2Marilyn G. Rimando3Bryan G. Fry4The Graduate School, University of Santo Tomas, España Boulevard, Manila 1008, PhilippinesAdaptive Biotoxicology Lab, School of the Environment, University of Queensland, St Lucia 4072, AustraliaAdaptive Biotoxicology Lab, School of the Environment, University of Queensland, St Lucia 4072, AustraliaThe Graduate School, University of Santo Tomas, España Boulevard, Manila 1008, PhilippinesAdaptive Biotoxicology Lab, School of the Environment, University of Queensland, St Lucia 4072, AustraliaThe Philippines has a high diversity of venomous snake species, but there is minimal information on their envenomation effects. This is evidenced by the small number of case reports, the poor reporting of envenomation cases, and the absence of specific antivenoms apart from one against the Philippine cobra (<i>Naja philippinensis</i>). This study sought to profile the action of selected Philippine pit viper venoms on blood coagulation and to investigate whether commercially available non-specific antivenoms can provide adequate protection against these venoms. Venom from the pit vipers <i>Trimeresurus flavomaculatus</i> and <i>Trimeresurus mcgregori</i> were subjected to coagulation assays, antivenom cross-neutralization tests, and thromboelastography. Venoms from both species were able to clot human plasma and isolated human fibrinogen. Consistent with pseudo-procoagulant/thrombin-like activity, the resulting fibrin clots were weak and transient, thereby contributing to net anticoagulation through the depletion of fibrinogen levels. Clotting factors fIXa and fXa were also inhibited by the venoms, further contributing to the net anticoagulant activity. Monovalent and polyvalent antivenoms from the Thai Red Cross Society were effective against both venoms, indicating cross-neutralization of venom toxins; the polyvalent antivenom was able to rescue fibrinogen clotting to a greater degree than the monovalent antivenom. Our findings highlight the coagulopathic effects of these pit viper venoms and suggest the utility of procuring the non-specific antivenoms for areas in the Philippines with a high risk for pit viper envenomation.https://www.mdpi.com/2072-6651/17/4/185<i>Trimeresurus</i>coagulotoxicityantivenompseudo-procoagulantfibrinogen
spellingShingle Daniel Albert E. Castillo
Lorenzo Seneci
Abhinandan Chowdhury
Marilyn G. Rimando
Bryan G. Fry
Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
Toxins
<i>Trimeresurus</i>
coagulotoxicity
antivenom
pseudo-procoagulant
fibrinogen
title Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
title_full Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
title_fullStr Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
title_full_unstemmed Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
title_short Bite First, Bleed Later: How Philippine <i>Trimeresurus</i> Pit Viper Venoms Hijack Blood Clotting
title_sort bite first bleed later how philippine i trimeresurus i pit viper venoms hijack blood clotting
topic <i>Trimeresurus</i>
coagulotoxicity
antivenom
pseudo-procoagulant
fibrinogen
url https://www.mdpi.com/2072-6651/17/4/185
work_keys_str_mv AT danielalbertecastillo bitefirstbleedlaterhowphilippineitrimeresurusipitvipervenomshijackbloodclotting
AT lorenzoseneci bitefirstbleedlaterhowphilippineitrimeresurusipitvipervenomshijackbloodclotting
AT abhinandanchowdhury bitefirstbleedlaterhowphilippineitrimeresurusipitvipervenomshijackbloodclotting
AT marilyngrimando bitefirstbleedlaterhowphilippineitrimeresurusipitvipervenomshijackbloodclotting
AT bryangfry bitefirstbleedlaterhowphilippineitrimeresurusipitvipervenomshijackbloodclotting