Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication

The escalating prevalence of clarithromycin resistance in cases of Helicobacter pylori, insufficient acid suppression, and pharmacodynamic variations secondary to inter-individual differences in CYP2C19 polymorphism collectively contribute to suboptimal eradication rates observed with proton pump in...

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Main Authors: Byeong Yun Ahn, Soo-Jeong Cho
Format: Article
Language:English
Published: Korean College of Helicobacter and Upper Gastrointestinal Research 2023-09-01
Series:The Korean Journal of Helicobacter and Upper Gastrointestinal Research
Subjects:
Online Access:http://www.helicojournal.org/upload/pdf/kjhugr-2023-0041.pdf
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author Byeong Yun Ahn
Soo-Jeong Cho
author_facet Byeong Yun Ahn
Soo-Jeong Cho
author_sort Byeong Yun Ahn
collection DOAJ
description The escalating prevalence of clarithromycin resistance in cases of Helicobacter pylori, insufficient acid suppression, and pharmacodynamic variations secondary to inter-individual differences in CYP2C19 polymorphism collectively contribute to suboptimal eradication rates observed with proton pump inhibitor (PPI)-based therapy. Compared with PPIs, potassium-competitive acid blockers (PCABs) produce rapid, potent, and long-lasting suppression of gastric acid through reversible inhibition of gastric H+, K+-ATPase. PCAB-based therapy results in significant inhibition of acid secretion and has therefore emerged as a novel and effective approach for H. pylori eradication. In this study, we review the efficacy and safety profile of PCAB-based eradication regimens comprising vonoprazan, tegoprazan, and fexuprazan.
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institution Kabale University
issn 1738-3331
language English
publishDate 2023-09-01
publisher Korean College of Helicobacter and Upper Gastrointestinal Research
record_format Article
series The Korean Journal of Helicobacter and Upper Gastrointestinal Research
spelling doaj-art-a29f4f1171df4405b9652e7f8ffc7e4a2025-08-20T03:35:50ZengKorean College of Helicobacter and Upper Gastrointestinal ResearchThe Korean Journal of Helicobacter and Upper Gastrointestinal Research1738-33312023-09-0123317417910.7704/kjhugr.2023.0041790Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori EradicationByeong Yun Ahn0Soo-Jeong Cho1Department of Internal Medicine and Liver Research Institute, Seoul National University Hospital, Seoul National University College of Medicine, Seoul, KoreaDepartment of Internal Medicine and Liver Research Institute, Seoul National University Hospital, Seoul National University College of Medicine, Seoul, KoreaThe escalating prevalence of clarithromycin resistance in cases of Helicobacter pylori, insufficient acid suppression, and pharmacodynamic variations secondary to inter-individual differences in CYP2C19 polymorphism collectively contribute to suboptimal eradication rates observed with proton pump inhibitor (PPI)-based therapy. Compared with PPIs, potassium-competitive acid blockers (PCABs) produce rapid, potent, and long-lasting suppression of gastric acid through reversible inhibition of gastric H+, K+-ATPase. PCAB-based therapy results in significant inhibition of acid secretion and has therefore emerged as a novel and effective approach for H. pylori eradication. In this study, we review the efficacy and safety profile of PCAB-based eradication regimens comprising vonoprazan, tegoprazan, and fexuprazan.http://www.helicojournal.org/upload/pdf/kjhugr-2023-0041.pdfdrug resistance, microbialdrug therapygastric acid proton pump inhibitors
spellingShingle Byeong Yun Ahn
Soo-Jeong Cho
Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
The Korean Journal of Helicobacter and Upper Gastrointestinal Research
drug resistance, microbial
drug therapy
gastric acid

proton pump inhibitors
title Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
title_full Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
title_fullStr Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
title_full_unstemmed Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
title_short Potassium-competitive Acid Blockers: A New Therapeutic Strategy for Helicobacter pylori Eradication
title_sort potassium competitive acid blockers a new therapeutic strategy for helicobacter pylori eradication
topic drug resistance, microbial
drug therapy
gastric acid

proton pump inhibitors
url http://www.helicojournal.org/upload/pdf/kjhugr-2023-0041.pdf
work_keys_str_mv AT byeongyunahn potassiumcompetitiveacidblockersanewtherapeuticstrategyforhelicobacterpylorieradication
AT soojeongcho potassiumcompetitiveacidblockersanewtherapeuticstrategyforhelicobacterpylorieradication